SG178721A1 - Amino acid prodrugs - Google Patents
Amino acid prodrugs Download PDFInfo
- Publication number
- SG178721A1 SG178721A1 SG2012005310A SG2012005310A SG178721A1 SG 178721 A1 SG178721 A1 SG 178721A1 SG 2012005310 A SG2012005310 A SG 2012005310A SG 2012005310 A SG2012005310 A SG 2012005310A SG 178721 A1 SG178721 A1 SG 178721A1
- Authority
- SG
- Singapore
- Prior art keywords
- amino acid
- drug
- group
- acid
- gly
- Prior art date
Links
- 229940002612 prodrug Drugs 0.000 title claims abstract description 94
- 239000000651 prodrug Substances 0.000 title claims abstract description 93
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- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
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NZ524087A (en) * | 2000-08-18 | 2004-08-27 | Univ Illinois | Prodrugs of betulinic acid derivatives for the treatment of cancer and HIV |
US20020160988A1 (en) * | 2001-02-20 | 2002-10-31 | Israel Institute For Biological Research | Compounds co-inducing cholinergic up-regulation and inflammation down-regulation and uses thereof |
US7045543B2 (en) * | 2001-11-05 | 2006-05-16 | Enzrel Inc. | Covalent conjugates of biologically-active compounds with amino acids and amino acid derivatives for targeting to physiologically-protected sites |
WO2004087699A2 (en) * | 2003-03-25 | 2004-10-14 | Vertex Pharmaceuticals Incorporated | Thiazoles useful as inhibitors of protein kinases |
EP1660017A4 (en) * | 2003-07-29 | 2011-03-09 | Signature R & D Holdings Llc | Amino acid PRODRUGS |
-
2004
- 2004-07-29 EP EP04816791A patent/EP1660017A4/en not_active Withdrawn
- 2004-07-29 AU AU2004289174A patent/AU2004289174B2/en not_active Ceased
- 2004-07-29 KR KR1020137015399A patent/KR20130081319A/ko not_active Application Discontinuation
- 2004-07-29 JP JP2006522125A patent/JP2007510621A/ja active Pending
- 2004-07-29 SG SG2012005310A patent/SG178721A1/en unknown
- 2004-07-29 WO PCT/US2004/024901 patent/WO2005046575A2/en active Application Filing
- 2004-07-29 NZ NZ545570A patent/NZ545570A/xx not_active IP Right Cessation
- 2004-07-29 KR KR1020067002214A patent/KR20060073584A/ko active Search and Examination
- 2004-07-29 NZ NZ601772A patent/NZ601772A/xx not_active IP Right Cessation
- 2004-07-29 CA CA2534342A patent/CA2534342C/en not_active Expired - Fee Related
- 2004-07-29 SG SG200805624-4A patent/SG145693A1/en unknown
- 2004-07-29 NZ NZ601780A patent/NZ601780A/xx not_active IP Right Cessation
- 2004-07-29 CN CNA2004800282229A patent/CN101123878A/zh active Pending
- 2004-07-29 KR KR1020127022817A patent/KR20120116991A/ko not_active Application Discontinuation
-
2005
- 2005-01-23 ZA ZA200600660A patent/ZA200600660B/xx unknown
-
2006
- 2006-01-26 IL IL173382A patent/IL173382A0/en unknown
-
2012
- 2012-10-01 JP JP2012219487A patent/JP2013035863A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
ZA200600660B (en) | 2007-04-25 |
EP1660017A2 (en) | 2006-05-31 |
NZ601780A (en) | 2012-10-26 |
WO2005046575A2 (en) | 2005-05-26 |
WO2005046575A3 (en) | 2007-10-04 |
NZ545570A (en) | 2012-07-27 |
KR20130081319A (ko) | 2013-07-16 |
KR20060073584A (ko) | 2006-06-28 |
AU2004289174A2 (en) | 2005-05-26 |
JP2013035863A (ja) | 2013-02-21 |
CN101123878A (zh) | 2008-02-13 |
AU2004289174A1 (en) | 2005-05-26 |
JP2007510621A (ja) | 2007-04-26 |
IL173382A0 (en) | 2006-06-11 |
CA2534342C (en) | 2016-05-10 |
CA2534342A1 (en) | 2005-05-26 |
NZ601772A (en) | 2012-10-26 |
EP1660017A4 (en) | 2011-03-09 |
KR20120116991A (ko) | 2012-10-23 |
SG145693A1 (en) | 2008-09-29 |
AU2004289174B2 (en) | 2011-05-19 |
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