TR200805741T2 - At-1 veya at-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı@ - Google Patents

At-1 veya at-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı@

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Publication number
TR200805741T2
TR200805741T2 TR2008/05741T TR200805741T TR200805741T2 TR 200805741 T2 TR200805741 T2 TR 200805741T2 TR 2008/05741 T TR2008/05741 T TR 2008/05741T TR 200805741 T TR200805741 T TR 200805741T TR 200805741 T2 TR200805741 T2 TR 200805741T2
Authority
TR
Turkey
Prior art keywords
receptors
treatment
receptor
increased
diseases caused
Prior art date
Application number
TR2008/05741T
Other languages
English (en)
Inventor
Rosemary Bullock Gillian
Maria Ganter Sabina
De Gasparo Marc
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26152118&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR200805741(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from EP98811258A external-priority patent/EP1013273A1/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of TR200805741T2 publication Critical patent/TR200805741T2/tr

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455—Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
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  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Buluş, sub-epitelial alandaki AT1 reseptörlerinin artışı veya epiteliadaki AT2 reseptörlerinin artışının neden olduğu hastalıkların ya da durumların tedavisi için farmasotik bir preparasyon üretmek amacıyla sırasıyla bir AT1 reseptör antagonistinin ya da bir AT2 reseptör modülatörünün ya da onun farmasotik olarak uygun bir tuzunun kullanımı ile ilgilidir.
TR2008/05741T 1998-12-23 1999-12-22 At-1 veya at-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı@ TR200805741T2 (tr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP98811258A EP1013273A1 (en) 1998-12-23 1998-12-23 Use of AT-1 receptor antagonist or AT-2 receptor modulator for treating diseases associated with an increase of AT-1 or AT-2 receptors
EP98811257 1998-12-23

Publications (1)

Publication Number Publication Date
TR200805741T2 true TR200805741T2 (tr) 2008-10-21

Family

ID=26152118

Family Applications (7)

Application Number Title Priority Date Filing Date
TR2008/05275T TR200805275T2 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı@
TR2006/05471T TR200605471T2 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı@
TR2001/01784T TR200101784T2 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı.
TR2008/05740T TR200805740T1 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı@
TR2002/00764T TR200200764T2 (tr) 1998-12-23 1999-12-22 At-1 veya at-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı
TR2008/05741T TR200805741T2 (tr) 1998-12-23 1999-12-22 At-1 veya at-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı@
TR2006/05472T TR200605472T1 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı@

Family Applications Before (5)

Application Number Title Priority Date Filing Date
TR2008/05275T TR200805275T2 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı@
TR2006/05471T TR200605471T2 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı@
TR2001/01784T TR200101784T2 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı.
TR2008/05740T TR200805740T1 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı@
TR2002/00764T TR200200764T2 (tr) 1998-12-23 1999-12-22 At-1 veya at-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için at-1 reseptör antagonisti veya at-2 reseptör modülatörünün kullanımı

Family Applications After (1)

Application Number Title Priority Date Filing Date
TR2006/05472T TR200605472T1 (tr) 1998-12-23 1999-12-22 AT-1 veya AT-2 reseptörlerindeki artışın neden olduğu hastalıkların tedavisi için AT-1 reseptör antagonisti veya AT-2 reseptör modülatörünün kullanımı@

Country Status (26)

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EP (3) EP2298298A3 (tr)
JP (2) JP2002533390A (tr)
KR (1) KR100646716B1 (tr)
CN (2) CN1636561A (tr)
AT (2) ATE354364T1 (tr)
AU (4) AU3043000A (tr)
BR (1) BR9916576A (tr)
CA (2) CA2351357A1 (tr)
CY (2) CY1106581T1 (tr)
CZ (2) CZ297795B6 (tr)
DE (1) DE69935249T2 (tr)
DK (2) DK1140071T3 (tr)
ES (2) ES2373556T3 (tr)
HK (1) HK1038888B (tr)
HU (1) HUP0104780A3 (tr)
ID (1) ID29856A (tr)
IL (5) IL143233A0 (tr)
NO (2) NO328775B1 (tr)
NZ (3) NZ587909A (tr)
PL (1) PL199100B1 (tr)
PT (2) PT1588706E (tr)
RU (3) RU2271809C2 (tr)
SI (2) SI1140071T1 (tr)
SK (1) SK9132001A3 (tr)
TR (7) TR200805275T2 (tr)
WO (1) WO2000038676A1 (tr)

