JP4704521B2 - アゾロトリアジン類およびアゾロピリミジン類 - Google Patents
アゾロトリアジン類およびアゾロピリミジン類 Download PDFInfo
- Publication number
- JP4704521B2 JP4704521B2 JP50723398A JP50723398A JP4704521B2 JP 4704521 B2 JP4704521 B2 JP 4704521B2 JP 50723398 A JP50723398 A JP 50723398A JP 50723398 A JP50723398 A JP 50723398A JP 4704521 B2 JP4704521 B2 JP 4704521B2
- Authority
- JP
- Japan
- Prior art keywords
- formula
- alkyl
- compound
- ome
- cor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- CVOYAMSQZCXQDY-UHFFFAOYSA-N Oc([n]1nc2)ncnc1c2-c(cc1)ccc1S(c1ccccc1)O Chemical compound Oc([n]1nc2)ncnc1c2-c(cc1)ccc1S(c1ccccc1)O CVOYAMSQZCXQDY-UHFFFAOYSA-N 0.000 description 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Detergent Compositions (AREA)
- Coloring (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2329096P | 1996-07-24 | 1996-07-24 | |
| US68604796A | 1996-07-24 | 1996-07-24 | |
| US08/686,047 | 1996-07-24 | ||
| US60/023,290 | 1996-07-24 | ||
| PCT/US1997/013072 WO1998003510A1 (en) | 1996-07-24 | 1997-07-23 | AZOLO TRIAZINES AND PYRIMIDINES |
| US08/899,242 | 1997-07-23 | ||
| US08/899,242 US6124289A (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004216483A Division JP4194539B2 (ja) | 1996-07-24 | 2004-07-23 | アゾロトリアジン類およびアゾロピリミジン類 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2002513382A JP2002513382A (ja) | 2002-05-08 |
| JP2002513382A5 JP2002513382A5 (zh) | 2005-12-02 |
| JP4704521B2 true JP4704521B2 (ja) | 2011-06-15 |
Family
ID=27362048
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP50723398A Expired - Fee Related JP4704521B2 (ja) | 1996-07-24 | 1997-07-23 | アゾロトリアジン類およびアゾロピリミジン類 |
| JP2004216483A Expired - Fee Related JP4194539B2 (ja) | 1996-07-24 | 2004-07-23 | アゾロトリアジン類およびアゾロピリミジン類 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004216483A Expired - Fee Related JP4194539B2 (ja) | 1996-07-24 | 2004-07-23 | アゾロトリアジン類およびアゾロピリミジン類 |
Country Status (15)
| Country | Link |
|---|---|
| JP (2) | JP4704521B2 (zh) |
| CN (3) | CN1104432C (zh) |
| AR (1) | AR049583A2 (zh) |
| BR (1) | BR9710544A (zh) |
| CA (1) | CA2259583C (zh) |
| CZ (1) | CZ299451B6 (zh) |
| EA (1) | EA004403B1 (zh) |
| EE (1) | EE04316B1 (zh) |
| HR (1) | HRP970413A2 (zh) |
| IL (4) | IL127871A0 (zh) |
| NO (1) | NO315610B1 (zh) |
| NZ (1) | NZ333777A (zh) |
| PL (1) | PL195762B1 (zh) |
| SI (1) | SI9720045B (zh) |
| SK (1) | SK286461B6 (zh) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA03008185A (es) * | 2001-03-13 | 2004-01-29 | Bristol Myers Squibb Pharma Co | 4-(2-butilamino)-2, 7-dimetil-8 -(2-metil-6-metoxipirid -3-il) pirazol-[1, 5-a]-1, 3, 5-triazina, sus enantiomeros y sales farmaceuticamente aceptables como ligandos del receptor del factor de liberacion de corticotropina. |
| WO2004110454A1 (ja) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物 |
| US7329662B2 (en) * | 2003-10-03 | 2008-02-12 | Hoffmann-La Roche Inc. | Pyrazolo-pyridine |
| GB0519957D0 (en) * | 2005-09-30 | 2005-11-09 | Sb Pharmco Inc | Chemical compound |
| MX2009003125A (es) * | 2006-09-20 | 2009-05-28 | Lilly Co Eli | Tiazol pirazolopirimidinas como antagonistas de receptor de crf1. |
| CN103694242B (zh) * | 2013-12-10 | 2016-01-06 | 昆明翔昊科技有限公司 | 吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用 |
| CN112592346B (zh) * | 2019-07-30 | 2022-04-26 | 厦门宝太生物科技股份有限公司 | 一种a2a和/或a2b抑制剂中间体的制备方法 |
| CN116322544A (zh) | 2020-08-12 | 2023-06-23 | 云杉生物科学公司 | 用于治疗多囊卵巢综合征的方法和组合物 |
