TR201802093T4 - Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu. - Google Patents

Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu. Download PDF

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Publication number
TR201802093T4
TR201802093T4 TR2018/02093T TR201802093T TR201802093T4 TR 201802093 T4 TR201802093 T4 TR 201802093T4 TR 2018/02093 T TR2018/02093 T TR 2018/02093T TR 201802093 T TR201802093 T TR 201802093T TR 201802093 T4 TR201802093 T4 TR 201802093T4
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Turkey
Prior art keywords
compound
mmol
cancer
abiraterone
combination
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TR2018/02093T
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English (en)
Turkish (tr)
Inventor
Nannini Michelle
Sampath Deepak
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Genentech Inc
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46931958&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR201802093(T4) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Genentech Inc filed Critical Genentech Inc
Publication of TR201802093T4 publication Critical patent/TR201802093T4/tr

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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  • Steroid Compounds (AREA)
TR2018/02093T 2011-04-01 2012-03-30 Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu. TR201802093T4 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161470803P 2011-04-01 2011-04-01
US201161470624P 2011-04-01 2011-04-01

Publications (1)

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TR201802093T4 true TR201802093T4 (tr) 2018-03-21

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TR2018/02093T TR201802093T4 (tr) 2011-04-01 2012-03-30 Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu.

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US (7) US9150548B2 (enExample)
EP (4) EP2694072B2 (enExample)
JP (4) JP6143739B2 (enExample)
KR (4) KR20140025434A (enExample)
CN (8) CN103874689B (enExample)
AU (4) AU2012236138A1 (enExample)
BR (4) BR112013025354A2 (enExample)
CA (4) CA2844699C (enExample)
DK (1) DK2694072T4 (enExample)
ES (3) ES2657750T3 (enExample)
FI (1) FI2694072T4 (enExample)
HK (1) HK1204575A1 (enExample)
HR (1) HRP20180223T4 (enExample)
HU (1) HUE036513T2 (enExample)
IL (4) IL228642A0 (enExample)
LT (1) LT2694072T (enExample)
ME (1) ME02998B (enExample)
MX (4) MX2013011329A (enExample)
MY (1) MY179607A (enExample)
PL (2) PL2694485T3 (enExample)
PT (1) PT2694072T (enExample)
RS (1) RS56759B2 (enExample)
RU (4) RU2013148732A (enExample)
SG (5) SG194048A1 (enExample)
SI (1) SI2694072T2 (enExample)
SM (1) SMT201800250T1 (enExample)
TR (1) TR201802093T4 (enExample)
WO (4) WO2012135759A1 (enExample)
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KR101653842B1 (ko) 2008-01-04 2016-09-02 인텔리카인, 엘엘씨 특정 화학 물질, 조성물 및 방법
DK2959900T3 (en) 2008-06-16 2017-06-26 Univ Tennessee Res Found CONNECTION TO TREATMENT OF CANCER
US9447049B2 (en) 2010-03-01 2016-09-20 University Of Tennessee Research Foundation Compounds for treatment of cancer
US11084811B2 (en) 2010-03-01 2021-08-10 Oncternal Therapeutics, Inc. Compounds for treatment of cancer
AR084824A1 (es) 2011-01-10 2013-06-26 Intellikine Inc Procesos para preparar isoquinolinonas y formas solidas de isoquinolinonas
SG10201600077RA (en) 2011-01-11 2016-02-26 Glaxosmithkline Llc Combination
WO2012135759A1 (en) 2011-04-01 2012-10-04 Genentech, Inc. Combinations of akt inhibitor compounds and abiraterone, and methods of use
US9216170B2 (en) 2012-03-19 2015-12-22 Hoffmann-La Roche Inc. Combination therapy for proliferative disorders
US20150023954A1 (en) * 2012-03-23 2015-01-22 Memorial Sloan-Kettering Cancer Center Potentiating antibody-induced complement-mediated cytotoxicity via pi3k inhibition
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