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DK0883401T3 (da) * 1996-02-29 2003-05-05 Novartis Ag AT1-receptorantagonist til stimulering af apoptose
GB9613470D0 (en) * 1996-06-27 1996-08-28 Ciba Geigy Ag Small solid oral dosage form
DE19628617A1 (de) * 1996-07-16 1998-01-22 Basf Ag Direkttablettierhilfsmittel
NZ527598A (en) 1998-07-10 2005-04-29 Novartis Ag Antihypersensitive combination of valsartan and calcium channel blocker
SK10522001A3 (sk) 1999-01-26 2001-12-03 Novartis Ag Použitie antagonistov receptora angiotenzínu ii na liečenie akútneho infarktu myokardu
HUP0301390A3 (en) * 2000-06-22 2005-04-28 Novartis Ag Oral pharmaceutical composition containing valsartan
US20070123498A1 (en) 2003-10-17 2007-05-31 Shetty Suraj S Combination of organic compounds
JP2009018990A (ja) 2005-10-25 2009-01-29 Univ Kurume Ｃ型肝炎ウイルス由来ペプチド

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PL199100B1 (pl) 2008-08-29
ES2281978T3 (es) 2007-10-01
JP2010090169A (ja) 2010-04-22
IL143233A0 (en) 2002-04-21
CY1112395T1 (el) 2015-12-09
TR200605472T1 (tr) 2007-02-21
CY1106581T1 (el) 2012-01-25
CA2622805C (en) 2011-05-10
AU2006203077B2 (en) 2009-10-08
AU2009220022B2 (en) 2011-11-03
CZ20012306A3 (cs) 2001-12-12
SK9132001A3 (en) 2002-01-07
BR9916576A (pt) 2001-10-02
AU2003266433B2 (en) 2006-08-10
CN1331590A (zh) 2002-01-16
PT1140071E (pt) 2007-05-31
DE69935249D1 (de) 2007-04-05
CN1304000C (zh) 2007-03-14
NZ587909A (en) 2012-05-25
IL179017A0 (en) 2007-03-08
DE69935249T2 (de) 2007-10-31
CZ297795B6 (cs) 2007-03-28
AU2006203077A1 (en) 2006-08-10
ID29856A (id) 2001-10-18
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EP1140071B1 (en) 2007-02-21
EP1588706B1 (en) 2011-09-14
TR200101784T2 (tr) 2001-10-22
EP1588706A2 (en) 2005-10-26
SI1588706T1 (sl) 2012-01-31
AU2009220022A1 (en) 2009-10-15
WO2000038676A1 (en) 2000-07-06
IL143233A (en) 2007-07-24
DK1588706T3 (da) 2012-01-16
HUP0104780A2 (hu) 2002-04-29
CZ293257B6 (cs) 2004-03-17
IL179016A0 (en) 2007-03-08
CA2622805A1 (en) 2000-07-06
IL179015A0 (en) 2007-03-08
RU2361575C2 (ru) 2009-07-20
EP1140071A1 (en) 2001-10-10
SI1140071T1 (sl) 2007-08-31
PL349424A1 (en) 2002-07-29
EP2298298A2 (en) 2011-03-23
ATE524176T1 (de) 2011-09-15
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DK1140071T3 (da) 2007-06-04
RU2271809C2 (ru) 2006-03-20
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ATE354364T1 (de) 2007-03-15
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EP1588706A3 (en) 2005-12-07
TR200805275T2 (tr) 2008-09-22
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