SI9720045B - Azolo triazini in pirimidini - Google Patents

Azolo triazini in pirimidini Download PDF

Info

Publication number
SI9720045B
SI9720045B SI9720045A SI9720045A SI9720045B SI 9720045 B SI9720045 B SI 9720045B SI 9720045 A SI9720045 A SI 9720045A SI 9720045 A SI9720045 A SI 9720045A SI 9720045 B SI9720045 B SI 9720045B
Authority
SI
Slovenia
Prior art keywords
formula
compounds
alkyl
nhch
cycloalkyl
Prior art date
Application number
SI9720045A
Other languages
English (en)
Slovenian (sl)
Other versions
SI9720045A (sl
Inventor
Argyrios Georgious Arvanitis
Robert John Chorvat
Liqi He
Paul Joseph Giligan
Original Assignee
Bristol Myers Squibb Pharma Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Pharma Co filed Critical Bristol Myers Squibb Pharma Co
Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en
Priority claimed from US08/899,242 external-priority patent/US6124289A/en
Publication of SI9720045A publication Critical patent/SI9720045A/sl
Publication of SI9720045B publication Critical patent/SI9720045B/sl

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Detergent Compositions (AREA)
  • Coloring (AREA)
SI9720045A 1996-07-24 1997-07-23 Azolo triazini in pirimidini SI9720045B (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US68604796A 1996-07-24 1996-07-24
US2329096P 1996-07-24 1996-07-24
PCT/US1997/013072 WO1998003510A1 (en) 1996-07-24 1997-07-23 AZOLO TRIAZINES AND PYRIMIDINES
US08/899,242 US6124289A (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines

Publications (2)

Publication Number Publication Date
SI9720045A SI9720045A (sl) 1999-10-31
SI9720045B true SI9720045B (sl) 2008-02-29

Family

ID=27362048

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9720045A SI9720045B (sl) 1996-07-24 1997-07-23 Azolo triazini in pirimidini

Country Status (15)

Country Link
JP (2) JP4704521B2 (zh)
CN (3) CN1104432C (zh)
AR (1) AR049583A2 (zh)
BR (1) BR9710544A (zh)
CA (1) CA2259583C (zh)
CZ (1) CZ299451B6 (zh)
EA (1) EA004403B1 (zh)
EE (1) EE04316B1 (zh)
HR (1) HRP970413A2 (zh)
IL (4) IL127871A0 (zh)
NO (1) NO315610B3 (zh)
NZ (1) NZ333777A (zh)
PL (1) PL195762B1 (zh)
SI (1) SI9720045B (zh)
SK (1) SK286461B6 (zh)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002072202A1 (en) * 2001-03-13 2002-09-19 Bristol-Myers Squibb Pharma Company 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands
WO2004110454A1 (ja) * 2003-06-13 2004-12-23 Ishihara Sangyo Kaisha, Ltd. アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物
US7329662B2 (en) * 2003-10-03 2008-02-12 Hoffmann-La Roche Inc. Pyrazolo-pyridine
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
DK2094709T3 (da) * 2006-09-20 2010-12-06 Lilly Co Eli Thiazol-pyrazolopyrimidiner som CRF1-receptorantagonister
CN103694242B (zh) * 2013-12-10 2016-01-06 昆明翔昊科技有限公司 吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用
EP3628005A4 (en) 2017-08-14 2021-01-20 Spruce Biosciences, Inc. CORTICOTROPIN RELEASE FACTOR RECEPTOR ANTAGONISTS
CN112479956A (zh) * 2019-07-30 2021-03-12 杭州阿诺生物医药科技有限公司 一种用于制备腺苷受体抑制剂中间体的方法
WO2022036123A1 (en) 2020-08-12 2022-02-17 Spruce Biosciences, Inc. Methods and compositions for treating polycystic ovary syndrome
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3995039A (en) * 1975-05-27 1976-11-30 Merck & Co., Inc. Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (ja) * 1984-08-29 1986-03-24 Shionogi & Co Ltd 縮合複素環誘導体および抗潰瘍剤
US4824834A (en) * 1986-10-31 1989-04-25 Otsuka Pharmaceutical Company, Limited Pyrazolotriazine compounds
JP2691317B2 (ja) * 1989-08-25 1997-12-17 株式会社大塚製薬工場 ４―ヒドロキシ―８―（３―低級アルコキシ―４―フェニルスルフィニルフェニル）ピラゾロ〔１，５―ａ〕―１，３，５―トリアジン光学活性体の塩類及びその製造方法
US5420128A (en) * 1990-10-09 1995-05-30 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor
DE69130683T2 (de) * 1991-04-22 1999-05-06 Otsuka Pharmaceutical Factory, Inc., Naruto, Tokushima PYRAZOLO[1,5-a]PYRIMIDINDERIVATE UND SIE ENTHALTENDE ANTIINFLAMMATORISCHE MITTEL
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

