RU2305682C2 - Производные 4-амино-5-фенил-7- циклобутилпирроло[2,3-d]пиримидина - Google Patents

Производные 4-амино-5-фенил-7- циклобутилпирроло[2,3-d]пиримидина Download PDF

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Publication number
RU2305682C2
RU2305682C2 RU2003134149/04A RU2003134149A RU2305682C2 RU 2305682 C2 RU2305682 C2 RU 2305682C2 RU 2003134149/04 A RU2003134149/04 A RU 2003134149/04A RU 2003134149 A RU2003134149 A RU 2003134149A RU 2305682 C2 RU2305682 C2 RU 2305682C2
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Prior art keywords
benzyloxyphenyl
pyrimidin
pyrrolo
amino
cyclobutylmethyl
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RU2003134149/04A
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English (en)
Russian (ru)
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RU2003134149A (ru
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Ханс-Георг КАПРАРО (CH)
Ханс-Георг Капраро
Паскаль ФЮРЕ (FR)
Паскаль Фюре
Карлос ГАРСИЯ-ЭЧЕВЕРРИЯ (CH)
Карлос ГАРСИЯ-ЭЧЕВЕРРИЯ
Пол Уилль м МАНЛИ (CH)
Пол Уилльям МАНЛИ
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Новартис Аг
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Priority claimed from GB0111764A external-priority patent/GB0111764D0/en
Priority claimed from GB0204752A external-priority patent/GB0204752D0/en
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Publication of RU2003134149A publication Critical patent/RU2003134149A/ru
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Publication of RU2305682C2 publication Critical patent/RU2305682C2/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RU2003134149/04A 2001-05-14 2002-05-13 Производные 4-амино-5-фенил-7- циклобутилпирроло[2,3-d]пиримидина RU2305682C2 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0111764A GB0111764D0 (en) 2001-05-14 2001-05-14 Organic compounds
GB0111764.7 2001-05-14
GB0204752.0 2002-02-28
GB0204752A GB0204752D0 (en) 2002-02-28 2002-02-28 Organic compounds

Publications (2)

Publication Number Publication Date
RU2003134149A RU2003134149A (ru) 2005-05-10
RU2305682C2 true RU2305682C2 (ru) 2007-09-10

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AT (1) ATE309245T1 (enExample)
AU (1) AU2002312905B2 (enExample)
BR (1) BR0209658A (enExample)
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RU (1) RU2305682C2 (enExample)
SK (1) SK14022003A3 (enExample)
TW (1) TWI238824B (enExample)
WO (1) WO2002092599A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2631655C2 (ru) * 2011-10-03 2017-09-26 Зэ Юниверсити Оф Норд Каролина Эт Чапель Хилл Пирролопиримидиновые соединения для лечения злокачественной опухоли

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