UA5971A1 - Спосіб отримання похідного [3н]-імідазо-[5,1-а]-1,2,3,5-тетразін-4-она - Google Patents

Спосіб отримання похідного [3н]-імідазо-[5,1-а]-1,2,3,5-тетразін-4-она

Info

Publication number
UA5971A1
UA5971A1 UA3482389A UA3482389A UA5971A1 UA 5971 A1 UA5971 A1 UA 5971A1 UA 3482389 A UA3482389 A UA 3482389A UA 3482389 A UA3482389 A UA 3482389A UA 5971 A1 UA5971 A1 UA 5971A1
Authority
UA
Ukraine
Prior art keywords
tetrazin
imidazo
derivative
preparation
isocyanate
Prior art date
Application number
UA3482389A
Other languages
English (en)
Russian (ru)
Ukrainian (uk)
Inventor
Лант Едвард
Френкіс Грахам Стівенс Малькольм
Стоун Роберт
Роберт Харрі Вулдрідж Кеннет
Original Assignee
Мбл (1991) Лімітед
МБЛ (1991) Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Мбл (1991) Лімітед, МБЛ (1991) Лимитед filed Critical Мбл (1991) Лімітед
Publication of UA5971A1 publication Critical patent/UA5971A1/uk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
UA3482389A 1981-08-24 1982-08-23 Спосіб отримання похідного [3н]-імідазо-[5,1-а]-1,2,3,5-тетразін-4-она UA5971A1 (uk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8125791 1981-08-24

Publications (1)

Publication Number Publication Date
UA5971A1 true UA5971A1 (uk) 1994-12-29

Family

ID=10524141

Family Applications (1)

Application Number Title Priority Date Filing Date
UA3482389A UA5971A1 (uk) 1981-08-24 1982-08-23 Спосіб отримання похідного [3н]-імідазо-[5,1-а]-1,2,3,5-тетразін-4-она

Country Status (29)

Country Link
JP (1) JPS5843975A (enExample)
KR (1) KR890000094B1 (enExample)
AT (1) AT380256B (enExample)
AU (1) AU571430B2 (enExample)
BE (1) BE894175A (enExample)
CA (1) CA1197247A (enExample)
CH (1) CH655114A5 (enExample)
DE (2) DE19975037I2 (enExample)
DK (1) DK161147C (enExample)
ES (1) ES515176A0 (enExample)
FI (1) FI73434C (enExample)
FR (1) FR2511679A1 (enExample)
GB (1) GB2104522B (enExample)
GE (1) GEP19960641B (enExample)
GR (1) GR76863B (enExample)
HU (1) HU186107B (enExample)
IE (1) IE53408B1 (enExample)
IL (1) IL66606A (enExample)
IT (1) IT1152505B (enExample)
LT (1) LT2436B (enExample)
LU (1) LU84347A1 (enExample)
LV (2) LV5511A3 (enExample)
NL (2) NL192739C (enExample)
NZ (1) NZ201668A (enExample)
OA (1) OA07174A (enExample)
SE (1) SE448543B (enExample)
SU (1) SU1447284A3 (enExample)
UA (1) UA5971A1 (enExample)
ZA (1) ZA826120B (enExample)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5260291A (en) * 1981-08-24 1993-11-09 Cancer Research Campaign Technology Limited Tetrazine derivatives
GR78688B (enExample) * 1982-08-17 1984-09-27 May & Baker Ltd
GB2125402B (en) * 1982-08-17 1985-11-13 May & Baker Ltd New tetrazine derivatives
US4517182A (en) * 1983-05-24 1985-05-14 Warner-Lambert Company 3-(Haloethyl)-4-oxopyrazolo-[5,1-d]-1,2,3,5-tetrazine-8-carboxamide composition
GB8616125D0 (en) * 1986-07-02 1986-08-06 May & Baker Ltd Compositions of matter
AU622330B2 (en) * 1989-06-23 1992-04-02 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
EP0866709B1 (en) * 1995-09-25 2007-01-10 Sanofi-Aventis U.S. LLC 1,2,4-benzotriazine oxides formulations
BRPI0417117A (pt) * 2003-12-30 2007-03-06 Chemagis Ltd temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica
CA2594477C (en) 2005-01-21 2016-07-12 Astex Therapeutics Limited Pharmaceutical compounds
AR060635A1 (es) 2006-04-27 2008-07-02 Banyu Pharma Co Ltd Derivados de 1,2-dihidro-3h-pirazolo[3,4-d]pirimidin-3-ona, composiciones farmaceuticas que los comprenden y su uso en el tratamiento del cancer
JP2008081492A (ja) 2006-08-31 2008-04-10 Banyu Pharmaceut Co Ltd オーロラａ選択的阻害作用を有する新規アミノピリジン誘導体
EP2073803B1 (en) 2006-10-12 2018-09-19 Astex Therapeutics Limited Pharmaceutical combinations
US8883790B2 (en) 2006-10-12 2014-11-11 Astex Therapeutics Limited Pharmaceutical combinations
JPWO2009054332A1 (ja) 2007-10-23 2011-03-03 萬有製薬株式会社 ピリドン置換ジヒドロピラゾロピリミジノン誘導体
PE20091101A1 (es) * 2007-12-18 2009-07-26 Pharminox Ltd AMIDAS DE ACIDO 3-SUBSTITUIDO-4-OXO-3,4-DIHIDRO-IMIDAZO[5,1-d] [1,2,3,5-TETRACINA-8-CARBOXILICO Y SU EMPLEO
KR20110111383A (ko) * 2008-11-24 2011-10-11 리라이언스 라이프 사이언시스 프라이빗. 리미티드 테트라진 유도체의 제조 방법
WO2010101734A1 (en) 2009-03-06 2010-09-10 Merck Sharp & Dohme Corp. Combination cancer therapy with an akt inhibitor and other anticancer agents
BRPI1011822A2 (pt) 2009-06-23 2016-03-29 Pharminox Ltd "compostos de 3-substituída-8-substituída-3h-imidazo[5,1-d][1,2,3,5-tetrazin-4-ona e sua aplicação"
RU2462466C1 (ru) * 2011-06-24 2012-09-27 Автономная Некоммерческая Организация "Научно-Исследовательский Центр Биотехнологии Антибиотиков И Других Биологически Активных Веществ "Биоан" Замещенные азоло[1,2,4,5]тетразины - ингибиторы актинобактериальных серин-треониновых протеинкиназ
WO2013055985A1 (en) 2011-10-12 2013-04-18 Children's Medical Center Corporation Combinatorial compositions and methods of treating hemoglobinopathies
CN120661674A (zh) 2016-03-15 2025-09-19 奥莱松基因组股份有限公司 用于治疗实体瘤的lsd1抑制剂的组合
KR101847342B1 (ko) * 2017-05-08 2018-04-11 (주)센텍코리아 웨어러블 체지방 연소량 측정기

