EE04316B1 - Azolotriazines and pyrimidines, their pharmaceutical compositions and their use in the manufacture of medicaments - Google Patents
Azolotriazines and pyrimidines, their pharmaceutical compositions and their use in the manufacture of medicamentsInfo
- Publication number
- EE04316B1 EE04316B1 EEP199900019A EE9900019A EE04316B1 EE 04316 B1 EE04316 B1 EE 04316B1 EE P199900019 A EEP199900019 A EE P199900019A EE 9900019 A EE9900019 A EE 9900019A EE 04316 B1 EE04316 B1 EE 04316B1
- Authority
- EE
- Estonia
- Prior art keywords
- azolotriazines
- pyrimidines
- medicaments
- manufacture
- pharmaceutical compositions
- Prior art date
Links
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US68604796A | 1996-07-24 | 1996-07-24 | |
US2329096P | 1996-07-24 | 1996-07-24 | |
US08/899,242 US6124289A (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
PCT/US1997/013072 WO1998003510A1 (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
Publications (2)
Publication Number | Publication Date |
---|---|
EE9900019A EE9900019A (en) | 1999-08-16 |
EE04316B1 true EE04316B1 (en) | 2004-06-15 |
Family
ID=27362048
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EEP199900019A EE04316B1 (en) | 1996-07-24 | 1997-07-23 | Azolotriazines and pyrimidines, their pharmaceutical compositions and their use in the manufacture of medicaments |
Country Status (15)
Country | Link |
---|---|
JP (2) | JP4704521B2 (en) |
CN (3) | CN1104432C (en) |
AR (1) | AR049583A2 (en) |
BR (1) | BR9710544A (en) |
CA (1) | CA2259583C (en) |
CZ (1) | CZ299451B6 (en) |
EA (1) | EA004403B1 (en) |
EE (1) | EE04316B1 (en) |
HR (1) | HRP970413A2 (en) |
IL (4) | IL127871A0 (en) |
NO (1) | NO315610B3 (en) |
NZ (1) | NZ333777A (en) |
PL (1) | PL195762B1 (en) |
SI (1) | SI9720045B (en) |
SK (1) | SK286461B6 (en) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MXPA03008185A (en) * | 2001-03-13 | 2004-01-29 | Bristol Myers Squibb Pharma Co | 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3, 5-triazine, its enantiomers and pharmaceutically acceptable salts as corticotropin releasing factor receptor ligands. |
WO2004110454A1 (en) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | COMPOSITION FOR TREATMENT FOR OR PREVENTION OF DISEASE NECESSITATING ADMINISTRATION OF ADENOSINE A2a RECEPTOR AGONIST |
US7329662B2 (en) * | 2003-10-03 | 2008-02-12 | Hoffmann-La Roche Inc. | Pyrazolo-pyridine |
GB0519957D0 (en) * | 2005-09-30 | 2005-11-09 | Sb Pharmco Inc | Chemical compound |
KR101088239B1 (en) * | 2006-09-20 | 2011-11-30 | 일라이 릴리 앤드 캄파니 | Thiazole pyrazolopyrimidines as crf1 receptor antagonists |
CN103694242B (en) * | 2013-12-10 | 2016-01-06 | 昆明翔昊科技有限公司 | Pyrazolopyrimidines and pharmaceutical composition thereof and its application in pharmacy |
CN112028891B (en) * | 2019-07-30 | 2022-07-05 | 厦门宝太生物科技股份有限公司 | Adenosine receptor antagonists |
KR20230043222A (en) | 2020-08-12 | 2023-03-30 | 스프루스 바이오사이언시스 인코포레이티드 | Methods and compositions for treating polycystic ovary syndrome |
US11708372B2 (en) | 2021-11-19 | 2023-07-25 | Spruce Biosciences, Inc. | Crystalline composition of tildacerfont and methods of use and preparation thereof |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3995039A (en) * | 1975-05-27 | 1976-11-30 | Merck & Co., Inc. | Pyrazolo [1,5-a] [1,3,5] triazines |
JPS6157587A (en) * | 1984-08-29 | 1986-03-24 | Shionogi & Co Ltd | Condensed heterocyclic derivative and antiulcerative |
US4824834A (en) * | 1986-10-31 | 1989-04-25 | Otsuka Pharmaceutical Company, Limited | Pyrazolotriazine compounds |
