SK53699A3 - 6-{3-[4-(fluorobenzyle)-piperidine-1-yl]-propionyl}-3h- -benzoxazole-2-one, method for its preparation, its use and pharmaceutical composition containing the same - Google Patents
6-{3-[4-(fluorobenzyle)-piperidine-1-yl]-propionyl}-3h- -benzoxazole-2-one, method for its preparation, its use and pharmaceutical composition containing the same Download PDFInfo
- Publication number
- SK53699A3 SK53699A3 SK536-99A SK53699A SK53699A3 SK 53699 A3 SK53699 A3 SK 53699A3 SK 53699 A SK53699 A SK 53699A SK 53699 A3 SK53699 A3 SK 53699A3
- Authority
- SK
- Slovakia
- Prior art keywords
- formula
- compound
- physiologically acceptable
- propionyl
- acceptable salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19643790A DE19643790A1 (de) | 1996-10-30 | 1996-10-30 | Benzoxazol-Derivat |
| PCT/EP1997/005590 WO1998018793A1 (de) | 1996-10-30 | 1997-10-10 | Benzoxazolderivat mit affinität zu bindungsstellen von aminosäurerezeptoren |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK53699A3 true SK53699A3 (en) | 2000-03-13 |
Family
ID=7809592
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK536-99A SK53699A3 (en) | 1996-10-30 | 1997-10-10 | 6-{3-[4-(fluorobenzyle)-piperidine-1-yl]-propionyl}-3h- -benzoxazole-2-one, method for its preparation, its use and pharmaceutical composition containing the same |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP0938485A1 (ko) |
| JP (1) | JP2001502713A (ko) |
| KR (1) | KR20000052876A (ko) |
| CN (1) | CN1235604A (ko) |
| AR (1) | AR008512A1 (ko) |
| AU (1) | AU4946597A (ko) |
| BR (1) | BR9712577A (ko) |
| CA (1) | CA2270359A1 (ko) |
| CZ (1) | CZ147999A3 (ko) |
| DE (1) | DE19643790A1 (ko) |
| HU (1) | HUP9904547A3 (ko) |
| NO (1) | NO992063L (ko) |
| PL (1) | PL332771A1 (ko) |
| SK (1) | SK53699A3 (ko) |
| WO (1) | WO1998018793A1 (ko) |
| ZA (1) | ZA979725B (ko) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9725541D0 (en) * | 1997-12-02 | 1998-02-04 | Pharmacia & Upjohn Spa | Amino-benzothiazole derivatives |
| DE19812331A1 (de) * | 1998-03-20 | 1999-09-23 | Merck Patent Gmbh | Piperidinderivate |
| PE20000728A1 (es) | 1998-06-26 | 2000-08-21 | Cocensys Inc | Heterociclos 4-bencil piperidina alquilsulfoxido y su uso como antagonistas receptores subtipo-selectivo nmda |
| US6476041B1 (en) | 1999-10-29 | 2002-11-05 | Merck & Co., Inc. | 1,4 substituted piperidinyl NMDA/NR2B antagonists |
| EP1674087A1 (en) | 2000-10-02 | 2006-06-28 | Pfizer Products Inc. | Prophylactic use of n-methyl-d-aspartate (NMDA) antagonists |
| DE10120159A1 (de) * | 2001-04-25 | 2002-10-31 | Merck Patent Gmbh | NMDA-Antagonisten und NMDA-Agonisten zur Behandlung von Suchterkrankungen |
| SI1409477T1 (sl) | 2001-07-24 | 2009-02-28 | Richter Gedeon Nyrt | Derivati piperidina kot antagonisti nmda-receptorjev |
| DE102007047737A1 (de) * | 2007-10-05 | 2009-04-30 | Merck Patent Gmbh | Piperidin- und Piperazinderivate |
| DE102009049211A1 (de) | 2009-10-13 | 2011-04-28 | Merck Patent Gmbh | Sulfoxide |
| CN103974698A (zh) | 2011-11-22 | 2014-08-06 | 加利福尼亚大学董事会 | 用于治疗缺血性损伤的半胱胺和/或胱胺 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK0709384T3 (da) * | 1994-10-31 | 1999-08-23 | Merck Patent Gmbh | Benzylpiperidinderivater med høj affinitet til aminosyrereceptorers bindingssteder |
-
1996
- 1996-10-30 DE DE19643790A patent/DE19643790A1/de not_active Withdrawn
-
1997
- 1997-10-10 CN CN97199279A patent/CN1235604A/zh active Pending
- 1997-10-10 AU AU49465/97A patent/AU4946597A/en not_active Abandoned
- 1997-10-10 HU HU9904547A patent/HUP9904547A3/hu unknown
- 1997-10-10 KR KR1019990703727A patent/KR20000052876A/ko not_active Application Discontinuation
- 1997-10-10 CA CA002270359A patent/CA2270359A1/en not_active Abandoned
- 1997-10-10 WO PCT/EP1997/005590 patent/WO1998018793A1/de not_active Application Discontinuation
- 1997-10-10 BR BR9712577-6A patent/BR9712577A/pt not_active Application Discontinuation
- 1997-10-10 EP EP97912162A patent/EP0938485A1/de not_active Withdrawn
- 1997-10-10 CZ CZ991479A patent/CZ147999A3/cs unknown
- 1997-10-10 SK SK536-99A patent/SK53699A3/sk unknown
- 1997-10-10 PL PL97332771A patent/PL332771A1/xx unknown
- 1997-10-10 JP JP10519971A patent/JP2001502713A/ja active Pending
- 1997-10-29 ZA ZA9709725A patent/ZA979725B/xx unknown
- 1997-10-29 AR ARP970105012A patent/AR008512A1/es unknown
-
1999
- 1999-04-29 NO NO992063A patent/NO992063L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA979725B (en) | 1998-05-22 |
| BR9712577A (pt) | 1999-10-19 |
| EP0938485A1 (de) | 1999-09-01 |
| PL332771A1 (en) | 1999-10-11 |
| CN1235604A (zh) | 1999-11-17 |
| NO992063D0 (no) | 1999-04-29 |
| JP2001502713A (ja) | 2001-02-27 |
| CZ147999A3 (cs) | 1999-08-11 |
| HUP9904547A3 (en) | 2001-01-29 |
| CA2270359A1 (en) | 1998-05-07 |
| AR008512A1 (es) | 2000-01-19 |
| KR20000052876A (ko) | 2000-08-25 |
| WO1998018793A1 (de) | 1998-05-07 |
| HUP9904547A2 (hu) | 2000-12-28 |
| DE19643790A1 (de) | 1998-05-07 |
| NO992063L (no) | 1999-04-29 |
| AU4946597A (en) | 1998-05-22 |
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