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2932305A1 (de) * 1979-08-09 1981-02-26 Basf Ag Azolo- eckige klammer auf 5,1-d eckige klammer zu - eckige klammer auf 1,2,3,5 eckige klammer zu -tetrazin-4-one und verfahren zur herstellung dieser verbindungen

Also Published As

Publication number Publication date
BE894175A (fr) 1983-02-23
FI822921A0 (fi) 1982-08-23
SE8204817L (sv) 1983-02-25
JPS5843975A (ja) 1983-03-14
DE19975037I2 (de) 2001-06-13
GB2104522A (en) 1983-03-09
LT2436B (lt) 1994-02-15
NL990010I1 (nl) 1999-07-01
LV5621A3 (lv) 1994-05-10
JPH045029B2 (enExample) 1992-01-30
DE3231255A1 (de) 1983-03-03
IL66606A0 (en) 1982-12-31
FR2511679A1 (fr) 1983-02-25
DK161147B (da) 1991-06-03
GB2104522B (en) 1985-06-12
ES8400438A1 (es) 1983-11-01
FI73434B (fi) 1987-06-30
AT380256B (de) 1986-05-12
DK377882A (da) 1983-02-25
SE8204817D0 (sv) 1982-08-23
ATA319182A (de) 1985-09-15
OA07174A (fr) 1984-04-30
IT1152505B (it) 1987-01-07
FR2511679B1 (enExample) 1985-02-01
LU84347A1 (fr) 1983-06-07
LV5511A3 (lv) 1994-03-10
KR890000094B1 (ko) 1989-03-07
NL8203286A (nl) 1983-03-16
NL990010I2 (nl) 1999-09-01
DK161147C (da) 1991-11-18
NL192739B (nl) 1997-09-01
NZ201668A (en) 1985-08-16
IE822026L (en) 1983-02-24
DE3231255C2 (enExample) 1992-02-27
CH655114A5 (fr) 1986-03-27
HU186107B (en) 1985-06-28
IT8222938A1 (it) 1984-02-23
ES515176A0 (es) 1983-11-01
IL66606A (en) 1987-07-31
IE53408B1 (en) 1988-11-09
KR840001175A (ko) 1984-03-28
FI73434C (fi) 1987-10-09
NL192739C (nl) 1998-01-06
IT8222938A0 (it) 1982-08-23
CA1197247A (fr) 1985-11-26
SE448543B (sv) 1987-03-02
GEP19960641B (en) 1996-11-15
AU571430B2 (en) 1988-04-21
GR76863B (enExample) 1984-09-04
FI822921L (fi) 1983-02-25
AU8749382A (en) 1983-03-03
SU1447284A3 (ru) 1988-12-23
ZA826120B (en) 1983-07-27

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