RS57559B1 - 1,3,4-oksadiazol i 1,3,4-tiadiazol derivativi kao imunomodulatori - Google Patents

1,3,4-oksadiazol i 1,3,4-tiadiazol derivativi kao imunomodulatori

Info

Publication number
RS57559B1
RS57559B1 RS20180936A RSP20180936A RS57559B1 RS 57559 B1 RS57559 B1 RS 57559B1 RS 20180936 A RS20180936 A RS 20180936A RS P20180936 A RSP20180936 A RS P20180936A RS 57559 B1 RS57559 B1 RS 57559B1
Authority
RS
Serbia
Prior art keywords
immunomodulators
oxadiazole
thiadiazole derivatives
thiadiazole
derivatives
Prior art date
Application number
RS20180936A
Other languages
English (en)
Inventor
Pottayil Govindan Nair Sasikumar
Muralidhara Ramachandra
Seetharamaiah Setty Sudarshan Naremaddepalli
Original Assignee
Aurigene Discovery Tech Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aurigene Discovery Tech Ltd filed Critical Aurigene Discovery Tech Ltd
Publication of RS57559B1 publication Critical patent/RS57559B1/sr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433Thidiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/101,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
RS20180936A 2013-09-06 2014-09-05 1,3,4-oksadiazol i 1,3,4-tiadiazol derivativi kao imunomodulatori RS57559B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN4012CH2013 2013-09-06
PCT/IB2014/064281 WO2015033301A1 (en) 2013-09-06 2014-09-05 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives as immunomodulators
EP14842822.0A EP3041828B1 (en) 2013-09-06 2014-09-05 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives as immunomodulators

Publications (1)

Publication Number Publication Date
RS57559B1 true RS57559B1 (sr) 2018-10-31

Family

ID=52627870

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20180936A RS57559B1 (sr) 2013-09-06 2014-09-05 1,3,4-oksadiazol i 1,3,4-tiadiazol derivativi kao imunomodulatori

Country Status (25)

Country Link
US (3) US20160194295A1 (sr)
EP (2) EP3041828B1 (sr)
JP (1) JP2016532711A (sr)
KR (1) KR20160081898A (sr)
CN (1) CN105849092A (sr)
AU (1) AU2014316684A1 (sr)
CA (1) CA2922655A1 (sr)
CU (1) CU24345B1 (sr)
CY (1) CY1120769T1 (sr)
DK (1) DK3041828T3 (sr)
EA (1) EA029661B1 (sr)
ES (1) ES2682040T3 (sr)
HR (1) HRP20181251T1 (sr)
HU (1) HUE039014T2 (sr)
IL (1) IL244313A0 (sr)
LT (1) LT3041828T (sr)
MX (1) MX2016002971A (sr)
PH (1) PH12016500405B1 (sr)
PL (1) PL3041828T3 (sr)
PT (1) PT3041828T (sr)
RS (1) RS57559B1 (sr)
SG (2) SG11201601679TA (sr)
SI (1) SI3041828T1 (sr)
TR (1) TR201811077T4 (sr)
WO (1) WO2015033301A1 (sr)

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