ECSP13012700A - Composiciones terapéuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato - Google Patents

Composiciones terapéuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato

Info

Publication number
ECSP13012700A
ECSP13012700A ECSP13012700A ECSP13012700A EC SP13012700 A ECSP13012700 A EC SP13012700A EC SP13012700 A ECSP13012700 A EC SP13012700A EC SP13012700 A ECSP13012700 A EC SP13012700A
Authority
EC
Ecuador
Prior art keywords
disoproxil fumarate
therapeutic compositions
tenofovir disoproxil
rilpivirine hcl
include rilpivirine
Prior art date
Application number
Other languages
English (en)
Inventor
Mark M Menning
Reza Oliyal
Lauren Wiser
Original Assignee
Gilead Sciences Inc
Janssen R & D Ireland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45094284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP13012700(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc, Janssen R & D Ireland filed Critical Gilead Sciences Inc
Publication of ECSP13012700A publication Critical patent/ECSP13012700A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La invención presenta tabletas multicapas que contienen rilpivirina clorhidrato, emtricitabina y tenofivir disoproxil fumarato. Las tabletas son útiles para el tratamiento del HIV.
ECSP13012700 2010-11-19 2013-06-18 Composiciones terapéuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato ECSP13012700A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41560010P 2010-11-19 2010-11-19

Publications (1)

Publication Number Publication Date
ECSP13012700A true ECSP13012700A (es) 2013-08-30

Family

ID=45094284

Family Applications (2)

Application Number Title Priority Date Filing Date
ECSP13012700 ECSP13012700A (es) 2010-11-19 2013-06-18 Composiciones terapéuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato
ECSENADI201978196A ECSP19078196A (es) 2010-11-19 2019-10-30 Composiciones terapéuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato

Family Applications After (1)

Application Number Title Priority Date Filing Date
ECSENADI201978196A ECSP19078196A (es) 2010-11-19 2019-10-30 Composiciones terapéuticas que comprenden rilpivirina hcl y tenofovir disoproxil fumarato

Country Status (35)

Country Link
US (1) US10857102B2 (es)
EP (2) EP2640362B2 (es)
JP (2) JP2014500261A (es)
KR (1) KR101923103B1 (es)
CN (2) CN106511357A (es)
AP (1) AP3816A (es)
AR (2) AR084500A1 (es)
AU (3) AU2011329642B2 (es)
BR (1) BR112013012245B1 (es)
CA (1) CA2818097C (es)
CL (1) CL2013001402A1 (es)
CO (1) CO6761300A2 (es)
CR (1) CR20130293A (es)
DK (1) DK2640362T4 (es)
EA (2) EA201691695A1 (es)
EC (2) ECSP13012700A (es)
ES (1) ES2524408T5 (es)
HK (2) HK1190064A1 (es)
HR (1) HRP20140946T1 (es)
IL (1) IL226300B (es)
MA (1) MA34735B1 (es)
ME (1) ME01980B (es)
MX (1) MX347512B (es)
MY (1) MY185604A (es)
NZ (1) NZ610729A (es)
PE (3) PE20140163A1 (es)
PL (1) PL2640362T5 (es)
PT (1) PT2640362E (es)
RS (1) RS53691B1 (es)
SG (3) SG10201912527XA (es)
SM (1) SMT201400150B (es)
TW (1) TWI556840B (es)
UA (1) UA114075C2 (es)
WO (1) WO2012068535A1 (es)
ZA (1) ZA201304481B (es)

