AU2002312905B2 - 4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives - Google Patents

4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives Download PDF

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Publication number
AU2002312905B2
AU2002312905B2 AU2002312905A AU2002312905A AU2002312905B2 AU 2002312905 B2 AU2002312905 B2 AU 2002312905B2 AU 2002312905 A AU2002312905 A AU 2002312905A AU 2002312905 A AU2002312905 A AU 2002312905A AU 2002312905 B2 AU2002312905 B2 AU 2002312905B2
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Prior art keywords
lower alkyl
amino
phenyl
pyrrolo
benzyloxy
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Ceased
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AU2002312905A
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AU2002312905A1 (en
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Hans-Georg Capraro
Pascal Furet
Carlos Garcia-Echeverria
Paul William Manley
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Novartis AG
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Novartis AG
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Priority claimed from GB0111764A external-priority patent/GB0111764D0/en
Priority claimed from GB0204752A external-priority patent/GB0204752D0/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2002312905A 2001-05-14 2002-05-13 4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives Ceased AU2002312905B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0111764A GB0111764D0 (en) 2001-05-14 2001-05-14 Organic compounds
GB0111764.7 2001-05-14
GB0204752A GB0204752D0 (en) 2002-02-28 2002-02-28 Organic compounds
GB0204752.0 2002-02-28
PCT/EP2002/005239 WO2002092599A1 (en) 2001-05-14 2002-05-13 4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives

Publications (2)

Publication Number Publication Date
AU2002312905A1 AU2002312905A1 (en) 2003-05-01
AU2002312905B2 true AU2002312905B2 (en) 2005-12-15

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AU2002312905A Ceased AU2002312905B2 (en) 2001-05-14 2002-05-13 4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives

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US (1) US7326699B2 (enExample)
EP (1) EP1390369B1 (enExample)
JP (1) JP4099399B2 (enExample)
KR (1) KR100583704B1 (enExample)
CN (1) CN1264844C (enExample)
AR (1) AR035885A1 (enExample)
AT (1) ATE309245T1 (enExample)
AU (1) AU2002312905B2 (enExample)
BR (1) BR0209658A (enExample)
CA (1) CA2446435C (enExample)
CO (1) CO5540346A2 (enExample)
CZ (1) CZ20033067A3 (enExample)
DE (1) DE60207241T2 (enExample)
ES (1) ES2252465T3 (enExample)
HU (1) HUP0304082A3 (enExample)
IL (1) IL158697A0 (enExample)
MX (1) MXPA03010402A (enExample)
MY (1) MY124853A (enExample)
NO (1) NO20034929D0 (enExample)
NZ (1) NZ529256A (enExample)
PE (1) PE20021096A1 (enExample)
PL (1) PL363866A1 (enExample)
RU (1) RU2305682C2 (enExample)
SK (1) SK14022003A3 (enExample)
TW (1) TWI238824B (enExample)
WO (1) WO2002092599A1 (enExample)

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