TN2009000469A1 - Organic compounds - Google Patents
Organic compoundsInfo
- Publication number
- TN2009000469A1 TN2009000469A1 TNP2009000469A TN2009000469A TN2009000469A1 TN 2009000469 A1 TN2009000469 A1 TN 2009000469A1 TN P2009000469 A TNP2009000469 A TN P2009000469A TN 2009000469 A TN2009000469 A TN 2009000469A TN 2009000469 A1 TN2009000469 A1 TN 2009000469A1
- Authority
- TN
- Tunisia
- Prior art keywords
- organic compounds
- conditions
- blockade
- tautomers
- solvates
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07107654 | 2007-05-07 | ||
| PCT/EP2008/055497 WO2008135557A1 (fr) | 2007-05-07 | 2008-05-05 | Composés organiques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TN2009000469A1 true TN2009000469A1 (en) | 2011-03-31 |
Family
ID=38581916
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TNP2009000469A TN2009000469A1 (en) | 2007-05-07 | 2009-11-06 | Organic compounds |
Country Status (32)
| Country | Link |
|---|---|
| US (1) | US8318935B2 (fr) |
| EP (2) | EP2155721B1 (fr) |
| JP (1) | JP5244904B2 (fr) |
| KR (1) | KR20100005730A (fr) |
| CN (1) | CN101687851B (fr) |
| AR (1) | AR066458A1 (fr) |
| AT (1) | ATE499363T1 (fr) |
| AU (1) | AU2008248598B2 (fr) |
| BR (1) | BRPI0811562A2 (fr) |
| CA (1) | CA2685546A1 (fr) |
| CL (1) | CL2008001301A1 (fr) |
| CO (1) | CO6290667A2 (fr) |
| CR (1) | CR11091A (fr) |
| DE (1) | DE602008005140D1 (fr) |
| EA (1) | EA200901489A1 (fr) |
| EC (1) | ECSP099718A (fr) |
| ES (1) | ES2361595T3 (fr) |
| GT (1) | GT200900289A (fr) |
| HK (1) | HK1141285A1 (fr) |
| HN (1) | HN2009003214A (fr) |
| IL (1) | IL201828A0 (fr) |
| MA (1) | MA31400B1 (fr) |
| MX (1) | MX2009012077A (fr) |
| NZ (1) | NZ580737A (fr) |
| PE (1) | PE20090733A1 (fr) |
| PL (1) | PL2155721T3 (fr) |
| PT (1) | PT2155721E (fr) |
| SV (1) | SV2009003406A (fr) |
| TN (1) | TN2009000469A1 (fr) |
| TW (1) | TWI351402B (fr) |
| WO (1) | WO2008135557A1 (fr) |
| ZA (1) | ZA200907491B (fr) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6858615B2 (en) | 2002-02-19 | 2005-02-22 | Parion Sciences, Inc. | Phenyl guanidine sodium channel blockers |
| WO2009139948A1 (fr) | 2008-02-26 | 2009-11-19 | Johnson Michael R | Bloqueurs poly-aromatiques de canaux sodiques |
| KR20110085768A (ko) | 2010-01-21 | 2011-07-27 | 삼성전자주식회사 | Ｃｍｏｓ 이미지 센서, 상기 이미지 센서의 데이터 리드아웃 방법, 및 상기 이미지 센서를 포함하는 전자 시스템 |
| US8372845B2 (en) * | 2010-09-17 | 2013-02-12 | Novartis Ag | Pyrazine derivatives as enac blockers |
| US9050339B2 (en) | 2010-09-17 | 2015-06-09 | Novartis Ag | Pyrazine derivatives as ENaC blockers |
| AR086745A1 (es) | 2011-06-27 | 2014-01-22 | Parion Sciences Inc | 3,5-diamino-6-cloro-n-(n-(4-(4-(2-(hexil(2,3,4,5,6-pentahidroxihexil)amino)etoxi)fenil)butil)carbamimidoil)pirazina-2-carboxamida |
| NO2773633T3 (fr) * | 2011-11-02 | 2017-12-30 | ||
| JP2015501324A (ja) * | 2011-11-02 | 2015-01-15 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | アシルグアニジン及びアシルチオ尿素の新規調製方法 |
| US8859559B2 (en) | 2011-12-20 | 2014-10-14 | Boehringer Ingelheim International Gmbh | Substituted pyrazines and their use in the treatment of disease |
| CA2863224A1 (fr) | 2012-01-09 | 2013-07-18 | The Scripps Research Institute | Regions determinant la complementarite ultralongues et utilisations associees |
| WO2013174757A1 (fr) | 2012-05-25 | 2013-11-28 | Boehringer Ingelheim International Gmbh | Amines tertiaires, médicaments contenant lesdites amines, leur utilisation et leurs procédés de préparation |
| WO2014044849A1 (fr) | 2012-09-24 | 2014-03-27 | Boehringer Ingelheim International Gmbh | Composés hétérocycliques, médicaments contenant ces composés, leur utilisation et procédés de leur préparation |
