IL150163A - PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS - Google Patents

PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS

Info

Publication number
IL150163A
IL150163A IL150163A IL15016302A IL150163A IL 150163 A IL150163 A IL 150163A IL 150163 A IL150163 A IL 150163A IL 15016302 A IL15016302 A IL 15016302A IL 150163 A IL150163 A IL 150163A
Authority
IL
Israel
Prior art keywords
pyrazolo
novel
compounds
pharmaceutical compositions
pyrimidine derivatives
Prior art date
Application number
IL150163A
Original Assignee
Du Pont Pharm Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en
Priority claimed from US08/899,242 external-priority patent/US6124289A/en
Application filed by Du Pont Pharm Co filed Critical Du Pont Pharm Co
Publication of IL150163A publication Critical patent/IL150163A/en

Links

IL150163A 1996-07-24 2002-06-11 PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS IL150163A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US68604796A 1996-07-24 1996-07-24
US2329096P 1996-07-24 1996-07-24
PCT/US1997/013072 WO1998003510A1 (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines
US08/899,242 US6124289A (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines

Publications (1)

Publication Number Publication Date
IL150163A true IL150163A (en) 2010-12-30

Family

ID=27362048

Family Applications (4)

Application Number Title Priority Date Filing Date
IL12787197A IL127871A0 (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines
IL127871A IL127871A (en) 1996-07-24 1998-12-30 PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES
IL150163A IL150163A (en) 1996-07-24 2002-06-11 PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS
IL164513A IL164513A (en) 1996-07-24 2004-10-12 Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments

Family Applications Before (2)

Application Number Title Priority Date Filing Date
IL12787197A IL127871A0 (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines
IL127871A IL127871A (en) 1996-07-24 1998-12-30 PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL164513A IL164513A (en) 1996-07-24 2004-10-12 Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments

Country Status (15)

Country Link
JP (2) JP4704521B2 (en)
CN (3) CN1104432C (en)
AR (1) AR049583A2 (en)
BR (1) BR9710544A (en)
CA (1) CA2259583C (en)
CZ (1) CZ299451B6 (en)
EA (1) EA004403B1 (en)
EE (1) EE04316B1 (en)
HR (1) HRP970413A2 (en)
IL (4) IL127871A0 (en)
NO (1) NO315610B3 (en)
NZ (1) NZ333777A (en)
PL (1) PL195762B1 (en)
SI (1) SI9720045B (en)
SK (1) SK286461B6 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0208357A (en) * 2001-03-13 2004-06-29 Bristol Myers Squibb Pharma Co Compound, pharmaceutical composition, corticotropin-releasing factor (crf) receptor antagonization method, dysfunction treatment method, ligand screening method, crf receptor detection method, crf binding inhibition method, article industrialized and uses of compost
WO2004110454A1 (en) * 2003-06-13 2004-12-23 Ishihara Sangyo Kaisha, Ltd. COMPOSITION FOR TREATMENT FOR OR PREVENTION OF DISEASE NECESSITATING ADMINISTRATION OF ADENOSINE A2a RECEPTOR AGONIST
US7329662B2 (en) * 2003-10-03 2008-02-12 Hoffmann-La Roche Inc. Pyrazolo-pyridine
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
US8030304B2 (en) * 2006-09-20 2011-10-04 Eli Lilly And Company Thiazole pyrazolopyrimidines CRF1 receptor antagonists
CN103694242B (en) * 2013-12-10 2016-01-06 昆明翔昊科技有限公司 Pyrazolopyrimidines and pharmaceutical composition thereof and its application in pharmacy
CN112028891B (en) * 2019-07-30 2022-07-05 厦门宝太生物科技股份有限公司 Adenosine receptor antagonists
KR20230043222A (en) 2020-08-12 2023-03-30 스프루스 바이오사이언시스 인코포레이티드 Methods and compositions for treating polycystic ovary syndrome
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3995039A (en) * 1975-05-27 1976-11-30 Merck & Co., Inc. Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (en) * 1984-08-29 1986-03-24 Shionogi & Co Ltd Condensed heterocyclic derivative and antiulcerative
US4824834A (en) * 1986-10-31 1989-04-25 Otsuka Pharmaceutical Company, Limited Pyrazolotriazine compounds
JP2691317B2 (en) * 1989-08-25 1997-12-17 株式会社大塚製薬工場 4-Hydroxy-8- (3-lower alkoxy-4-phenylsulfinylphenyl) pyrazolo [1,5-a] -1,3,5-triazine optically active salts and process for producing the same
US5420128A (en) * 1990-10-09 1995-05-30 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor
EP0591528B1 (en) * 1991-04-22 1998-12-23 Otsuka Pharmaceutical Factory, Inc. PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVE AND ANTI-INFLAMMATORY CONTAINING THE SAME
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

Also Published As

Publication number Publication date
BR9710544A (en) 1999-08-17
CA2259583A1 (en) 1998-01-29
CN1250223C (en) 2006-04-12
SK9799A3 (en) 2005-04-01
EA199900158A1 (en) 1999-10-28
IL164513A (en) 2010-04-29
PL195762B1 (en) 2007-10-31
CN1104432C (en) 2003-04-02
AR049583A2 (en) 2006-08-16
EE04316B1 (en) 2004-06-15
CN1327793A (en) 2001-12-26
CA2259583C (en) 2009-11-17
JP4704521B2 (en) 2011-06-15
SI9720045A (en) 1999-10-31
CZ299451B6 (en) 2008-07-30
NO990264D0 (en) 1999-01-21
SK286461B6 (en) 2008-10-07
EE9900019A (en) 1999-08-16
NO990264L (en) 1999-03-10
JP2002513382A (en) 2002-05-08
NO315610B1 (en) 2003-09-29
CN1388126A (en) 2003-01-01
JP4194539B2 (en) 2008-12-10
EA004403B1 (en) 2004-04-29
JP2005097257A (en) 2005-04-14
CZ18499A3 (en) 1999-11-17
NO315610B3 (en) 2003-09-29
IL127871A (en) 2010-04-29
HRP970413A2 (en) 1998-10-31
NZ333777A (en) 2000-07-28
IL127871A0 (en) 1999-10-28
PL331523A1 (en) 1999-07-19
SI9720045B (en) 2008-02-29
IL164513A0 (en) 2005-12-18
CN1225637A (en) 1999-08-11

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Legal Events

Date Code Title Description
KB Patent renewed
EXP Patent expired