SG11201505680RA - Solid forms of a selective cdk4/6 inhibitor - Google Patents

Solid forms of a selective cdk4/6 inhibitor

Info

Publication number
SG11201505680RA
SG11201505680RA SG11201505680RA SG11201505680RA SG11201505680RA SG 11201505680R A SG11201505680R A SG 11201505680RA SG 11201505680R A SG11201505680R A SG 11201505680RA SG 11201505680R A SG11201505680R A SG 11201505680RA SG 11201505680R A SG11201505680R A SG 11201505680RA
Authority
SG
Singapore
Prior art keywords
inhibitor
solid forms
selective cdk4
cdk4
selective
Prior art date
Application number
SG11201505680RA
Other languages
English (en)
Inventor
Brian Patrick Chekal
Nathan D Ide
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50151343&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201505680R(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of SG11201505680RA publication Critical patent/SG11201505680RA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SG11201505680RA 2013-02-21 2014-02-08 Solid forms of a selective cdk4/6 inhibitor SG11201505680RA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361767761P 2013-02-21 2013-02-21
PCT/IB2014/058865 WO2014128588A1 (en) 2013-02-21 2014-02-08 Solid forms of a selective cdk4/6 inhibitor

Publications (1)

Publication Number Publication Date
SG11201505680RA true SG11201505680RA (en) 2015-09-29

Family

ID=50151343

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201505680RA SG11201505680RA (en) 2013-02-21 2014-02-08 Solid forms of a selective cdk4/6 inhibitor

Country Status (24)

Country Link
US (2) US20160002223A1 (https=)
EP (2) EP2958916B1 (https=)
JP (3) JP6381016B2 (https=)
KR (2) KR20150107872A (https=)
CN (3) CN105008357A (https=)
AR (1) AR094842A1 (https=)
AU (1) AU2014220354B2 (https=)
BR (1) BR112015019508A8 (https=)
CA (1) CA2900322C (https=)
CY (2) CY1120734T1 (https=)
DK (2) DK2958916T3 (https=)
ES (2) ES2869277T3 (https=)
HK (2) HK1211032A1 (https=)
HU (2) HUE040434T2 (https=)
IL (1) IL240277B (https=)
MX (2) MX386473B (https=)
PL (2) PL3431475T3 (https=)
PT (2) PT3431475T (https=)
RU (1) RU2619944C2 (https=)
SG (1) SG11201505680RA (https=)
SI (2) SI2958916T1 (https=)
TR (1) TR201816077T4 (https=)
TW (2) TWI633103B (https=)
WO (1) WO2014128588A1 (https=)

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