JP2691317B2 (en) * | 1989-08-25 | 1997-12-17 | 株式会社大塚製薬工場 | 4-Hydroxy-8- (3-lower alkoxy-4-phenylsulfinylphenyl) pyrazolo [1,5-a] -1,3,5-triazine optically active salts and process for producing the same |
US5420128A (en) * | 1990-10-09 | 1995-05-30 | Otsuka Pharmaceutical Co., Ltd. | Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor |
DE69130683T2 (en) * | 1991-04-22 | 1999-05-06 | Otsuka Pharma Co Ltd | PYRAZOLO [1,5-a] PYRIMIDINE DERIVATIVES AND ANTI-INFLAMMATORY CONTAINERS THEREOF |
US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
-
1997
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-23 CN CN97196525A patent/CN1104432C/en not_active Expired - Lifetime
- 1997-07-23 SK SK97-99A patent/SK286461B6/en not_active IP Right Cessation
- 1997-07-23 BR BR9710544A patent/BR9710544A/en not_active IP Right Cessation
- 1997-07-23 PL PL97331523A patent/PL195762B1/en unknown
- 1997-07-23 IL IL12787197A patent/IL127871A0/en unknown
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/en not_active IP Right Cessation
- 1997-07-23 EE EEP199900019A patent/EE04316B1/en unknown
- 1997-07-23 CA CA002259583A patent/CA2259583C/en not_active Expired - Lifetime
- 1997-07-23 EA EA199900158A patent/EA004403B1/en not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/en not_active Expired - Fee Related
- 1997-07-23 SI SI9720045A patent/SI9720045B/en active Search and Examination
- 1997-07-24 HR HRP970413 patent/HRP970413A2/en not_active Application Discontinuation
-
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
-
1999
- 1999-01-21 NO NO19990264A patent/NO315610B3/en not_active IP Right Cessation
-
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/en not_active Expired - Lifetime
-
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/en active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
-
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/en not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
-
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EE9900019A (en) | 1999-08-16 |
CN1225637A (en) | 1999-08-11 |
CA2259583A1 (en) | 1998-01-29 |
NZ333777A (en) | 2000-07-28 |
CN1250223C (en) | 2006-04-12 |
SI9720045A (en) | 1999-10-31 |
EA199900158A1 (en) | 1999-10-28 |
IL164513A (en) | 2010-04-29 |
IL150163A (en) | 2010-12-30 |
NO990264D0 (en) | 1999-01-21 |
EA004403B1 (en) | 2004-04-29 |
IL164513A0 (en) | 2005-12-18 |
NO315610B1 (en) | 2003-09-29 |
NO315610B3 (en) | 2003-09-29 |
JP2002513382A (en) | 2002-05-08 |
IL127871A0 (en) | 1999-10-28 |
CN1327793A (en) | 2001-12-26 |
AR049583A2 (en) | 2006-08-16 |
NO990264L (en) | 1999-03-10 |
SK286461B6 (en) | 2008-10-07 |
CN1388126A (en) | 2003-01-01 |
PL195762B1 (en) | 2007-10-31 |
JP4704521B2 (en) | 2011-06-15 |
CZ299451B6 (en) | 2008-07-30 |
IL127871A (en) | 2010-04-29 |
CA2259583C (en) | 2009-11-17 |
CN1104432C (en) | 2003-04-02 |
JP2005097257A (en) | 2005-04-14 |
PL331523A1 (en) | 1999-07-19 |
SK9799A3 (en) | 2005-04-01 |
CZ18499A3 (en) | 1999-11-17 |
BR9710544A (en) | 1999-08-17 |
SI9720045B (en) | 2008-02-29 |
JP4194539B2 (en) | 2008-12-10 |
HRP970413A2 (en) | 1998-10-31 |
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Legal Events
Date | Code | Title | Description |
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KB4A | Valid patent at the end of a year |
Effective date: 20041231 |
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LD4A | Amendment in the specification | ||
KB4A | Valid patent at the end of a year |
Effective date: 20051231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20061231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20071231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20081231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20101231 |