UA114075C2 - БАГАТОШАРОВА ТАБЛЕТКА, ЩО МІСТИТЬ РИЛПІВІРИН HCl, ЕМТРИЦИТАБІН І ТЕНОФОВІРУ ДИЗОПРОКСИЛФУМАРАТ - Google Patents

БАГАТОШАРОВА ТАБЛЕТКА, ЩО МІСТИТЬ РИЛПІВІРИН HCl, ЕМТРИЦИТАБІН І ТЕНОФОВІРУ ДИЗОПРОКСИЛФУМАРАТ

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Publication number
UA114075C2
UA114075C2 UAA201306403A UAA201306403A UA114075C2 UA 114075 C2 UA114075 C2 UA 114075C2 UA A201306403 A UAA201306403 A UA A201306403A UA A201306403 A UAA201306403 A UA A201306403A UA 114075 C2 UA114075 C2 UA 114075C2
Authority
UA
Ukraine
Prior art keywords
tenofovir
disoproxylfumarate
emtricitabin
table containing
layer table
Prior art date
Application number
UAA201306403A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45094284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA114075(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of UA114075C2 publication Critical patent/UA114075C2/uk

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

У даному винаході запропоновані багатошарові таблетки, що містять гідрохлорид рилпівірину, емтрицитабін і тенофовіру дизопроксилфумарат. Зазначені таблетки підходять для лікування ВІЛ.
UAA201306403A 2010-11-19 2011-11-18 БАГАТОШАРОВА ТАБЛЕТКА, ЩО МІСТИТЬ РИЛПІВІРИН HCl, ЕМТРИЦИТАБІН І ТЕНОФОВІРУ ДИЗОПРОКСИЛФУМАРАТ UA114075C2 (xx)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41560010P 2010-11-19 2010-11-19
PCT/US2011/061515 WO2012068535A1 (en) 2010-11-19 2011-11-18 Therapeutic compositions comprising rilpivirine hcl and tenofovir disoproxil fumarate

Publications (1)

Publication Number Publication Date
UA114075C2 true UA114075C2 (xx) 2017-04-25

Family

ID=45094284

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201306403A UA114075C2 (xx) 2010-11-19 2011-11-18 БАГАТОШАРОВА ТАБЛЕТКА, ЩО МІСТИТЬ РИЛПІВІРИН HCl, ЕМТРИЦИТАБІН І ТЕНОФОВІРУ ДИЗОПРОКСИЛФУМАРАТ

Country Status (35)

Country Link
US (1) US10857102B2 (uk)
EP (2) EP2640362B2 (uk)
JP (2) JP2014500261A (uk)
KR (1) KR101923103B1 (uk)
CN (2) CN106511357A (uk)
AP (1) AP3816A (uk)
AR (2) AR084500A1 (uk)
AU (3) AU2011329642B2 (uk)
BR (1) BR112013012245B1 (uk)
CA (1) CA2818097C (uk)
CL (1) CL2013001402A1 (uk)
CO (1) CO6761300A2 (uk)
CR (1) CR20130293A (uk)
DK (1) DK2640362T4 (uk)
EA (2) EA025852B1 (uk)
EC (2) ECSP13012700A (uk)
ES (1) ES2524408T5 (uk)
HK (2) HK1190064A1 (uk)
HR (1) HRP20140946T1 (uk)
IL (1) IL226300B (uk)
MA (1) MA34735B1 (uk)
ME (1) ME01980B (uk)
MX (1) MX347512B (uk)
MY (1) MY185604A (uk)
NZ (1) NZ610729A (uk)
PE (3) PE20140163A1 (uk)
PL (1) PL2640362T5 (uk)
PT (1) PT2640362E (uk)
RS (1) RS53691B1 (uk)
SG (3) SG10201912527XA (uk)
SM (1) SMT201400150B (uk)
TW (1) TWI556840B (uk)
UA (1) UA114075C2 (uk)
WO (1) WO2012068535A1 (uk)
ZA (1) ZA201304481B (uk)

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AU2012296622C1 (en) 2011-08-16 2017-02-16 Gilead Sciences, Inc. Tenofovir alafenamide hemifumarate
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JP2022538338A (ja) * 2019-07-03 2022-09-01 ヤンセン・サイエンシズ・アイルランド・アンリミテッド・カンパニー リルピビリンを用いて小児患者におけるｈｉｖを治療する方法
CN112137981A (zh) * 2020-11-02 2020-12-29 成都晶富医药科技有限公司 富马酸丙酚替诺福韦片及其制备工艺

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Also Published As

Publication number Publication date
AP2013006931A0 (en) 2013-06-30
AU2018202635A1 (en) 2018-05-10
EP2826466A1 (en) 2015-01-21
EP2640362A1 (en) 2013-09-25
KR101923103B1 (ko) 2018-11-28
CA2818097A1 (en) 2012-05-24
HRP20140946T1 (hr) 2015-02-13
AU2011329642B2 (en) 2016-08-11
HK1190064A1 (en) 2014-06-27
AR084500A1 (es) 2013-05-22
MX347512B (es) 2017-04-28
JP2015131853A (ja) 2015-07-23
WO2012068535A1 (en) 2012-05-24
EA201390651A1 (ru) 2013-11-29
PT2640362E (pt) 2014-11-28
DK2640362T4 (da) 2022-03-07
ECSP19078196A (es) 2019-11-30
MX2013005669A (es) 2013-11-04
CO6761300A2 (es) 2013-09-30
ECSP13012700A (es) 2013-08-30
CN106511357A (zh) 2017-03-22
ZA201304481B (en) 2022-03-30
KR20140037799A (ko) 2014-03-27
EP2640362B2 (en) 2021-12-01
HK1206592A1 (en) 2016-01-15
EP2640362B1 (en) 2014-09-10
AP3816A (en) 2016-09-30
EA025852B1 (ru) 2017-02-28
PE20170521A1 (es) 2017-05-27
CN103491948A (zh) 2014-01-01
SG10201509521WA (en) 2015-12-30
CL2013001402A1 (es) 2013-12-27
ES2524408T5 (es) 2022-04-25
PE20140163A1 (es) 2014-02-08
SMT201400150B (it) 2015-01-15
AU2011329642A1 (en) 2013-05-02
AR123409A2 (es) 2022-11-30
JP2014500261A (ja) 2014-01-09
TW201238612A (en) 2012-10-01
TWI556840B (zh) 2016-11-11
CA2818097C (en) 2019-07-30
IL226300B (en) 2019-05-30
US10857102B2 (en) 2020-12-08
BR112013012245B1 (pt) 2022-09-27
MA34735B1 (fr) 2013-12-03
PL2640362T3 (pl) 2015-03-31
MY185604A (en) 2021-05-25
SG190333A1 (en) 2013-06-28
AU2016208417B2 (en) 2018-04-05
NZ610729A (en) 2015-10-30
AU2016208417A1 (en) 2016-08-18
CN103491948B (zh) 2016-11-02
RS53691B1 (en) 2015-04-30
EA201691695A1 (ru) 2017-11-30
ES2524408T3 (es) 2014-12-09
CR20130293A (es) 2013-10-03
JP6138851B2 (ja) 2017-05-31
ME01980B (me) 2015-05-20
US20130243857A1 (en) 2013-09-19
SG10201912527XA (en) 2020-02-27
BR112013012245A2 (pt) 2016-08-09
PL2640362T5 (pl) 2022-05-02
DK2640362T3 (en) 2014-12-01
PE20211657A1 (es) 2021-08-24

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