RU2359967C2 - Производные тиофена и фармацевтическая композиция (варианты) - Google Patents

Производные тиофена и фармацевтическая композиция (варианты) Download PDF

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RU2359967C2
RU2359967C2 RU2004138787/04A RU2004138787A RU2359967C2 RU 2359967 C2 RU2359967 C2 RU 2359967C2 RU 2004138787/04 A RU2004138787/04 A RU 2004138787/04A RU 2004138787 A RU2004138787 A RU 2004138787A RU 2359967 C2 RU2359967 C2 RU 2359967C2
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Russia
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alkyl
methyl
phenyl
sulfonyl
amino
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RU2004138787/04A
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English (en)
Russian (ru)
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RU2004138787A (ru
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Фарах АЛИ (US)
Фарах АЛИ
Шелли К. БОЛЛЕНТАЙН (US)
Шелли К. БОЛЛЕНТАЙН
Джоан ГАШУ (US)
Джоан ГАШУ
Максвелл Д. КАММИНГС (US)
Максвелл Д. Каммингс
Кристи ЛЕОНАРД (US)
Кристи Леонард
Санат МИГАЛЛА (US)
Санат МИГАЛЛА
Уэнкси ПЭН (US)
Уэнкси ПЭН
М. Джонатан РУДОЛФ (US)
М. Джонатан РУДОЛФ
Налин СУБАСИНГХ (US)
Налин СУБАСИНГХ
Джерими М. ТРЭВИНС (US)
Джерими М. ТРЭВИНС
Кеннет Т. УИЛСОН (US)
Кеннет Т. УИЛСОН
Марк УОЛЛ (US)
Марк УОЛЛ
Эхаб ХАЛИЛ (US)
Эхаб Халил
Хуэй ХУАН (US)
Хуэй ХУАН
Хетер Рей ХУФНАГЕЛЬ (US)
Хетер Рей ХУФНАГЕЛЬ
Цзиньшэн ЧЭНЬ (US)
Цзиньшэн Чэнь
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Джонсон энд Джонсон Фамэсьютикэл Рисеч энд Дивелопмент, эЛ.эЛ.Си
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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D333/34—Sulfur atoms
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    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
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    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
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    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms
    • C07F9/655345—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms the sulfur atom being part of a five-membered ring

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Immunology (AREA)
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  • Hematology (AREA)
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  • Biomedical Technology (AREA)
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  • Molecular Biology (AREA)
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RU2004138787/04A 2002-05-28 2003-05-28 Производные тиофена и фармацевтическая композиция (варианты) RU2359967C2 (ru)

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US38313002P 2002-05-28 2002-05-28
US60/383.130 2002-05-28

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RU2359967C2 true RU2359967C2 (ru) 2009-06-27

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JP (1) JP2005538953A (enExample)
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EP2363396A1 (en) * 2001-06-11 2011-09-07 Virochem Pharma Inc. Thiophene derivatives as antiviral agents for flavivirus infection
DE10162114A1 (de) * 2001-12-12 2003-06-26 Schering Ag Neue Amidin-Derivate und deren Verwendung in Arzneimitteln
UA80131C2 (en) 2002-05-28 2007-08-27 Dimensional Pharm Inc Thiophene amidines, compositions thereof, and methods of treating complement-mediated diseases and conditions
DE60332482D1 (de) 2002-12-10 2010-06-17 Virochem Pharma Inc Verbindungen und methoden zum behandeln oder vorbeugen von flavivirus infektionen
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