ATE309245T1 - 5-amino-5-phenyl-7-cyclobutyl-pyrrolo(2,3- d)pyrimidin-derivate - Google Patents

5-amino-5-phenyl-7-cyclobutyl-pyrrolo(2,3- d)pyrimidin-derivate

Info

Publication number
ATE309245T1
ATE309245T1 AT02738065T AT02738065T ATE309245T1 AT E309245 T1 ATE309245 T1 AT E309245T1 AT 02738065 T AT02738065 T AT 02738065T AT 02738065 T AT02738065 T AT 02738065T AT E309245 T1 ATE309245 T1 AT E309245T1
Authority
AT
Austria
Prior art keywords
pyrrolo
cyclobutyl
phenyl
amino
pyrimidine derivatives
Prior art date
Application number
AT02738065T
Other languages
English (en)
Inventor
Hans-Georg Capraro
Pascal Furet
Carlos Garcia-Echeverria
Paul William Manley
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0111764A external-priority patent/GB0111764D0/en
Priority claimed from GB0204752A external-priority patent/GB0204752D0/en
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE309245T1 publication Critical patent/ATE309245T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT02738065T 2001-05-14 2002-05-13 5-amino-5-phenyl-7-cyclobutyl-pyrrolo(2,3- d)pyrimidin-derivate ATE309245T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0111764A GB0111764D0 (en) 2001-05-14 2001-05-14 Organic compounds
GB0204752A GB0204752D0 (en) 2002-02-28 2002-02-28 Organic compounds
PCT/EP2002/005239 WO2002092599A1 (en) 2001-05-14 2002-05-13 4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives

Publications (1)

Publication Number Publication Date
ATE309245T1 true ATE309245T1 (de) 2005-11-15

Family

ID=26246078

Family Applications (1)

Application Number Title Priority Date Filing Date
AT02738065T ATE309245T1 (de) 2001-05-14 2002-05-13 5-amino-5-phenyl-7-cyclobutyl-pyrrolo(2,3- d)pyrimidin-derivate

Country Status (26)

Country Link
US (1) US7326699B2 (de)
EP (1) EP1390369B1 (de)
JP (1) JP4099399B2 (de)
KR (1) KR100583704B1 (de)
CN (1) CN1264844C (de)
AR (1) AR035885A1 (de)
AT (1) ATE309245T1 (de)
AU (1) AU2002312905B2 (de)
BR (1) BR0209658A (de)
CA (1) CA2446435C (de)
CO (1) CO5540346A2 (de)
CZ (1) CZ20033067A3 (de)
DE (1) DE60207241T2 (de)
ES (1) ES2252465T3 (de)
HU (1) HUP0304082A3 (de)
IL (1) IL158697A0 (de)
MX (1) MXPA03010402A (de)
MY (1) MY124853A (de)
NO (1) NO20034929L (de)
NZ (1) NZ529256A (de)
PE (1) PE20021096A1 (de)
PL (1) PL363866A1 (de)
RU (1) RU2305682C2 (de)
SK (1) SK14022003A3 (de)
TW (1) TWI238824B (de)
WO (1) WO2002092599A1 (de)

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