UA76977C2 - Aryl- and heteroaryl substituted chk1 inhibitors and their use as radiosensitizers and chemosensitizers - Google Patents
Aryl- and heteroaryl substituted chk1 inhibitors and their use as radiosensitizers and chemosensitizers Download PDFInfo
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- UA76977C2 UA76977C2 UA2003098173A UA2003098173A UA76977C2 UA 76977 C2 UA76977 C2 UA 76977C2 UA 2003098173 A UA2003098173 A UA 2003098173A UA 2003098173 A UA2003098173 A UA 2003098173A UA 76977 C2 UA76977 C2 UA 76977C2
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- aryl
- group containing
- alkyl
- heteroaryl
- alkylene
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Classifications
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
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- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US27312401P | 2001-03-02 | 2001-03-02 | |
PCT/US2002/006452 WO2002070494A1 (fr) | 2001-03-02 | 2002-03-01 | Uree aryle et heteroaryle utilisee en tant qu'inhibiteur de chk1, a utiliser en tant que radiosensibilisants et chimiosensibilisants |
Publications (1)
Publication Number | Publication Date |
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UA76977C2 true UA76977C2 (en) | 2006-10-16 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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UA2003098173A UA76977C2 (en) | 2001-03-02 | 2002-01-03 | Aryl- and heteroaryl substituted chk1 inhibitors and their use as radiosensitizers and chemosensitizers |
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US (3) | US7067506B2 (fr) |
EP (1) | EP1379510B1 (fr) |
JP (1) | JP4222833B2 (fr) |
KR (2) | KR20080046228A (fr) |
CN (1) | CN100374425C (fr) |
AT (1) | ATE511503T1 (fr) |
AU (1) | AU2002258451B2 (fr) |
BR (1) | BR0207811A (fr) |
CA (1) | CA2439709C (fr) |
CY (1) | CY1111590T1 (fr) |
DK (1) | DK1379510T3 (fr) |
EA (1) | EA014954B1 (fr) |
ES (1) | ES2365504T3 (fr) |
GE (1) | GEP20053659B (fr) |
HK (1) | HK1062438A1 (fr) |
HR (1) | HRP20030688B1 (fr) |
IL (1) | IL157563A0 (fr) |
IS (1) | IS6935A (fr) |
MX (1) | MXPA03007920A (fr) |
NO (1) | NO326776B1 (fr) |
NZ (1) | NZ527787A (fr) |
PL (1) | PL212707B1 (fr) |
PT (1) | PT1379510E (fr) |
RS (1) | RS52077B (fr) |
SI (1) | SI1379510T1 (fr) |
UA (1) | UA76977C2 (fr) |
WO (1) | WO2002070494A1 (fr) |
ZA (1) | ZA200306721B (fr) |
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-
2002
- 2002-01-03 UA UA2003098173A patent/UA76977C2/uk unknown
- 2002-03-01 ES ES02728396T patent/ES2365504T3/es not_active Expired - Lifetime
- 2002-03-01 MX MXPA03007920A patent/MXPA03007920A/es active IP Right Grant
- 2002-03-01 SI SI200230957T patent/SI1379510T1/sl unknown
- 2002-03-01 GE GE5316A patent/GEP20053659B/en unknown
- 2002-03-01 BR BR0207811-2A patent/BR0207811A/pt not_active IP Right Cessation
- 2002-03-01 US US10/087,715 patent/US7067506B2/en not_active Expired - Fee Related
- 2002-03-01 CN CNB028093216A patent/CN100374425C/zh not_active Expired - Fee Related
- 2002-03-01 KR KR1020087008269A patent/KR20080046228A/ko not_active Application Discontinuation
- 2002-03-01 KR KR1020037011393A patent/KR100861829B1/ko not_active IP Right Cessation
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- 2002-03-01 EP EP02728396A patent/EP1379510B1/fr not_active Expired - Lifetime
- 2002-03-01 WO PCT/US2002/006452 patent/WO2002070494A1/fr active Application Filing
- 2002-03-01 EA EA200300947A patent/EA014954B1/ru not_active IP Right Cessation
- 2002-03-01 AU AU2002258451A patent/AU2002258451B2/en not_active Ceased
- 2002-03-01 PL PL364564A patent/PL212707B1/pl unknown
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- 2002-03-01 CA CA2439709A patent/CA2439709C/fr not_active Expired - Fee Related
- 2002-03-01 AT AT02728396T patent/ATE511503T1/de active
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- 2002-03-01 RS YU69003A patent/RS52077B/sr unknown
- 2002-03-01 IL IL15756302A patent/IL157563A0/xx unknown
- 2002-03-01 DK DK02728396.9T patent/DK1379510T3/da active
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2003
- 2003-08-28 HR HRP20030688AA patent/HRP20030688B1/hr not_active IP Right Cessation
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- 2003-08-29 IS IS6935A patent/IS6935A/is unknown
- 2003-09-01 NO NO20033858A patent/NO326776B1/no not_active IP Right Cessation
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2004
- 2004-07-12 HK HK04105049.6A patent/HK1062438A1/xx not_active IP Right Cessation
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2005
- 2005-04-27 US US11/115,993 patent/US7608618B2/en not_active Expired - Fee Related
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2009
- 2009-09-01 US US12/551,623 patent/US20100105683A1/en not_active Abandoned
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2011
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