AR056729A1 - Compuesto de benzofurano carboxamida, composicion farmaceutica que lo comprende su uso para preparar un medicamento y procesos para su preparcion - Google Patents
Compuesto de benzofurano carboxamida, composicion farmaceutica que lo comprende su uso para preparar un medicamento y procesos para su preparcionInfo
- Publication number
- AR056729A1 AR056729A1 ARP060104683A ARP060104683A AR056729A1 AR 056729 A1 AR056729 A1 AR 056729A1 AR P060104683 A ARP060104683 A AR P060104683A AR P060104683 A ARP060104683 A AR P060104683A AR 056729 A1 AR056729 A1 AR 056729A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- processes
- pharmaceutical composition
- benzofuran
- prepare
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Un compuesto 4-amino-5-cloro-N-{[1-(tetrahidro-2H-piran-4-ilmetil]metil}-1-benzofuran-7-carboxamida (A), o una de sus sales farmacéuticamente aceptables, por ejemplo hidrocloruro, tosilato como monohidrato o anhidrato. Composicion farmacéutica que lo comprende. Su uso para la preparacion de un medicamento util para el tratamiento de enfermedades tratables mediante agonismo de 5-HT4. Procesos para su preparacion a partir de 4-amino-5-cloro-N-(4-piperidinilmetil)-1-benzofuran-7-carboxamida y tetrahidro-2H-piran-4-carbaldehído o de ácido 4-amino-5-cloro-1-benzofuran-7-carboxílico y {[1-(tetrahídro-2H-piranilmetil)-4-piperidinil]metil}amina.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0522071A GB0522071D0 (en) | 2005-10-28 | 2005-10-28 | Novel compound |
| GB0619950A GB0619950D0 (en) | 2006-10-09 | 2006-10-09 | Novel compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR056729A1 true AR056729A1 (es) | 2007-10-17 |
Family
ID=37591731
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP060104683A AR056729A1 (es) | 2005-10-28 | 2006-10-26 | Compuesto de benzofurano carboxamida, composicion farmaceutica que lo comprende su uso para preparar un medicamento y procesos para su preparcion |
Country Status (4)
| Country | Link |
|---|---|
| AR (1) | AR056729A1 (es) |
| PE (1) | PE20070713A1 (es) |
| TW (1) | TW200732327A (es) |
| WO (1) | WO2007048643A1 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR080055A1 (es) | 2010-02-01 | 2012-03-07 | Novartis Ag | Derivados de pirazolo-[5,1-b]-oxazol como antagonistas de los receptores de crf -1 |
| AR080056A1 (es) | 2010-02-01 | 2012-03-07 | Novartis Ag | Derivados de ciclohexil-amida como antagonistas de los receptores de crf |
| EP2531490B1 (en) | 2010-02-02 | 2014-10-15 | Novartis AG | Cyclohexyl amide derivatives as crf receptor antagonists |
| ES2734734T3 (es) * | 2015-02-13 | 2019-12-11 | Suven Life Sciences Ltd | Compuestos de amida como agonistas del receptor 5-HT4 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0820586A (ja) * | 1994-07-05 | 1996-01-23 | Sanwa Kagaku Kenkyusho Co Ltd | １−アザビシクロ［３．３．０］オクタン誘導体、その塩及び製法並びに用途 |
| WO2005092882A1 (en) * | 2004-03-01 | 2005-10-06 | Pfizer Japan, Inc. | 4-amino-5-halogeno-benzamide derivatives as 5-ht4 receptor agonists for the treatment of gastrointestinal, cns, neurological and cardiovascular disorders |
-
2006
- 2006-10-26 WO PCT/EP2006/010438 patent/WO2007048643A1/en active Application Filing
- 2006-10-26 AR ARP060104683A patent/AR056729A1/es unknown
- 2006-10-26 PE PE2006001310A patent/PE20070713A1/es not_active Application Discontinuation
- 2006-10-26 TW TW095139451A patent/TW200732327A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PE20070713A1 (es) | 2007-09-27 |
| WO2007048643A1 (en) | 2007-05-03 |
| TW200732327A (en) | 2007-09-01 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| WO2010136474A3 (en) | Substituted aminobutyric derivatives as neprilysin inhibitors | |
| EA200970585A1 (ru) | Бензамидные производные как агонисты ер-рецепторов | |
| IL184932A0 (en) | Glucagon receptor antagonists, preperation and therapeutic uses | |
| EA201200763A1 (ru) | Замещенные производные карбамоилметиламиноуксусной кислоты в качестве новых ингибиторов nep | |
| BRPI0514691A (pt) | composto ou um sal farmaceuticamente aceitável do mesmo, processo para preparar o mesmo, composição farmacêutica, e, uso de um composto ou um sal farmaceuticamente aceitável do mesmo | |
| WO2007135527A3 (en) | Benzimidazolyl compounds | |
| WO2006082523A3 (en) | Pharmaceutical sustained release composition of metformin | |
| RS53521B1 (en) | PREPARATION AND THERAPY APPLICATIONS (2S, 3R) -N-2 - ((3-pyridinyl) methyl) -1-AZABICYCLO [2.2.2] OCT-3-IL) -3,5-DIFLUOROBENZAMIDE | |
| BRPI0611202C1 (pt) | compostos de benzimidazola-carboxamida como agonistas do receptor 5-ht4 | |
| TW200800984A (en) | New compounds | |
| DE602007012313D1 (de) | Als a2b-adenosinrezeptorantagonisten geeignete 5-phenyl-6-pyridin-4-yl-1,3-dihydro-2h-imidazoä4,5-büpyridin-2-onderivate | |
| BRPI0606639A2 (pt) | novo processo para a preparação de indóis substituìdos | |
| CL2007003223A1 (es) | Compuestos derivados de piperidinil 4-arilsulfonamidas n-sustituidas, que actuan como moduladores de la proteina sfrp-1; proceso para preparar los compuestos; co mposicion farmaceutica que comprende a dichos copmpuestos y uso de los compuestos para preparar medicamentos para el tratamiento de enfermedades. | |
| AR059864A1 (es) | Compuesto de benzamida composicion farmaceutica que lo comprende su uso para preparar un medicamento y procedimientos para su preparacion | |
| UY29358A1 (es) | Tiazolidinonas, su preparacion y su uso como medicamento | |
| BRPI0821611A8 (pt) | Derivado de 3-carboxipropil-aminotetralina e compostos relacionados como antagonistas do receptor opióide mu | |
| AR056729A1 (es) | Compuesto de benzofurano carboxamida, composicion farmaceutica que lo comprende su uso para preparar un medicamento y procesos para su preparcion | |
| UA107702C2 (en) | Novel benzamide derivatives | |
| SE0401655D0 (sv) | New compounds | |
| BRPI0618873A2 (pt) | polimorfos c e g purificados, formulação farmacêutica de suspensão e métodos para administrar 17-aag a um indivíduo e para preparar uma formulação farmacêutica, 17-aag purificada e o polimorfo c purificado de 17-aag | |
| MY179041A (en) | Crystalline forms of a 3-carboxypropyl-aminotetralin compound | |
| WO2006106432A3 (en) | 4-arylpiperidine derivatives and use thereof for preparing a medicament for the treatment of cns disorders | |
| EA200802000A1 (ru) | Фармацевтически приемлемые соли и полиморфные формы | |
| NO20090448L (no) | En aminoisoquinolin trombin inhibitor med forbedret biotilgjengelighet | |
| BR112014013590A8 (pt) | derivados de ácidos carboxilícos de cicloalcano como antagonistas do receptor cxcr3 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB | Suspension of granting procedure |