SG1189G - Derivatives of cis,endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid,process for their preparation,medicines containing them and their use - Google Patents

Derivatives of cis,endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid,process for their preparation,medicines containing them and their use

Info

Publication number
SG1189G
SG1189G SG11/89A SG1189A SG1189G SG 1189 G SG1189 G SG 1189G SG 11/89 A SG11/89 A SG 11/89A SG 1189 A SG1189 A SG 1189A SG 1189 G SG1189 G SG 1189G
Authority
SG
Singapore
Prior art keywords
azabicyclo
endo
octane
cis
derivatives
Prior art date
Application number
SG11/89A
Other languages
English (en)
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25797115&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG1189(G) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of SG1189G publication Critical patent/SG1189G/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SG11/89A 1981-11-05 1989-01-07 Derivatives of cis,endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid,process for their preparation,medicines containing them and their use SG1189G (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3143946 1981-11-05
DE19823226768 DE3226768A1 (de) 1981-11-05 1982-07-17 Derivate der cis, endo-2-azabicyclo-(3.3.0)-octan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung

Publications (1)

Publication Number Publication Date
SG1189G true SG1189G (en) 1993-02-19

Family

ID=25797115

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11/89A SG1189G (en) 1981-11-05 1989-01-07 Derivatives of cis,endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid,process for their preparation,medicines containing them and their use

Country Status (31)

Country Link
US (4) US4727160A (fr)
EP (2) EP0079022B1 (fr)
JP (3) JPH02104526A (fr)
KR (1) KR890000007B1 (fr)
AR (1) AR240675A1 (fr)
AU (3) AU565200B2 (fr)
BG (1) BG60532B2 (fr)
CA (1) CA1187087A (fr)
CS (1) CS247159B2 (fr)
CZ (1) CZ416291A3 (fr)
DD (2) DD203047A5 (fr)
DE (3) DE3226768A1 (fr)
DK (2) DK166624C (fr)
DZ (1) DZ473A1 (fr)
ES (3) ES517066A0 (fr)
FI (1) FI81087C (fr)
GR (1) GR77381B (fr)
HK (1) HK74889A (fr)
HU (2) HU186339B (fr)
IE (1) IE56476B1 (fr)
IL (1) IL67172A (fr)
JO (1) JO1224B1 (fr)
LU (1) LU88260I2 (fr)
MA (1) MA19639A1 (fr)
NL (1) NL930039I2 (fr)
NO (2) NO156940C (fr)
NZ (1) NZ202378A (fr)
PH (2) PH22417A (fr)
PT (1) PT75792A (fr)
SG (1) SG1189G (fr)
SU (1) SU1277895A3 (fr)

Families Citing this family (127)

* Cited by examiner, † Cited by third party
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DE3226768A1 (de) 1983-05-26
JPH0355449B2 (fr) 1991-08-23
LU88260I2 (fr) 1994-02-03
ES518133A0 (es) 1983-09-01
PT75792A (de) 1982-12-01
EP0079022B1 (fr) 1986-03-12
FI81087C (fi) 1990-09-10
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CZ416291A3 (en) 1993-09-15
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US4727160A (en) 1988-02-23
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