| MX368353B (es) | 2012-11-02 | 2019-09-30 | Vertex Pharma | Composiciones farmaceuticas para el tratamiento de enfermedades mediadas por cftr. |
| US9029382B2 (en) | 2012-12-17 | 2015-05-12 | Parion Sciences, Inc. | 3,5-diamino-6-chloro-N-(N-(4-phenylbutyl)carbamimidoyl) pyrazine-2-carboxamide compounds |
| EP3150585A1 (fr) | 2012-12-17 | 2017-04-05 | Parion Sciences, Inc. | Dérivés de carboxamide de chloro-pyrazine avec une activité de blocage de canal de sodium épithélial |
| JP6353032B2 (ja) * | 2013-04-30 | 2018-07-04 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ジアミノピラジン化合物、前記化合物を含有する医薬、その使用、およびその調製方法 |
| US9656972B2 (en) | 2013-07-02 | 2017-05-23 | The California Institute For Biomedical Research | Compounds for treatment of cystic fibrosis |
| US9102633B2 (en) | 2013-12-13 | 2015-08-11 | Parion Sciences, Inc. | Arylalkyl- and aryloxyalkyl-substituted epithelial sodium channel blocking compounds |
| UY36034A (es) | 2014-03-18 | 2015-09-30 | Astrazeneca Ab | Derivados de 3,5-diamino-6-cloro-pirazina-2-carboxamida y sales farmaceuticamente aceptables de estos |
| CA2940599A1 (fr) | 2014-03-27 | 2015-10-01 | Novartis Ag | Dispersions d'huile-dans-l'eau solides sechees par pulverisation pour l'inhalation de principes pharmaceutiques actifs |
| GB201412545D0 (en) * | 2014-07-15 | 2014-08-27 | Univ Manchester The And Manchester Metropolitan University | Enzymatic processes and uses |
| WO2016112120A1 (fr) * | 2015-01-07 | 2016-07-14 | The California Institute For Biomedical Research | Composés destinés au traitement de la mucosviscidose |
| JP6671378B2 (ja) * | 2015-01-12 | 2020-03-25 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 呼吸器系疾患の治療に有用な置換ベンズイミダゾリウム化合物 |
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| US10291868B2 (en) * | 2016-01-29 | 2019-05-14 | SK Hynix Inc. | Image sensing device |
| GB201610854D0 (en) | 2016-06-21 | 2016-08-03 | Entpr Therapeutics Ltd | Compounds |
| GB201619694D0 (en) | 2016-11-22 | 2017-01-04 | Entpr Therapeutics Ltd | Compounds |
| WO2018175302A1 (fr) | 2017-03-20 | 2018-09-27 | Sienna Biopharmaceuticals, Inc. | Conjugués polymères ciblant c-src à exposition réduite |
| EP3600440A1 (fr) | 2017-03-20 | 2020-02-05 | Sienna Biopharmaceuticals, Inc. | Conjugués d'exposition réduite modulant des cibles thérapeutiques |
| GB201717051D0 (en) | 2017-10-17 | 2017-11-29 | Enterprise Therapeutics Ltd | Compounds |
| GB201808093D0 (en) | 2018-05-18 | 2018-07-04 | Enterprise Therapeutics Ltd | Compounds |
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- 2008-05-05 BR BRPI0811562-1A2A patent/BRPI0811562A2/pt not_active IP Right Cessation
- 2008-05-05 AT AT08759419T patent/ATE499363T1/de active
- 2008-05-05 US US12/451,152 patent/US8318935B2/en not_active Expired - Fee Related
- 2008-05-05 MX MX2009012077A patent/MX2009012077A/es active IP Right Grant
- 2008-05-05 EP EP08759419A patent/EP2155721B1/fr active Active
- 2008-05-05 PL PL08759419T patent/PL2155721T3/pl unknown
- 2008-05-05 DE DE602008005140T patent/DE602008005140D1/de active Active
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- 2008-05-05 JP JP2010506915A patent/JP5244904B2/ja not_active Expired - Fee Related
- 2008-05-05 EA EA200901489A patent/EA200901489A1/ru unknown
- 2008-05-05 CA CA002685546A patent/CA2685546A1/fr not_active Abandoned
- 2008-05-05 WO PCT/EP2008/055497 patent/WO2008135557A1/fr active Application Filing
- 2008-05-05 AU AU2008248598A patent/AU2008248598B2/en not_active Ceased
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- 2008-05-05 CN CN2008800226814A patent/CN101687851B/zh not_active Expired - Fee Related
- 2008-05-05 EP EP11152559A patent/EP2332933A1/fr not_active Withdrawn
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