NO315610B3 - Azolotriaziner og -pyrimidiner - Google Patents

Azolotriaziner og -pyrimidiner

Info

Publication number
NO315610B3
NO315610B3 NO19990264A NO990264A NO315610B3 NO 315610 B3 NO315610 B3 NO 315610B3 NO 19990264 A NO19990264 A NO 19990264A NO 990264 A NO990264 A NO 990264A NO 315610 B3 NO315610 B3 NO 315610B3
Authority
NO
Norway
Prior art keywords
azolotriazines
pyrimidines
Prior art date
Application number
NO19990264A
Other languages
English (en)
Norwegian (no)
Other versions
NO990264D0 (no
NO990264L (no
NO315610B1 (no
Inventor
Argyrios Georgios Arvanitis
Robert John Chorvat
Paul Joseph Gilligan
Liqi He
Original Assignee
Du Pont Pharm Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en
Priority claimed from US08/899,242 external-priority patent/US6124289A/en
Application filed by Du Pont Pharm Co filed Critical Du Pont Pharm Co
Publication of NO990264D0 publication Critical patent/NO990264D0/no
Publication of NO990264L publication Critical patent/NO990264L/no
Publication of NO315610B3 publication Critical patent/NO315610B3/no
Publication of NO315610B1 publication Critical patent/NO315610B1/no

Links

NO19990264A 1996-07-24 1999-01-21 Azolotriaziner og -pyrimidiner NO315610B1 (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US2329096P 1996-07-24 1996-07-24
US68604796A 1996-07-24 1996-07-24
PCT/US1997/013072 WO1998003510A1 (en) 1996-07-24 1997-07-23 AZOLO TRIAZINES AND PYRIMIDINES
US08/899,242 US6124289A (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines

Publications (4)

Publication Number Publication Date
NO990264D0 NO990264D0 (no) 1999-01-21
NO990264L NO990264L (no) 1999-03-10
NO315610B3 true NO315610B3 (no) 2003-09-29
NO315610B1 NO315610B1 (no) 2003-09-29

Family

ID=27362048

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19990264A NO315610B1 (no) 1996-07-24 1999-01-21 Azolotriaziner og -pyrimidiner

Country Status (15)

Country Link
JP (2) JP4704521B2 (zh)
CN (3) CN1104432C (zh)
AR (1) AR049583A2 (zh)
BR (1) BR9710544A (zh)
CA (1) CA2259583C (zh)
CZ (1) CZ299451B6 (zh)
EA (1) EA004403B1 (zh)
EE (1) EE04316B1 (zh)
HR (1) HRP970413A2 (zh)
IL (4) IL127871A0 (zh)
NO (1) NO315610B1 (zh)
NZ (1) NZ333777A (zh)
PL (1) PL195762B1 (zh)
SI (1) SI9720045B (zh)
SK (1) SK286461B6 (zh)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA03008185A (es) * 2001-03-13 2004-01-29 Bristol Myers Squibb Pharma Co 4-(2-butilamino)-2, 7-dimetil-8 -(2-metil-6-metoxipirid -3-il) pirazol-[1, 5-a]-1, 3, 5-triazina, sus enantiomeros y sales farmaceuticamente aceptables como ligandos del receptor del factor de liberacion de corticotropina.
WO2004110454A1 (ja) * 2003-06-13 2004-12-23 Ishihara Sangyo Kaisha, Ltd. アデノシンA2a受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物
US7329662B2 (en) * 2003-10-03 2008-02-12 Hoffmann-La Roche Inc. Pyrazolo-pyridine
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
MX2009003125A (es) * 2006-09-20 2009-05-28 Lilly Co Eli Tiazol pirazolopirimidinas como antagonistas de receptor de crf1.
CN103694242B (zh) * 2013-12-10 2016-01-06 昆明翔昊科技有限公司 吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用
CN112592346B (zh) * 2019-07-30 2022-04-26 厦门宝太生物科技股份有限公司 一种a2a和/或a2b抑制剂中间体的制备方法
CN116322544A (zh) 2020-08-12 2023-06-23 云杉生物科学公司 用于治疗多囊卵巢综合征的方法和组合物
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3995039A (en) * 1975-05-27 1976-11-30 Merck & Co., Inc. Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (ja) * 1984-08-29 1986-03-24 Shionogi & Co Ltd 縮合複素環誘導体および抗潰瘍剤
US4824834A (en) * 1986-10-31 1989-04-25 Otsuka Pharmaceutical Company, Limited Pyrazolotriazine compounds
JP2691317B2 (ja) * 1989-08-25 1997-12-17 株式会社大塚製薬工場 4―ヒドロキシ―8―(3―低級アルコキシ―4―フェニルスルフィニルフェニル)ピラゾロ〔1,5―a〕―1,3,5―トリアジン光学活性体の塩類及びその製造方法
AU639615B2 (en) * 1990-10-09 1993-07-29 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivative, production thereof, and androgen inhibitor
ATE174917T1 (de) * 1991-04-22 1999-01-15 Otsuka Pharma Co Ltd Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

Also Published As

Publication number Publication date
JP4194539B2 (ja) 2008-12-10
AR049583A2 (es) 2006-08-16
SK286461B6 (sk) 2008-10-07
IL150163A (en) 2010-12-30
CN1104432C (zh) 2003-04-02
PL195762B1 (pl) 2007-10-31
EE9900019A (et) 1999-08-16
NZ333777A (en) 2000-07-28
NO990264D0 (no) 1999-01-21
EA004403B1 (ru) 2004-04-29
CZ18499A3 (cs) 1999-11-17
SI9720045B (sl) 2008-02-29
NO990264L (no) 1999-03-10
EE04316B1 (et) 2004-06-15
IL164513A (en) 2010-04-29
BR9710544A (pt) 1999-08-17
IL127871A (en) 2010-04-29
SI9720045A (sl) 1999-10-31
CN1250223C (zh) 2006-04-12
CN1225637A (zh) 1999-08-11
CA2259583A1 (en) 1998-01-29
HRP970413A2 (en) 1998-10-31
IL127871A0 (en) 1999-10-28
JP2005097257A (ja) 2005-04-14
CZ299451B6 (cs) 2008-07-30
NO315610B1 (no) 2003-09-29
EA199900158A1 (ru) 1999-10-28
JP2002513382A (ja) 2002-05-08
CA2259583C (en) 2009-11-17
CN1388126A (zh) 2003-01-01
SK9799A3 (sk) 2005-04-01
IL164513A0 (en) 2005-12-18
CN1327793A (zh) 2001-12-26
JP4704521B2 (ja) 2011-06-15
PL331523A1 (en) 1999-07-19

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