Also Published As

Publication number Publication date
NZ333777A (en) 2000-07-28
HRP970413A2 (en) 1998-10-31
IL164513A0 (en) 2005-12-18
CN1250223C (zh) 2006-04-12
CZ18499A3 (cs) 1999-11-17
IL127871A (en) 2010-04-29
JP2005097257A (ja) 2005-04-14
IL127871A0 (en) 1999-10-28
SK9799A3 (sk) 2005-04-01
EE04316B1 (et) 2004-06-15
NO315610B1 (no) 2003-09-29
SI9720045A (sl) 1999-10-31
EA199900158A1 (ru) 1999-10-28
NO990264L (no) 1999-03-10
CN1327793A (zh) 2001-12-26
CZ299451B6 (cs) 2008-07-30
CN1225637A (zh) 1999-08-11
JP4194539B2 (ja) 2008-12-10
NO315610B3 (no) 2003-09-29
EE9900019A (et) 1999-08-16
EA004403B1 (ru) 2004-04-29
JP2002513382A (ja) 2002-05-08
AR049583A2 (es) 2006-08-16
SK286461B6 (sk) 2008-10-07
IL164513A (en) 2010-04-29
NO990264D0 (no) 1999-01-21
PL195762B1 (pl) 2007-10-31
CN1388126A (zh) 2003-01-01
IL150163A (en) 2010-12-30
BR9710544A (pt) 1999-08-17
CN1104432C (zh) 2003-04-02
PL331523A1 (en) 1999-07-19
JP4704521B2 (ja) 2011-06-15
CA2259583A1 (en) 1998-01-29
CA2259583C (en) 2009-11-17

Similar Documents

Publication Publication Date Title
ES2289475T3 (es) Derivados de l-aminotieno(2,3-d)pirimidina-6-carbonitrilo como inhibidores de pde7.
CA2588761C (en) 2,4(4,6)pyrimidine derivatives
ES2291628T3 (es) Compuestos triciclicos a base de tiofeno y composiciones farmaceuticas que comprenden dichos compuestos.
ES2330789T3 (es) Anilino-piridinotriazinas ciclicas como inhibidores de gsk-3.
DE60101158T2 (de) 8-chinolinxanthin and 8-isochinolinxanthin derivate als pde 5 inhibitoren
ES2221679T3 (es) Derivados de diamino-1,3,5-triazina sustituidos.
SI9720045B (sl) Azolo triazini in pirimidini
Taylor et al. Pyrimido [4, 5-d] pyrimidines. Part I
HRP20170317T1 (hr) Spojevi pirimidin-2-amina i njihova uporaba kao inhibitora jak kinaza
CA3118908A1 (en) Pyridazinone compounds and uses thereof
AU2011336764A1 (en) Novel compounds as respiratory stimulants for treatment of breathing control disorders or diseases
NZ603896A (en) 3-amino-5,6-dihydro-1h-pyrazin-2-one derivatives useful for the treatement of alzheimer's disease and other forms of dementia
ATE162521T1 (de) 3-aminopiperidine derivate und verwandete stickstoff enthaltende heterocyclische verbindungen
HUP0202810A2 (hu) Szubsztituált 2-tio-3.5-diciano-4-aril-6-aminopiridinek és eljárás az előállításukra, valamint ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk
CA3085333A1 (en) Substituted indole ether compounds
IL102367A (en) Triazolopyrimidine derivatives which are angiotensin ii receptor antagonists, processes for preparing them and pharmaceutical compositions containing them
HUT62582A (en) Process for producing pyrimidine nucleoside derivatives and pharmaceutical compositions comprising same as active ingredient
CA1320203C (en) Intermediates for 9-deazaguanines
CA1260934A (en) Purine derivatives
Roth et al. 2, 4-Diamino-5-benzylpyrimidines as antibacterial agents. 4. 6-Substituted trimethoprim derivatives from phenolic Mannich intermediates. Application to the synthesis of trimethoprim and 3, 5-dialkylbenzyl analogs
WO2022064458A1 (en) Indazoles as hematopoietic progenitor kinase 1 (hpk1) inhibitors and methods of using same
CA1294960C (en) 7-deazaguanines as immunomodulators
US4921858A (en) 7-deazaguanines as immunomodulators
EP4426704A1 (en) Condensed pyridazine amine derivatives treating sca3
DE69029547T2 (de) Purinverbindungen, Verfahren zu ihrer Herstellung, pharmazeutische Präparate und Zwischenverbindungen

Legal Events

Date Code Title Description
IF Valid on the event date
OU02 Decision according to article 73(2) ipa 1992, publication of decision on partial fulfilment of the invention and change of patent claims

Effective date: 20080108