SI1283839T1 - - Google Patents

Info

Publication number
SI1283839T1
SI1283839T1 SI200130336T SI200130336T SI1283839T1 SI 1283839 T1 SI1283839 T1 SI 1283839T1 SI 200130336 T SI200130336 T SI 200130336T SI 200130336 T SI200130336 T SI 200130336T SI 1283839 T1 SI1283839 T1 SI 1283839T1
Authority
SI
Slovenia
Application number
SI200130336T
Inventor
Bernard R Neustadt
Neil A Lindo
William J Greenlee
Deen Tulshian
Lisa S Silverman
Yan Xia
Craig D Boyle
Samuel Chackalamannil
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of SI1283839T1 publication Critical patent/SI1283839T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SI200130336T 2000-05-26 2001-05-24 SI1283839T1 (OSRAM)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20714300P 2000-05-26 2000-05-26
EP01945991A EP1283839B1 (en) 2000-05-26 2001-05-24 Adenosine a2a receptor antagonists
PCT/US2001/016954 WO2001092264A1 (en) 2000-05-26 2001-05-24 Adenosine a2a receptor antagonists

Publications (1)

Publication Number Publication Date
SI1283839T1 true SI1283839T1 (OSRAM) 2005-08-31

Family

ID=22769372

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200130336T SI1283839T1 (OSRAM) 2000-05-26 2001-05-24

Country Status (31)

Country Link
US (4) US6630475B2 (OSRAM)
EP (1) EP1283839B1 (OSRAM)
JP (3) JP4574112B2 (OSRAM)
KR (1) KR100520907B1 (OSRAM)
CN (2) CN100384847C (OSRAM)
AR (1) AR028621A1 (OSRAM)
AT (1) ATE293627T1 (OSRAM)
AU (2) AU2001268089C1 (OSRAM)
BR (1) BRPI0111015B8 (OSRAM)
CA (1) CA2410237C (OSRAM)
CZ (1) CZ303790B6 (OSRAM)
DE (1) DE60110219T2 (OSRAM)
DK (1) DK1283839T3 (OSRAM)
EC (1) ECSP024364A (OSRAM)
ES (1) ES2237576T3 (OSRAM)
HK (1) HK1049007B (OSRAM)
HU (1) HU230420B1 (OSRAM)
IL (3) IL152726A0 (OSRAM)
MX (1) MXPA02011625A (OSRAM)
MY (1) MY132006A (OSRAM)
NO (1) NO325008B1 (OSRAM)
NZ (1) NZ522326A (OSRAM)
PE (1) PE20020062A1 (OSRAM)
PL (1) PL218764B1 (OSRAM)
PT (1) PT1283839E (OSRAM)
RU (1) RU2315053C2 (OSRAM)
SI (1) SI1283839T1 (OSRAM)
SK (1) SK287748B6 (OSRAM)
TW (1) TWI288137B (OSRAM)
WO (1) WO2001092264A1 (OSRAM)
ZA (1) ZA200208898B (OSRAM)

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JP2022540583A (ja) * 2019-07-17 2022-09-16 テオン セラピューティクス，インク． アデノシンａ２ａ受容体アンタゴニスト及びその使用
CN112608330B (zh) 2019-07-30 2021-09-28 杭州阿诺生物医药科技有限公司 A2a和/或a2b受体抑制剂
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CN111072675A (zh) * 2019-12-12 2020-04-28 广东东阳光药业有限公司 含氮稠合三环衍生物及其用途
CN113773327B (zh) * 2021-09-13 2022-07-15 八叶草健康产业研究院(厦门)有限公司 一种吡唑并嘧啶并三唑环类化合物的制备方法
CN118812544A (zh) * 2024-06-19 2024-10-22 厦门大学 一种腺苷a2ar靶向小分子化合物、核素标记探针及其制备方法、应用和药物组合物
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Publication number Publication date
ATE293627T1 (de) 2005-05-15
US6897216B2 (en) 2005-05-24
CZ303790B6 (cs) 2013-05-09
MY132006A (en) 2007-09-28
NO20025651L (no) 2003-01-23
SK16712002A3 (sk) 2003-08-05
BR0111015A (pt) 2005-01-11
DE60110219D1 (de) 2005-05-25
HUP0600239A2 (en) 2006-07-28
US20040023997A1 (en) 2004-02-05
CN100384847C (zh) 2008-04-30
IL152726A (en) 2012-07-31
HK1049007B (en) 2005-09-16
TWI288137B (en) 2007-10-11
DK1283839T3 (da) 2005-07-25
CN1247588C (zh) 2006-03-29
CA2410237C (en) 2008-01-08
HUP0600239A3 (en) 2008-06-30
US7067655B2 (en) 2006-06-27
JP2003535094A (ja) 2003-11-25
NZ522326A (en) 2006-03-31
DE60110219T2 (de) 2006-03-09
ECSP024364A (es) 2003-03-31
RU2315053C2 (ru) 2008-01-20
JP4574112B2 (ja) 2010-11-04
PL360472A1 (en) 2004-09-06
BRPI0111015B8 (pt) 2021-05-25
ES2237576T3 (es) 2005-08-01
CZ20023886A3 (cs) 2003-02-12
HU230420B1 (hu) 2016-05-30
WO2001092264A1 (en) 2001-12-06
NO325008B1 (no) 2008-01-14
IL152726A0 (en) 2003-06-24
EP1283839B1 (en) 2005-04-20
IL220174A0 (en) 2012-07-31
NO20025651D0 (no) 2002-11-25
AU2001268089C1 (en) 2006-04-13
AU2001268089B2 (en) 2005-04-28
AR028621A1 (es) 2003-05-14
MXPA02011625A (es) 2003-03-27
EP1283839A1 (en) 2003-02-19
IL220174A (en) 2015-07-30
JP4938348B2 (ja) 2012-05-23
SK287748B6 (sk) 2011-08-04
JP2007145875A (ja) 2007-06-14
BRPI0111015B1 (pt) 2017-11-07
PE20020062A1 (es) 2002-02-02
USRE44205E1 (en) 2013-05-07
AU6808901A (en) 2001-12-11
CN1451007A (zh) 2003-10-22
CA2410237A1 (en) 2001-12-06
KR20030003746A (ko) 2003-01-10
US20020099061A1 (en) 2002-07-25
PT1283839E (pt) 2005-08-31
ZA200208898B (en) 2004-03-01
CN1800186A (zh) 2006-07-12
US20050026932A1 (en) 2005-02-03
PL218764B1 (pl) 2015-01-30
US6630475B2 (en) 2003-10-07
HK1049007A1 (en) 2003-04-25
KR100520907B1 (ko) 2005-10-11
JP2006219497A (ja) 2006-08-24

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