UY33210A - DERIVADOS DE PIRAZOLO-[5, 1b]-OXAZOL COMO ANTAGONISTAS DE LOS RECEPTORES DE CRF-1 - Google Patents

DERIVADOS DE PIRAZOLO-[5, 1b]-OXAZOL COMO ANTAGONISTAS DE LOS RECEPTORES DE CRF-1

Info

Publication number
UY33210A
UY33210A UY0001033210A UY33210A UY33210A UY 33210 A UY33210 A UY 33210A UY 0001033210 A UY0001033210 A UY 0001033210A UY 33210 A UY33210 A UY 33210A UY 33210 A UY33210 A UY 33210A
Authority
UY
Uruguay
Prior art keywords
antagonists
derivatives
pirazolo
crf
oxazol
Prior art date
Application number
UY0001033210A
Other languages
English (en)
Inventor
Nicholas James Devereux
Mckenna Jeffrey
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of UY33210A publication Critical patent/UY33210A/es

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    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
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Abstract

Se describen derivados de 4-difluoro-metoxi-fenil-pirazolo-[5.1- b]-oxazol útiles como antagonistas de los receptores del factor de liberación de co rticotropina (CRF1).
UY0001033210A 2010-02-01 2011-01-31 DERIVADOS DE PIRAZOLO-[5, 1b]-OXAZOL COMO ANTAGONISTAS DE LOS RECEPTORES DE CRF-1 UY33210A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30023110P 2010-02-01 2010-02-01

Publications (1)

Publication Number Publication Date
UY33210A true UY33210A (es) 2011-08-31

Family

ID=43641912

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001033210A UY33210A (es) 2010-02-01 2011-01-31 DERIVADOS DE PIRAZOLO-[5, 1b]-OXAZOL COMO ANTAGONISTAS DE LOS RECEPTORES DE CRF-1

Country Status (8)

Country Link
US (2) US20120295942A1 (es)
EP (1) EP2531510B1 (es)
JP (1) JP2013518085A (es)
CN (1) CN102762572A (es)
AR (1) AR080055A1 (es)
TW (1) TW201130853A (es)
UY (1) UY33210A (es)
WO (1) WO2011092290A1 (es)

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