HUE039014T2 - 1,3,4-Oxadiazol és 1,3,4-tiadiazol származékok, mint immunomodulátorok - Google Patents

1,3,4-Oxadiazol és 1,3,4-tiadiazol származékok, mint immunomodulátorok

Info

Publication number
HUE039014T2
HUE039014T2 HUE14842822A HUE14842822A HUE039014T2 HU E039014 T2 HUE039014 T2 HU E039014T2 HU E14842822 A HUE14842822 A HU E14842822A HU E14842822 A HUE14842822 A HU E14842822A HU E039014 T2 HUE039014 T2 HU E039014T2
Authority
HU
Hungary
Prior art keywords
immunomodulators
oxadiazole
thiadiazole derivatives
thiadiazole
derivatives
Prior art date
Application number
HUE14842822A
Other languages
English (en)
Inventor
Pottayil Govindan Nair Sasikumar
Muralidhara Ramachandra
Seetharamaiah Setty Sudarshan Naremaddepalli
Original Assignee
Aurigene Discovery Tech Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aurigene Discovery Tech Ltd filed Critical Aurigene Discovery Tech Ltd
Publication of HUE039014T2 publication Critical patent/HUE039014T2/hu

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/101,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433Thidiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
HUE14842822A 2013-09-06 2014-09-05 1,3,4-Oxadiazol és 1,3,4-tiadiazol származékok, mint immunomodulátorok HUE039014T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN4012CH2013 2013-09-06

Publications (1)

Publication Number Publication Date
HUE039014T2 true HUE039014T2 (hu) 2018-12-28

Family

ID=52627870

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE14842822A HUE039014T2 (hu) 2013-09-06 2014-09-05 1,3,4-Oxadiazol és 1,3,4-tiadiazol származékok, mint immunomodulátorok

Country Status (25)

Country Link
US (3) US20160194295A1 (hu)
EP (2) EP3041828B1 (hu)
JP (1) JP2016532711A (hu)
KR (1) KR20160081898A (hu)
CN (1) CN105849092A (hu)
AU (1) AU2014316684A1 (hu)
CA (1) CA2922655A1 (hu)
CU (1) CU24345B1 (hu)
CY (1) CY1120769T1 (hu)
DK (1) DK3041828T3 (hu)
EA (1) EA029661B1 (hu)
ES (1) ES2682040T3 (hu)
HR (1) HRP20181251T1 (hu)
HU (1) HUE039014T2 (hu)
IL (1) IL244313A0 (hu)
LT (1) LT3041828T (hu)
MX (1) MX2016002971A (hu)
PH (1) PH12016500405A1 (hu)
PL (1) PL3041828T3 (hu)
PT (1) PT3041828T (hu)
RS (1) RS57559B1 (hu)
SG (2) SG10201800508SA (hu)
SI (1) SI3041828T1 (hu)
TR (1) TR201811077T4 (hu)
WO (1) WO2015033301A1 (hu)

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