TR199800027T1 - Difenilmetilen piperidin türevleri. - Google Patents

Difenilmetilen piperidin türevleri.

Info

Publication number
TR199800027T1
TR199800027T1 TR1998/00027T TR9800027T TR199800027T1 TR 199800027 T1 TR199800027 T1 TR 199800027T1 TR 1998/00027 T TR1998/00027 T TR 1998/00027T TR 9800027 T TR9800027 T TR 9800027T TR 199800027 T1 TR199800027 T1 TR 199800027T1
Authority
TR
Turkey
Prior art keywords
revleri
difenilmethylene
piperidin
pharmaceutically acceptable
acceptable salt
Prior art date
Application number
TR1998/00027T
Other languages
English (en)
Inventor
Robertson Rae Duncan
Robert Jaap David
Original Assignee
Akzo Nobel N.V
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel N.V filed Critical Akzo Nobel N.V
Publication of TR199800027T1 publication Critical patent/TR199800027T1/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Abstract

Bulus, terapide kullanim için, özelde, psikotik düzensizliklerin profilaksinda ya da iyilestirilmesinde bir dopamin antagonisti olarak kullanim için, (I) formülünün bir difenil-metilen türevine ya da bu türevin farmasötik olarak kabul edilebilir bir tuzuna iliskindir, bu formülde, n, 1 ya da 2'dir.
TR1998/00027T 1995-07-12 1996-07-09 Difenilmetilen piperidin türevleri. TR199800027T1 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP95201910 1995-07-12

Publications (1)

Publication Number Publication Date
TR199800027T1 true TR199800027T1 (tr) 1998-05-21

Family

ID=8220478

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1998/00027T TR199800027T1 (tr) 1995-07-12 1996-07-09 Difenilmetilen piperidin türevleri.

Country Status (27)

