IL150163A - PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS - Google Patents
PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDSInfo
- Publication number
- IL150163A IL150163A IL150163A IL15016302A IL150163A IL 150163 A IL150163 A IL 150163A IL 150163 A IL150163 A IL 150163A IL 15016302 A IL15016302 A IL 15016302A IL 150163 A IL150163 A IL 150163A
- Authority
- IL
- Israel
- Prior art keywords
- pyrazolo
- novel
- compounds
- pharmaceutical compositions
- pyrimidine derivatives
- Prior art date
Links
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US68604796A | 1996-07-24 | 1996-07-24 | |
| US2329096P | 1996-07-24 | 1996-07-24 | |
| US08/899,242 US6124289A (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
| PCT/US1997/013072 WO1998003510A1 (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL150163A true IL150163A (en) | 2010-12-30 |
Family
ID=27362048
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL12787197A IL127871A0 (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
| IL127871A IL127871A (en) | 1996-07-24 | 1998-12-30 | PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES |
| IL150163A IL150163A (en) | 1996-07-24 | 2002-06-11 | PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS |
| IL164513A IL164513A (en) | 1996-07-24 | 2004-10-12 | Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL12787197A IL127871A0 (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
| IL127871A IL127871A (en) | 1996-07-24 | 1998-12-30 | PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL164513A IL164513A (en) | 1996-07-24 | 2004-10-12 | Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments |
Country Status (15)
| Country | Link |
|---|---|
| JP (2) | JP4704521B2 (en) |
| CN (3) | CN1104432C (en) |
| AR (1) | AR049583A2 (en) |
| BR (1) | BR9710544A (en) |
| CA (1) | CA2259583C (en) |
| CZ (1) | CZ299451B6 (en) |
| EA (1) | EA004403B1 (en) |
| EE (1) | EE04316B1 (en) |
| HR (1) | HRP970413A2 (en) |
| IL (4) | IL127871A0 (en) |
| NO (1) | NO315610B1 (en) |
| NZ (1) | NZ333777A (en) |
| PL (1) | PL195762B1 (en) |
| SI (1) | SI9720045B (en) |
| SK (1) | SK286461B6 (en) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR0208357A (en) * | 2001-03-13 | 2004-06-29 | Bristol Myers Squibb Pharma Co | Compound, pharmaceutical composition, corticotropin-releasing factor (crf) receptor antagonization method, dysfunction treatment method, ligand screening method, crf receptor detection method, crf binding inhibition method, article industrialized and uses of compost |
| WO2004110454A1 (en) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | COMPOSITION FOR TREATMENT FOR OR PREVENTION OF DISEASE NECESSITATING ADMINISTRATION OF ADENOSINE A2a RECEPTOR AGONIST |
| US7329662B2 (en) * | 2003-10-03 | 2008-02-12 | Hoffmann-La Roche Inc. | Pyrazolo-pyridine |
| GB0519957D0 (en) * | 2005-09-30 | 2005-11-09 | Sb Pharmco Inc | Chemical compound |
| UA96458C2 (en) * | 2006-09-20 | 2011-11-10 | Эли Лилли Энд Компани | Thiazole pyrazolopyrimidines as crf1 receptor antagonists |
| CN103694242B (en) * | 2013-12-10 | 2016-01-06 | 昆明翔昊科技有限公司 | Pyrazolopyrimidines and pharmaceutical composition thereof and its application in pharmacy |
| AU2018317398A1 (en) | 2017-08-14 | 2019-11-21 | Spruce Biosciences, Inc. | Corticotropin releasing factor receptor antagonists |
| CN112592346B (en) * | 2019-07-30 | 2022-04-26 | 厦门宝太生物科技股份有限公司 | Preparation method of A2A and/or A2B inhibitor intermediate |
| MX2023001688A (en) | 2020-08-12 | 2023-02-22 | Spruce Biosciences Inc | Methods and compositions for treating polycystic ovary syndrome. |
