RU2230553C2 - Способ модулирования функции серин/треонин протеинкиназы соединением на основе азабензимидазола, способ идентификации соединений, модулирующих функцию серин/треонин протеинкиназы, способ профилактики или лечения патологических состояний в организме, соединение на основе азабензимидазола, способ его синтеза и фармацевтическая композиция - Google Patents

Способ модулирования функции серин/треонин протеинкиназы соединением на основе азабензимидазола, способ идентификации соединений, модулирующих функцию серин/треонин протеинкиназы, способ профилактики или лечения патологических состояний в организме, соединение на основе азабензимидазола, способ его синтеза и фармацевтическая композиция Download PDF

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Publication number
RU2230553C2
RU2230553C2 RU2000110736/15A RU2000110736A RU2230553C2 RU 2230553 C2 RU2230553 C2 RU 2230553C2 RU 2000110736/15 A RU2000110736/15 A RU 2000110736/15A RU 2000110736 A RU2000110736 A RU 2000110736A RU 2230553 C2 RU2230553 C2 RU 2230553C2
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group
protein kinase
serine
pyridine
alkyl
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RU2000110736/15A
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English (en)
Russian (ru)
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RU2000110736A (ru
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Хейнц ВЕЙНБЕРГЕР (DE)
Хейнц ВЕЙНБЕРГЕР
Бернгард Кучер (DE)
Бернгард Кучер
Джеральд МАКМЭЙХОН (US)
Джеральд МАКМЭЙХОН
Гаральд ЭПП (DE)
Гаральд ЭПП
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Центарис АГ
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
RU2000110736/15A 1997-09-26 1998-09-23 Способ модулирования функции серин/треонин протеинкиназы соединением на основе азабензимидазола, способ идентификации соединений, модулирующих функцию серин/треонин протеинкиназы, способ профилактики или лечения патологических состояний в организме, соединение на основе азабензимидазола, способ его синтеза и фармацевтическая композиция RU2230553C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6014597P 1997-09-26 1997-09-26
US60/060,145 1997-09-26

Publications (2)

Publication Number Publication Date
RU2000110736A RU2000110736A (ru) 2002-02-10
RU2230553C2 true RU2230553C2 (ru) 2004-06-20

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RU2000110736/15A RU2230553C2 (ru) 1997-09-26 1998-09-23 Способ модулирования функции серин/треонин протеинкиназы соединением на основе азабензимидазола, способ идентификации соединений, модулирующих функцию серин/треонин протеинкиназы, способ профилактики или лечения патологических состояний в организме, соединение на основе азабензимидазола, способ его синтеза и фармацевтическая композиция

Country Status (27)

Country Link
US (2) US6093728A (enExample)
EP (1) EP1017384B1 (enExample)
JP (1) JP2001517699A (enExample)
KR (1) KR100547929B1 (enExample)
CN (1) CN1167420C (enExample)
AR (1) AR017266A1 (enExample)
AT (1) ATE281834T1 (enExample)
AU (1) AU748849B2 (enExample)
BG (1) BG64784B1 (enExample)
BR (1) BR9812682A (enExample)
CA (1) CA2305370C (enExample)
DE (1) DE69827516T2 (enExample)
DK (1) DK1017384T3 (enExample)
ES (1) ES2230719T3 (enExample)
HU (1) HUP0004024A3 (enExample)
IL (4) IL158649A0 (enExample)
NO (1) NO325663B1 (enExample)
NZ (2) NZ503432A (enExample)
PL (1) PL191618B1 (enExample)
PT (1) PT1017384E (enExample)
RU (1) RU2230553C2 (enExample)
SK (1) SK285357B6 (enExample)
TR (1) TR200001546T2 (enExample)
TW (1) TW581815B (enExample)
UA (1) UA72448C2 (enExample)
WO (1) WO1999016438A1 (enExample)
ZA (1) ZA988797B (enExample)

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Also Published As

Publication number Publication date
CN1278172A (zh) 2000-12-27
US6855723B2 (en) 2005-02-15
CA2305370C (en) 2006-11-28
PL191618B1 (pl) 2006-06-30
ATE281834T1 (de) 2004-11-15
BG64784B1 (bg) 2006-04-28
AU748849B2 (en) 2002-06-13
SK285357B6 (sk) 2006-11-03
TR200001546T2 (tr) 2000-10-23
PL339744A1 (en) 2001-01-02
NZ517808A (en) 2003-07-25
JP2001517699A (ja) 2001-10-09
PT1017384E (pt) 2005-03-31
BR9812682A (pt) 2000-08-22
ZA988797B (en) 1999-12-02
NO325663B1 (no) 2008-07-07
AR017266A1 (es) 2001-09-05
IL135109A (en) 2007-07-04
NO20001555L (no) 2000-03-24
CA2305370A1 (en) 1999-04-08
KR100547929B1 (ko) 2006-02-02
KR20010015623A (ko) 2001-02-26
EP1017384B1 (en) 2004-11-10
IL158649A (en) 2006-12-10
UA72448C2 (en) 2005-03-15
HUP0004024A3 (en) 2001-10-29
TW581815B (en) 2004-04-01
US20030181480A1 (en) 2003-09-25
BG104356A (en) 2000-12-29
US6093728A (en) 2000-07-25
EP1017384A1 (en) 2000-07-12
HK1032206A1 (en) 2001-07-13
NO20001555D0 (no) 2000-03-24
HUP0004024A2 (hu) 2001-04-28
DK1017384T3 (da) 2005-01-31
IL158649A0 (en) 2004-05-12
DE69827516D1 (de) 2004-12-16
ES2230719T3 (es) 2005-05-01
AU9578198A (en) 1999-04-23
WO1999016438A1 (en) 1999-04-08
NZ503432A (en) 2002-11-26
IL135109A0 (en) 2001-05-20
CN1167420C (zh) 2004-09-22
DE69827516T2 (de) 2005-12-01
SK4152000A3 (en) 2002-02-05

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