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PL2640362T5 (pl) 2010-11-19 2022-05-02 Gilead Sciences, Inc. Kompozycje terapeutyczne zawierające hcl rylpiwiryny i fumaran dizoproksylu tenofowiru
AR087546A1 (es) 2011-08-16 2014-04-03 Gilead Sciences Inc Hemifumarato de tenofovir alafenamida
CA2779052A1 (en) * 2012-05-31 2013-11-30 Pharmascience Inc. Pharmaceutical composition of entecavir and process of manufacturing
MD4736C1 (ro) 2012-12-21 2021-07-31 Gilead Sciences, Inc. Compus policiclic de carbamoilpiridonă şi utilizarea farmaceutică a acestuia
EP2832351A1 (en) * 2013-07-29 2015-02-04 Sanovel Ilac Sanayi ve Ticaret A.S. Multilayer Tablet Formulations Comprising Tenofovir and Entecavir
CZ2013985A3 (cs) * 2013-12-09 2015-06-17 Zentiva, K.S. Stabilní farmaceutická kompozice obsahující tenofovir disoproxil fumarát
WO2015152433A1 (en) * 2014-03-31 2015-10-08 Hanmi Pharm. Co., Ltd. Amorphous solid dispersion comprising paclitaxel, tablet comprising the same, and method for preparing the same
KR20230130175A (ko) 2014-12-26 2023-09-11 에모리 유니버시티 Ｎ4-하이드록시시티딘, 이와 관련된 유도체 및 이의 항 바이러스적 용도
US9839212B2 (en) 2015-04-16 2017-12-12 Bio-Lab, Inc. Multicomponent and multilayer compacted tablets
CA2921336A1 (en) * 2015-06-30 2016-12-30 Gilead Sciences, Inc. Pharmaceutical formulations
KR20170003063A (ko) * 2015-06-30 2017-01-09 한미약품 주식회사 테노포비어 디소프록실 함유 경구용 고형제제 및 그 제조방법
BR102016026127A2 (pt) * 2015-11-09 2017-05-16 Gilead Sciences Inc composições terapêuticas para o tratamento do vírus da imunodeficiência humana
JP2019513754A (ja) * 2016-04-08 2019-05-30 塩野義製薬株式会社 安定化した固形製剤
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WO2021001508A1 (en) * 2019-07-03 2021-01-07 Janssen Sciences Ireland Unlimited Company Methods of treating hiv in pediatric patients with rilpivirine
CN112137981A (zh) * 2020-11-02 2020-12-29 成都晶富医药科技有限公司 富马酸丙酚替诺福韦片及其制备工艺

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Also Published As

Publication number Publication date
AU2011329642B2 (en) 2016-08-11
ZA201304481B (en) 2022-03-30
AU2016208417B2 (en) 2018-04-05
UA114075C2 (xx) 2017-04-25
MX2013005669A (es) 2013-11-04
AU2018202635A1 (en) 2018-05-10
PE20140163A1 (es) 2014-02-08
DK2640362T3 (en) 2014-12-01
AU2016208417A1 (en) 2016-08-18
CN103491948A (zh) 2014-01-01
AP3816A (en) 2016-09-30
SMT201400150B (it) 2015-01-15
AR084500A1 (es) 2013-05-22
SG10201912527XA (en) 2020-02-27
CA2818097A1 (en) 2012-05-24
EP2826466A1 (en) 2015-01-21
TWI556840B (zh) 2016-11-11
PE20211657A1 (es) 2021-08-24
EA025852B1 (ru) 2017-02-28
CL2013001402A1 (es) 2013-12-27
HRP20140946T1 (hr) 2015-02-13
RS53691B1 (en) 2015-04-30
CO6761300A2 (es) 2013-09-30
IL226300B (en) 2019-05-30
AU2011329642A1 (en) 2013-05-02
DK2640362T4 (da) 2022-03-07
ECSP19078196A (es) 2019-11-30
EA201390651A1 (ru) 2013-11-29
ES2524408T5 (es) 2022-04-25
MA34735B1 (fr) 2013-12-03
MX347512B (es) 2017-04-28
MY185604A (en) 2021-05-25
SG10201509521WA (en) 2015-12-30
ES2524408T3 (es) 2014-12-09
KR20140037799A (ko) 2014-03-27
SG190333A1 (en) 2013-06-28
CR20130293A (es) 2013-10-03
PL2640362T5 (pl) 2022-05-02
BR112013012245B1 (pt) 2022-09-27
CN106511357A (zh) 2017-03-22
EP2640362B2 (en) 2021-12-01
US20130243857A1 (en) 2013-09-19
AR123409A2 (es) 2022-11-30
JP6138851B2 (ja) 2017-05-31
ME01980B (me) 2015-05-20
CN103491948B (zh) 2016-11-02
JP2014500261A (ja) 2014-01-09
PE20170521A1 (es) 2017-05-27
PL2640362T3 (pl) 2015-03-31
JP2015131853A (ja) 2015-07-23
CA2818097C (en) 2019-07-30
BR112013012245A2 (pt) 2016-08-09
EP2640362B1 (en) 2014-09-10
HK1206592A1 (en) 2016-01-15
US10857102B2 (en) 2020-12-08
AP2013006931A0 (en) 2013-06-30
WO2012068535A1 (en) 2012-05-24
NZ610729A (en) 2015-10-30
KR101923103B1 (ko) 2018-11-28
TW201238612A (en) 2012-10-01
HK1190064A1 (en) 2014-06-27
EP2640362A1 (en) 2013-09-25
PT2640362E (pt) 2014-11-28
EA201691695A1 (ru) 2017-11-30

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