| US11708372B2 (en) | 2021-11-19 | 2023-07-25 | Spruce Biosciences, Inc. | Crystalline composition of tildacerfont and methods of use and preparation thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3995039A (en) * | 1975-05-27 | 1976-11-30 | Merck & Co., Inc. | Pyrazolo [1,5-a] [1,3,5] triazines |
| JPS6157587A (en) * | 1984-08-29 | 1986-03-24 | Shionogi & Co Ltd | Condensed heterocyclic derivative and antiulcerative |
| US4824834A (en) * | 1986-10-31 | 1989-04-25 | Otsuka Pharmaceutical Company, Limited | Pyrazolotriazine compounds |
| JP2691317B2 (en) * | 1989-08-25 | 1997-12-17 | 株式会社大塚製薬工場 | 4-Hydroxy-8- (3-lower alkoxy-4-phenylsulfinylphenyl) pyrazolo [1,5-a] -1,3,5-triazine optically active salts and process for producing the same |
| WO1992006096A1 (en) * | 1990-10-09 | 1992-04-16 | Otsuka Pharmaceutical Co., Ltd. | Pyrimidine derivative, production thereof, and androgen inhibitor |
| ES2126573T3 (en) * | 1991-04-22 | 1999-04-01 | Otsuka Pharma Co Ltd | DERIVATIVE OF PYRAZOLE (1,5-A) PIRIMIDINE AND ANTI-INFLAMMATORY AGENT CONTAINING THIS DERIVATIVE. |
| US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
-
1997
- 1997-07-23 CA CA002259583A patent/CA2259583C/en not_active Expired - Lifetime
- 1997-07-23 EA EA199900158A patent/EA004403B1/en not_active IP Right Cessation
- 1997-07-23 SK SK97-99A patent/SK286461B6/en not_active IP Right Cessation
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-23 CN CN97196525A patent/CN1104432C/en not_active Expired - Lifetime
- 1997-07-23 IL IL12787197A patent/IL127871A0/en unknown
- 1997-07-23 SI SI9720045A patent/SI9720045B/en active Search and Examination
- 1997-07-23 EE EEP199900019A patent/EE04316B1/en unknown
- 1997-07-23 BR BR9710544A patent/BR9710544A/en not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/en not_active Expired - Fee Related
- 1997-07-23 PL PL97331523A patent/PL195762B1/en unknown
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/en not_active IP Right Cessation
- 1997-07-24 HR HRP970413 patent/HRP970413A2/en not_active Application Discontinuation
-
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
-
1999
- 1999-01-21 NO NO19990264A patent/NO315610B1/en not_active IP Right Cessation
-
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/en not_active Expired - Lifetime
-
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/en active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
-
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/en not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
-
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| SI9720045B (en) | 2008-02-29 |
| EA199900158A1 (en) | 1999-10-28 |
| PL331523A1 (en) | 1999-07-19 |
| JP2005097257A (en) | 2005-04-14 |
| IL127871A0 (en) | 1999-10-28 |
| JP4194539B2 (en) | 2008-12-10 |
| IL127871A (en) | 2010-04-29 |
| SI9720045A (en) | 1999-10-31 |
| PL195762B1 (en) | 2007-10-31 |
| NO990264L (en) | 1999-03-10 |
| CN1104432C (en) | 2003-04-02 |
| EE9900019A (en) | 1999-08-16 |
| NZ333777A (en) | 2000-07-28 |
| AR049583A2 (en) | 2006-08-16 |
| IL164513A0 (en) | 2005-12-18 |
| CN1250223C (en) | 2006-04-12 |
| NO990264D0 (en) | 1999-01-21 |
| CN1388126A (en) | 2003-01-01 |
| CN1225637A (en) | 1999-08-11 |
| JP2002513382A (en) | 2002-05-08 |
| CZ299451B6 (en) | 2008-07-30 |
| CA2259583C (en) | 2009-11-17 |
| HRP970413A2 (en) | 1998-10-31 |
| SK9799A3 (en) | 2005-04-01 |
| JP4704521B2 (en) | 2011-06-15 |
| CZ18499A3 (en) | 1999-11-17 |
| CA2259583A1 (en) | 1998-01-29 |
| NO315610B3 (en) | 2003-09-29 |
| NO315610B1 (en) | 2003-09-29 |
| EE04316B1 (en) | 2004-06-15 |
| IL164513A (en) | 2010-04-29 |
| EA004403B1 (en) | 2004-04-29 |
| BR9710544A (en) | 1999-08-17 |
| SK286461B6 (en) | 2008-10-07 |
| CN1327793A (en) | 2001-12-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| KB | Patent renewed | ||
| EXP | Patent expired |