HUP0300832A2 - Új, lassú hatású bétamimetikumok, eljárás előállításukra és alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények - Google Patents

Új, lassú hatású bétamimetikumok, eljárás előállításukra és alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények

Info

Publication number
HUP0300832A2
HUP0300832A2 HU0300832A HUP0300832A HUP0300832A2 HU P0300832 A2 HUP0300832 A2 HU P0300832A2 HU 0300832 A HU0300832 A HU 0300832A HU P0300832 A HUP0300832 A HU P0300832A HU P0300832 A2 HUP0300832 A2 HU P0300832A2
Authority
HU
Hungary
Prior art keywords
group
production
medicaments
slow
novel
Prior art date
Application number
HU0300832A
Other languages
English (en)
Inventor
Karl-Heinz Bozung
Hermann Schollenberger
Kurt Schromm
Alexander Walland
Original Assignee
Boehringer Ingelheim Pharma Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from ECSP003424 external-priority patent/ECSP003424A/es
Priority claimed from DE2000151318 external-priority patent/DE10051318A1/de
Application filed by Boehringer Ingelheim Pharma Gmbh & Co. Kg filed Critical Boehringer Ingelheim Pharma Gmbh & Co. Kg
Publication of HUP0300832A2 publication Critical patent/HUP0300832A2/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06—Antiabortive agents; Labour repressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • H—ELECTRICITY
    • H03—ELECTRONIC CIRCUITRY
    • H03F—AMPLIFIERS
    • H03F2200/00—Indexing scheme relating to amplifiers
    • H03F2200/331—Sigma delta modulation being used in an amplifying circuit

Abstract

A találmány tárgyát az általános képletű vegyületek - ahol R1 egy általános képletű csoport, amelyben R3 adott esetben metoxi-szubsztituált benzilcsoport; R4 hidrogénatom; vagy R3 és R4 együtt egy-CO-CH2-O- képletű hidat képez, ahol a híd karbonilcsoport anitrogénatomhoz kapcsolódik; R2 az általános képletű csoportok közülválasztott csoport, amelyben R5 dimetil-amino-, metoxi- vagybutoxicsoport; X nitrogén- vagy szénatom; R6 metoxi-fenil-csoport,amennyiben X jelentése nitrogénatom; vagy szintén az X-hez kapcsolódóanellált fenilcsoport, amennyiben X jelentése szénatom - éselőállításuk és alkalmazásuk képezik. Ó
HU0300832A 2000-04-27 2001-04-14 Új, lassú hatású bétamimetikumok, eljárás előállításukra és alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények HUP0300832A2 (hu)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ECSP003424 ECSP003424A (es) 2000-04-27 2000-04-27 NUEVAS COMPOSICIONES DE MEDICAMENTOS A BASE DE COMPUESTOS ANTICOLINERGICAMENTE ACTIVOS Y ß-MIMETICOS
DE2000151318 DE10051318A1 (de) 2000-10-17 2000-10-17 Neu, langwirksame Betamimetika, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
PCT/EP2001/004278 WO2001083462A1 (de) 2000-04-27 2001-04-14 Neue, langwirksame betamimetika, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
HUP0300832A2 true HUP0300832A2 (hu) 2003-08-28

Family

ID=40317111

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0300832A HUP0300832A2 (hu) 2000-04-27 2001-04-14 Új, lassú hatású bétamimetikumok, eljárás előállításukra és alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények

Country Status (23)

Country Link
US (2) US20020022625A1 (hu)
EP (1) EP1305300A1 (hu)
JP (1) JP2003533448A (hu)
KR (1) KR20020093083A (hu)
CN (1) CN1426401A (hu)
AR (1) AR035637A1 (hu)
AU (1) AU5629301A (hu)
BG (1) BG107120A (hu)
BR (1) BR0110331A (hu)
CA (1) CA2405745A1 (hu)
CZ (1) CZ20023537A3 (hu)
EA (1) EA200201056A1 (hu)
EE (1) EE200200602A (hu)
HR (1) HRP20020845A2 (hu)
HU (1) HUP0300832A2 (hu)
IL (1) IL152140A0 (hu)
MX (1) MXPA02010179A (hu)
NO (1) NO20025133L (hu)
NZ (1) NZ522677A (hu)
PL (1) PL362868A1 (hu)
SK (1) SK15382002A3 (hu)
WO (1) WO2001083462A1 (hu)
YU (1) YU79502A (hu)

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Also Published As

Publication number Publication date
NO20025133D0 (no) 2002-10-25
SK15382002A3 (sk) 2003-03-04
CA2405745A1 (en) 2001-11-08
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US20020022625A1 (en) 2002-02-21
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CN1426401A (zh) 2003-06-25
AU5629301A (en) 2001-11-12
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EE200200602A (et) 2004-04-15
WO2001083462A1 (de) 2001-11-08
YU79502A (sh) 2006-05-25
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BG107120A (en) 2003-05-30
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