| US11708372B2 (en) | 2021-11-19 | 2023-07-25 | Spruce Biosciences, Inc. | Crystalline composition of tildacerfont and methods of use and preparation thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3995039A (en) * | 1975-05-27 | 1976-11-30 | Merck & Co., Inc. | Pyrazolo [1,5-a] [1,3,5] triazines |
| JPS6157587A (ja) * | 1984-08-29 | 1986-03-24 | Shionogi & Co Ltd | 縮合複素環誘導体および抗潰瘍剤 |
| US4824834A (en) * | 1986-10-31 | 1989-04-25 | Otsuka Pharmaceutical Company, Limited | Pyrazolotriazine compounds |
| JP2691317B2 (ja) * | 1989-08-25 | 1997-12-17 | 株式会社大塚製薬工場 | ４―ヒドロキシ―８―（３―低級アルコキシ―４―フェニルスルフィニルフェニル）ピラゾロ〔１，５―ａ〕―１，３，５―トリアジン光学活性体の塩類及びその製造方法 |
| AU639615B2 (en) * | 1990-10-09 | 1993-07-29 | Otsuka Pharmaceutical Co., Ltd. | Pyrimidine derivative, production thereof, and androgen inhibitor |
| ATE174917T1 (de) * | 1991-04-22 | 1999-01-15 | Otsuka Pharma Co Ltd | Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel |
| US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
-
1997
- 1997-07-23 SI SI9720045A patent/SI9720045B/sl active Search and Examination
- 1997-07-23 CA CA002259583A patent/CA2259583C/en not_active Expired - Lifetime
- 1997-07-23 PL PL97331523A patent/PL195762B1/pl unknown
- 1997-07-23 CN CN97196525A patent/CN1104432C/zh not_active Expired - Lifetime
- 1997-07-23 EA EA199900158A patent/EA004403B1/ru not_active IP Right Cessation
- 1997-07-23 BR BR9710544A patent/BR9710544A/pt not_active IP Right Cessation
- 1997-07-23 EE EEP199900019A patent/EE04316B1/xx unknown
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/cs not_active IP Right Cessation
- 1997-07-23 SK SK97-99A patent/SK286461B6/sk not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/ja not_active Expired - Fee Related
- 1997-07-23 IL IL12787197A patent/IL127871A0/xx unknown
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-24 HR HRP970413 patent/HRP970413A2/hr not_active Application Discontinuation
-
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
-
1999
- 1999-01-21 NO NO19990264A patent/NO315610B1/no not_active IP Right Cessation
-
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/zh not_active Expired - Lifetime
-
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/zh active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
-
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/ja not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
-
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JP4194539B2 (ja) | 2008-12-10 |
| AR049583A2 (es) | 2006-08-16 |
| SK286461B6 (sk) | 2008-10-07 |
| IL150163A (en) | 2010-12-30 |
| CN1104432C (zh) | 2003-04-02 |
| PL195762B1 (pl) | 2007-10-31 |
| EE9900019A (et) | 1999-08-16 |
| NZ333777A (en) | 2000-07-28 |
| NO990264D0 (no) | 1999-01-21 |
| EA004403B1 (ru) | 2004-04-29 |
| CZ18499A3 (cs) | 1999-11-17 |
| SI9720045B (sl) | 2008-02-29 |
| NO990264L (no) | 1999-03-10 |
| EE04316B1 (et) | 2004-06-15 |
| IL164513A (en) | 2010-04-29 |
| BR9710544A (pt) | 1999-08-17 |
| IL127871A (en) | 2010-04-29 |
| SI9720045A (sl) | 1999-10-31 |
| NO315610B3 (no) | 2003-09-29 |
| CN1250223C (zh) | 2006-04-12 |
| CN1225637A (zh) | 1999-08-11 |
| CA2259583A1 (en) | 1998-01-29 |
| HRP970413A2 (en) | 1998-10-31 |
| IL127871A0 (en) | 1999-10-28 |
| JP2005097257A (ja) | 2005-04-14 |
| CZ299451B6 (cs) | 2008-07-30 |
| NO315610B1 (no) | 2003-09-29 |
| EA199900158A1 (ru) | 1999-10-28 |
| JP2002513382A (ja) | 2002-05-08 |
| CA2259583C (en) | 2009-11-17 |
| CN1388126A (zh) | 2003-01-01 |
| SK9799A3 (sk) | 2005-04-01 |
| IL164513A0 (en) | 2005-12-18 |
| CN1327793A (zh) | 2001-12-26 |
| PL331523A1 (en) | 1999-07-19 |
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