EE04316B1 - Azolotriazines and pyrimidines, their pharmaceutical compositions and their use in the manufacture of medicaments - Google Patents

Azolotriazines and pyrimidines, their pharmaceutical compositions and their use in the manufacture of medicaments

Info

Publication number
EE04316B1
EE04316B1 EEP199900019A EE9900019A EE04316B1 EE 04316 B1 EE04316 B1 EE 04316B1 EE P199900019 A EEP199900019 A EE P199900019A EE 9900019 A EE9900019 A EE 9900019A EE 04316 B1 EE04316 B1 EE 04316B1
Authority
EE
Estonia
Prior art keywords
azolotriazines
pyrimidines
medicaments
manufacture
pharmaceutical compositions
Prior art date
Application number
EEP199900019A
Other languages
Estonian (et)
Other versions
EE9900019A (en
Inventor
Georgios Arvanitis Argyrios
John Chorvat Robert
Original Assignee
Dupont Pharmaceuticals Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dupont Pharmaceuticals Company filed Critical Dupont Pharmaceuticals Company
Priority claimed from US08/899,242 external-priority patent/US6124289A/en
Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en
Publication of EE9900019A publication Critical patent/EE9900019A/en
Publication of EE04316B1 publication Critical patent/EE04316B1/en

Links

EEP199900019A 1996-07-24 1997-07-23 Azolotriazines and pyrimidines, their pharmaceutical compositions and their use in the manufacture of medicaments EE04316B1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US68604796A 1996-07-24 1996-07-24
US2329096P 1996-07-24 1996-07-24
US08/899,242 US6124289A (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines
PCT/US1997/013072 WO1998003510A1 (en) 1996-07-24 1997-07-23 Azolo triazines and pyrimidines

Publications (2)

Publication Number Publication Date
EE9900019A EE9900019A (en) 1999-08-16
EE04316B1 true EE04316B1 (en) 2004-06-15

Family

ID=27362048

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP199900019A EE04316B1 (en) 1996-07-24 1997-07-23 Azolotriazines and pyrimidines, their pharmaceutical compositions and their use in the manufacture of medicaments

Country Status (15)

Country Link
JP (2) JP4704521B2 (en)
CN (3) CN1104432C (en)
AR (1) AR049583A2 (en)
BR (1) BR9710544A (en)
CA (1) CA2259583C (en)
CZ (1) CZ299451B6 (en)
EA (1) EA004403B1 (en)
EE (1) EE04316B1 (en)
HR (1) HRP970413A2 (en)
IL (4) IL127871A0 (en)
NO (1) NO315610B3 (en)
NZ (1) NZ333777A (en)
PL (1) PL195762B1 (en)
SI (1) SI9720045B (en)
SK (1) SK286461B6 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA03008185A (en) * 2001-03-13 2004-01-29 Bristol Myers Squibb Pharma Co 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3, 5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands.
WO2004110454A1 (en) * 2003-06-13 2004-12-23 Ishihara Sangyo Kaisha, Ltd. COMPOSITION FOR TREATMENT FOR OR PREVENTION OF DISEASE NECESSITATING ADMINISTRATION OF ADENOSINE A2a RECEPTOR AGONIST
US7329662B2 (en) * 2003-10-03 2008-02-12 Hoffmann-La Roche Inc. Pyrazolo-pyridine
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
KR101088239B1 (en) * 2006-09-20 2011-11-30 일라이 릴리 앤드 캄파니 Thiazole pyrazolopyrimidines as crf1 receptor antagonists
CN103694242B (en) * 2013-12-10 2016-01-06 昆明翔昊科技有限公司 Pyrazolopyrimidines and pharmaceutical composition thereof and its application in pharmacy
CN112028891B (en) * 2019-07-30 2022-07-05 厦门宝太生物科技股份有限公司 Adenosine receptor antagonists
KR20230043222A (en) 2020-08-12 2023-03-30 스프루스 바이오사이언시스 인코포레이티드 Methods and compositions for treating polycystic ovary syndrome
US11708372B2 (en) 2021-11-19 2023-07-25 Spruce Biosciences, Inc. Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3995039A (en) * 1975-05-27 1976-11-30 Merck & Co., Inc. Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (en) * 1984-08-29 1986-03-24 Shionogi & Co Ltd Condensed heterocyclic derivative and antiulcerative
US4824834A (en) * 1986-10-31 1989-04-25 Otsuka Pharmaceutical Company, Limited Pyrazolotriazine compounds
JP2691317B2 (en) * 1989-08-25 1997-12-17 株式会社大塚製薬工場 4-Hydroxy-8- (3-lower alkoxy-4-phenylsulfinylphenyl) pyrazolo [1,5-a] -1,3,5-triazine optically active salts and process for producing the same
US5420128A (en) * 1990-10-09 1995-05-30 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor
DE69130683T2 (en) * 1991-04-22 1999-05-06 Otsuka Pharma Co Ltd PYRAZOLO [1,5-a] PYRIMIDINE DERIVATIVES AND ANTI-INFLAMMATORY CONTAINERS THEREOF
US5356897A (en) * 1991-09-09 1994-10-18 Fujisawa Pharmaceutical Co., Ltd. 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

Also Published As

Publication number Publication date
EE9900019A (en) 1999-08-16
CN1225637A (en) 1999-08-11
CA2259583A1 (en) 1998-01-29
NZ333777A (en) 2000-07-28
CN1250223C (en) 2006-04-12
SI9720045A (en) 1999-10-31
EA199900158A1 (en) 1999-10-28
IL164513A (en) 2010-04-29
IL150163A (en) 2010-12-30
NO990264D0 (en) 1999-01-21
EA004403B1 (en) 2004-04-29
IL164513A0 (en) 2005-12-18
NO315610B1 (en) 2003-09-29
NO315610B3 (en) 2003-09-29
JP2002513382A (en) 2002-05-08
IL127871A0 (en) 1999-10-28
CN1327793A (en) 2001-12-26
AR049583A2 (en) 2006-08-16
NO990264L (en) 1999-03-10
SK286461B6 (en) 2008-10-07
CN1388126A (en) 2003-01-01
PL195762B1 (en) 2007-10-31
JP4704521B2 (en) 2011-06-15
CZ299451B6 (en) 2008-07-30
IL127871A (en) 2010-04-29
CA2259583C (en) 2009-11-17
CN1104432C (en) 2003-04-02
JP2005097257A (en) 2005-04-14
PL331523A1 (en) 1999-07-19
SK9799A3 (en) 2005-04-01
CZ18499A3 (en) 1999-11-17
BR9710544A (en) 1999-08-17
SI9720045B (en) 2008-02-29
JP4194539B2 (en) 2008-12-10
HRP970413A2 (en) 1998-10-31

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Legal Events

Date Code Title Description
KB4A Valid patent at the end of a year

Effective date: 20041231

LD4A Amendment in the specification
KB4A Valid patent at the end of a year

Effective date: 20051231

KB4A Valid patent at the end of a year

Effective date: 20061231

KB4A Valid patent at the end of a year

Effective date: 20071231

KB4A Valid patent at the end of a year

Effective date: 20081231

KB4A Valid patent at the end of a year

Effective date: 20101231