Country Link
US (1) US5935974A (tr)
EP (1) EP0842170B1 (tr)
JP (1) JPH11508907A (tr)
KR (1) KR19990028807A (tr)
CN (1) CN1091108C (tr)
AR (1) AR003966A1 (tr)
AT (1) ATE199150T1 (tr)
AU (1) AU699370B2 (tr)
BR (1) BR9609330A (tr)
CA (1) CA2226851A1 (tr)
CZ (1) CZ288909B6 (tr)
DE (1) DE69611788T2 (tr)
DK (1) DK0842170T3 (tr)
ES (1) ES2156287T3 (tr)
GR (1) GR3035849T3 (tr)
HK (1) HK1010818A1 (tr)
HU (1) HUP9802762A3 (tr)
IL (1) IL118768A (tr)
NO (1) NO309765B1 (tr)
NZ (1) NZ315318A (tr)
PL (1) PL183837B1 (tr)
PT (1) PT842170E (tr)
RU (1) RU2162846C2 (tr)
TR (1) TR199800027T1 (tr)
TW (1) TW419477B (tr)
WO (1) WO1997003065A1 (tr)
ZA (1) ZA965691B (tr)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999019324A2 (en) * 1997-10-07 1999-04-22 Akzo Nobel N.V. Antipsychotic substituted piperidine derivatives
AU2517499A (en) * 1998-01-09 1999-07-26 Akzo Nobel N.V. Use of diphenylmethylene piperidine derivatives in the manufacture of a medicament for the treatment of movement disorders
WO1999034801A1 (en) * 1998-01-09 1999-07-15 Akzo Nobel N.V. Use of diphenylmethylene piperidine derivatives in the manufacture of a medicament for the treatment of depression
US6432981B1 (en) 1999-06-11 2002-08-13 Merck & Co., Inc. Cyclopentyl modulators of chemokine receptor activity
US6538002B1 (en) 1999-06-11 2003-03-25 Merck & Co., Inc. Cyclopentyl modulators of chemokine receptor activity
WO2000076512A1 (en) 1999-06-11 2000-12-21 Merck & Co., Inc. Cyclopentyl modulators of chemokine receptor activity
US6358979B1 (en) 1999-06-11 2002-03-19 Merck & Co., Inc. N-cyclopentyl modulators of chemokine receptor activity
WO2000076513A1 (en) 1999-06-11 2000-12-21 Merck & Co., Inc. Cyclopentyl modulators of chemokine receptor activity
AU5328500A (en) 1999-06-11 2001-01-02 Merck & Co., Inc. N-cyclopentyl modulators of chemokine receptor activity
KR20010113007A (ko) * 2000-06-15 2001-12-24 주정호 항암제로서 유용한 ｎ-치환된 피페리디닐우레아 유도체 및그의 제조방법
TW200303304A (en) * 2002-02-18 2003-09-01 Astrazeneca Ab Chemical compounds
US6770659B2 (en) * 2002-08-26 2004-08-03 Sk Corporation Benzoyl piperidine compounds
MXPA05006427A (es) * 2002-12-18 2005-09-08 Fmc Corp Piperidinas y piridinas (arilmetilo sustituido)-n-4-(metilo disustituido).
SE0400208D0 (sv) * 2004-02-02 2004-02-02 Astrazeneca Ab Chemical compounds
TW200812582A (en) * 2006-04-06 2008-03-16 Astrazeneca Ab Medicaments
SG11201701315VA (en) 2014-08-28 2017-03-30 Asceneuron Sa Glycosidase inhibitors
WO2017106254A1 (en) * 2015-12-18 2017-06-22 Merck Sharp & Dohme Corp. Glycosidase inhibitors and uses thereof
CA3012560A1 (en) 2016-02-25 2017-08-31 Asceneuron S.A. Glycosidase inhibitors
US11261183B2 (en) 2016-02-25 2022-03-01 Asceneuron Sa Sulfoximine glycosidase inhibitors
US10556902B2 (en) 2016-02-25 2020-02-11 Asceneuron Sa Glycosidase inhibitors
EP3419976B1 (en) 2016-02-25 2021-04-07 Asceneuron SA Acid addition salts of piperazine derivatives
EP3672959A1 (en) 2017-08-24 2020-07-01 Asceneuron SA Linear glycosidase inhibitors
WO2020039028A1 (en) 2018-08-22 2020-02-27 Asceneuron S. A. Tetrahydro-benzoazepine glycosidase inhibitors
US11731972B2 (en) 2018-08-22 2023-08-22 Asceneuron Sa Spiro compounds as glycosidase inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US450780A (en) * 1891-04-21 Steam-engine
US4180583A (en) * 1972-01-28 1979-12-25 Richardson-Merrell Inc. Olefinic 4-substituted piperidino derivatives as therapeutics
US3922276A (en) * 1974-12-11 1975-11-25 Robins Co Inc A H 1-Substituted-4-benzylidenepiperidines
US4666905A (en) * 1983-06-02 1987-05-19 Warner-Lambert Company Diphenylmethylene piperidines compositions and methods for their use
US4540780A (en) * 1983-06-02 1985-09-10 Warner-Lambert Company Diphenylmethylene piperidines

Also Published As

Publication number Publication date
NZ315318A (en) 1999-10-28
IL118768A0 (en) 1996-10-31
PT842170E (pt) 2001-06-29
CN1190965A (zh) 1998-08-19
DE69611788D1 (de) 2001-03-22
AU699370B2 (en) 1998-12-03
ATE199150T1 (de) 2001-02-15
CZ288909B6 (cs) 2001-09-12
HUP9802762A2 (hu) 1999-10-28
PL183837B1 (pl) 2002-07-31
PL324451A1 (en) 1998-05-25
DK0842170T3 (da) 2001-06-18
HK1010818A1 (en) 1999-07-02
KR19990028807A (ko) 1999-04-15
EP0842170B1 (en) 2001-02-14
ZA965691B (en) 1997-01-24
CA2226851A1 (en) 1997-01-30
NO309765B1 (no) 2001-03-26
IL118768A (en) 2000-10-31
NO980109L (no) 1998-01-09
EP0842170A1 (en) 1998-05-20
TW419477B (en) 2001-01-21
AR003966A1 (es) 1998-09-30
AU6699396A (en) 1997-02-10
HUP9802762A3 (en) 2002-10-28
WO1997003065A1 (en) 1997-01-30
US5935974A (en) 1999-08-10
BR9609330A (pt) 1999-05-25
GR3035849T3 (en) 2001-08-31
NO980109D0 (no) 1998-01-09
CN1091108C (zh) 2002-09-18
MX9800368A (es) 1998-03-31
DE69611788T2 (de) 2001-08-02
RU2162846C2 (ru) 2001-02-10
ES2156287T3 (es) 2001-06-16
CZ8398A3 (cs) 1998-06-17
JPH11508907A (ja) 1999-08-03

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