TR201802093T4 - Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu. - Google Patents

Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu. Download PDF

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Publication number
TR201802093T4
TR201802093T4 TR2018/02093T TR201802093T TR201802093T4 TR 201802093 T4 TR201802093 T4 TR 201802093T4 TR 2018/02093 T TR2018/02093 T TR 2018/02093T TR 201802093 T TR201802093 T TR 201802093T TR 201802093 T4 TR201802093 T4 TR 201802093T4
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Turkey
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mmol
mixture
compound
methyl
solution
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TR2018/02093T
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English (en)
Turkish (tr)
Inventor
Nannini Michelle
Sampath Deepak
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Genentech Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46931958&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR201802093(T4) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Genentech Inc filed Critical Genentech Inc
Publication of TR201802093T4 publication Critical patent/TR201802093T4/tr

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
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    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
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  • Oncology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
TR2018/02093T 2011-04-01 2012-03-30 Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu. TR201802093T4 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161470803P 2011-04-01 2011-04-01
US201161470624P 2011-04-01 2011-04-01

Publications (1)

Publication Number Publication Date
TR201802093T4 true TR201802093T4 (tr) 2018-03-21

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TR2018/02093T TR201802093T4 (tr) 2011-04-01 2012-03-30 Terapötik terapilerde kullanım için akt inhibitör bileşiği ve abirateron kombinasyonu.

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Country Link
US (7) US20150064171A1 (enExample)
EP (4) EP2694072B2 (enExample)
JP (4) JP6239497B2 (enExample)
KR (4) KR101950044B1 (enExample)
CN (8) CN104586861A (enExample)
AU (4) AU2012236135A1 (enExample)
BR (4) BR112013025386B1 (enExample)
CA (4) CA2831937A1 (enExample)
DK (1) DK2694072T4 (enExample)
ES (3) ES2660263T5 (enExample)
FI (1) FI2694072T4 (enExample)
HK (1) HK1204575A1 (enExample)
HR (1) HRP20180223T4 (enExample)
HU (1) HUE036513T2 (enExample)
IL (4) IL228638A0 (enExample)
LT (1) LT2694072T (enExample)
ME (1) ME02998B (enExample)
MX (4) MX354509B (enExample)
MY (1) MY179607A (enExample)
PL (2) PL2694072T5 (enExample)
PT (1) PT2694072T (enExample)
RS (1) RS56759B2 (enExample)
RU (4) RU2013148721A (enExample)
SG (5) SG10201504303SA (enExample)
SI (1) SI2694072T2 (enExample)
SM (1) SMT201800250T1 (enExample)
TR (1) TR201802093T4 (enExample)
WO (4) WO2012135750A1 (enExample)
ZA (4) ZA201308062B (enExample)

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KR101660050B1 (ko) 2008-01-04 2016-09-26 인텔리카인, 엘엘씨 특정 화학 물질, 조성물 및 방법
US9447049B2 (en) 2010-03-01 2016-09-20 University Of Tennessee Research Foundation Compounds for treatment of cancer
HUE034598T2 (en) 2008-06-16 2018-02-28 Univ Tennessee Res Found Compound for cancer treatment
US11084811B2 (en) 2010-03-01 2021-08-10 Oncternal Therapeutics, Inc. Compounds for treatment of cancer
NZ612909A (en) 2011-01-10 2015-09-25 Infinity Pharmaceuticals Inc Processes for preparing isoquinolinones and solid forms of isoquinolinones
MX356704B (es) 2011-01-11 2018-06-11 Novartis Ag Combinación.
JP6239497B2 (ja) 2011-04-01 2017-11-29 ジェネンテック， インコーポレイテッド Ａｋｔ阻害剤化合物及びアビラテロンの組み合わせ、及び使用方法
US9216170B2 (en) 2012-03-19 2015-12-22 Hoffmann-La Roche Inc. Combination therapy for proliferative disorders
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