SE447259B - Forfarande for framstellning av ett 1-n-/l-(-)-omega-amino-alfa-hydroxialkanoyl/kanamycin a eller b - Google Patents

Forfarande for framstellning av ett 1-n-/l-(-)-omega-amino-alfa-hydroxialkanoyl/kanamycin a eller b

Info

Publication number
SE447259B
SE447259B SE7804973A SE7804973A SE447259B SE 447259 B SE447259 B SE 447259B SE 7804973 A SE7804973 A SE 7804973A SE 7804973 A SE7804973 A SE 7804973A SE 447259 B SE447259 B SE 447259B
Authority
SE
Sweden
Prior art keywords
kanamycin
acid
mmol
silyl
mixture
Prior art date
Application number
SE7804973A
Other languages
English (en)
Swedish (sv)
Other versions
SE7804973L (sv
Inventor
Martin John Cron
John Gerard Keil
Jeng Shyong Lin
Mariano Vecchio Ruggeri
Derek Walker
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of SE7804973L publication Critical patent/SE7804973L/xx
Publication of SE447259B publication Critical patent/SE447259B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SE7804973A 1977-04-28 1978-04-28 Forfarande for framstellning av ett 1-n-/l-(-)-omega-amino-alfa-hydroxialkanoyl/kanamycin a eller b SE447259B (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79180677A 1977-04-28 1977-04-28
US88858578A 1978-03-20 1978-03-20

Publications (2)

Publication Number Publication Date
SE7804973L SE7804973L (sv) 1978-10-29
SE447259B true SE447259B (sv) 1986-11-03

Family

ID=27121201

Family Applications (2)

Application Number Title Priority Date Filing Date
SE7804973A SE447259B (sv) 1977-04-28 1978-04-28 Forfarande for framstellning av ett 1-n-/l-(-)-omega-amino-alfa-hydroxialkanoyl/kanamycin a eller b
SE8305538A SE461148B (sv) 1977-04-28 1983-10-07 Polysilylerat kanamycin a eller b derivat

Family Applications After (1)

Application Number Title Priority Date Filing Date
SE8305538A SE461148B (sv) 1977-04-28 1983-10-07 Polysilylerat kanamycin a eller b derivat

Country Status (27)

Country Link
JP (1) JPS53149951A (de)
AR (1) AR218910A1 (de)
AT (1) AT357675B (de)
CA (2) CA1100953A (de)
CH (1) CH639104A5 (de)
CS (1) CS207607B2 (de)
CY (1) CY1241A (de)
DE (2) DE2818992A1 (de)
DK (2) DK172543B1 (de)
EG (1) EG13710A (de)
ES (1) ES469303A1 (de)
FI (1) FI781288A (de)
FR (2) FR2388826A1 (de)
GB (1) GB1598294A (de)
HK (1) HK51484A (de)
IE (2) IE46945B1 (de)
IT (2) IT1156718B (de)
KE (1) KE3398A (de)
LU (1) LU79541A1 (de)
MY (1) MY8500528A (de)
NL (1) NL178790C (de)
NO (2) NO149635C (de)
PL (1) PL117307B1 (de)
PT (1) PT67959B (de)
SE (2) SE447259B (de)
SG (1) SG22884G (de)
YU (2) YU102578A (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS55306A (en) * 1978-04-28 1980-01-05 Bristol Myers Co Manufacture of 11nn*omegaaaminooalphaahydroxy alkanoyl**aminoglycoside antibiotic
CA2480002A1 (en) * 2002-02-19 2003-08-28 Amato Pharmaceutical Products, Ltd. Lactic acid derivative
AU2008326297B2 (en) 2007-11-21 2012-11-08 Cipla USA, Inc. Antibacterial aminoglycoside analogs
WO2010132760A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of tobramycin
WO2010132759A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of dibekacin
WO2010132768A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of sisomicin
WO2010132757A2 (en) * 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132765A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs

Also Published As

Publication number Publication date
NO154697C (no) 1986-12-03
DE2818822A1 (de) 1978-11-09
NL7804503A (nl) 1978-10-31
NO149635B (no) 1984-02-13
YU102578A (en) 1983-01-21
JPS5721277B2 (de) 1982-05-06
IE47271B1 (en) 1984-02-08
FR2388827A1 (fr) 1978-11-24
AR218910A1 (es) 1980-07-15
NO831197L (no) 1978-10-31
CS207607B2 (en) 1981-08-31
SE8305538L (sv) 1983-10-07
DE2818992C2 (de) 1988-03-17
FR2388826A1 (fr) 1978-11-24
DK183078A (da) 1978-10-29
SE461148B (sv) 1990-01-15
SE7804973L (sv) 1978-10-29
ES469303A1 (es) 1979-09-16
NO781437L (no) 1978-10-31
FR2388827B1 (de) 1982-07-09
DE2818992A1 (de) 1978-11-23
MY8500528A (en) 1985-12-31
HK51484A (en) 1984-06-22
CH639104A5 (en) 1983-10-31
IT1105500B (it) 1985-11-04
JPS53149951A (en) 1978-12-27
YU41590B (en) 1987-12-31
IE780841L (en) 1978-10-28
DK165450C (da) 1993-04-13
FR2388826B1 (de) 1982-12-10
IT1156718B (it) 1987-02-04
NL178790C (nl) 1986-05-16
DK172543B1 (da) 1998-12-07
DK165450B (da) 1992-11-30
NO149635C (no) 1984-05-23
SG22884G (en) 1985-01-04
ATA312778A (de) 1979-12-15
CA1105454A (en) 1981-07-21
SE8305538D0 (sv) 1983-10-07
AT357675B (de) 1980-07-25
EG13710A (en) 1982-09-30
CY1241A (en) 1984-06-29
PT67959B (en) 1980-03-05
IT7849137A0 (it) 1978-04-28
FI781288A (fi) 1978-10-29
YU102478A (en) 1982-10-31
PL206457A1 (de) 1980-03-24
KE3398A (en) 1984-06-08
NO154697B (no) 1986-08-25
LU79541A1 (fr) 1978-11-28
DK182978A (da) 1978-10-29
DE2818822C2 (de) 1989-01-26
PL117307B1 (en) 1981-07-31
IE780842L (en) 1978-10-28
NL178790B (nl) 1985-12-16
IE46945B1 (en) 1983-11-16
CA1100953A (en) 1981-05-12
PT67959A (en) 1978-05-01
GB1598294A (en) 1981-09-16
IT7849136A0 (it) 1978-04-28

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