PT2603513T - Composto heterocíclico e sua utilização como modulador alostérico positivo do recetor de ampa - Google Patents

Composto heterocíclico e sua utilização como modulador alostérico positivo do recetor de ampa

Info

Publication number
PT2603513T
PT2603513T PT117499442T PT11749944T PT2603513T PT 2603513 T PT2603513 T PT 2603513T PT 117499442 T PT117499442 T PT 117499442T PT 11749944 T PT11749944 T PT 11749944T PT 2603513 T PT2603513 T PT 2603513T
Authority
PT
Portugal
Prior art keywords
heterocyclic compound
heterocyclic
compound
Prior art date
Application number
PT117499442T
Other languages
English (en)
Portuguese (pt)
Original Assignee
Takeda Pharmaceuticals Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceuticals Co filed Critical Takeda Pharmaceuticals Co
Publication of PT2603513T publication Critical patent/PT2603513T/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
PT117499442T 2010-08-10 2011-08-09 Composto heterocíclico e sua utilização como modulador alostérico positivo do recetor de ampa PT2603513T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2010179577 2010-08-10

Publications (1)

Publication Number Publication Date
PT2603513T true PT2603513T (pt) 2020-06-08

Family

ID=44534564

Family Applications (1)

Application Number Title Priority Date Filing Date
PT117499442T PT2603513T (pt) 2010-08-10 2011-08-09 Composto heterocíclico e sua utilização como modulador alostérico positivo do recetor de ampa

Country Status (39)

Country Link
US (11) US9150591B2 (cg-RX-API-DMAC7.html)
EP (1) EP2603513B1 (cg-RX-API-DMAC7.html)
JP (2) JP5788496B2 (cg-RX-API-DMAC7.html)
KR (1) KR101852215B1 (cg-RX-API-DMAC7.html)
CN (2) CN103180326B (cg-RX-API-DMAC7.html)
AR (1) AR082618A1 (cg-RX-API-DMAC7.html)
AU (1) AU2011290126B2 (cg-RX-API-DMAC7.html)
BR (1) BR112013002250B1 (cg-RX-API-DMAC7.html)
CA (1) CA2807460C (cg-RX-API-DMAC7.html)
CL (1) CL2013000380A1 (cg-RX-API-DMAC7.html)
CO (1) CO6680700A2 (cg-RX-API-DMAC7.html)
CR (1) CR20130066A (cg-RX-API-DMAC7.html)
CY (1) CY1123507T1 (cg-RX-API-DMAC7.html)
DK (1) DK2603513T3 (cg-RX-API-DMAC7.html)
DO (1) DOP2013000030A (cg-RX-API-DMAC7.html)
EA (1) EA022078B1 (cg-RX-API-DMAC7.html)
EC (1) ECSP13012478A (cg-RX-API-DMAC7.html)
ES (1) ES2793723T3 (cg-RX-API-DMAC7.html)
GE (1) GEP20156216B (cg-RX-API-DMAC7.html)
HR (1) HRP20200844T1 (cg-RX-API-DMAC7.html)
HU (1) HUE049460T2 (cg-RX-API-DMAC7.html)
IL (1) IL224452A (cg-RX-API-DMAC7.html)
LT (1) LT2603513T (cg-RX-API-DMAC7.html)
MA (1) MA34509B1 (cg-RX-API-DMAC7.html)
MX (1) MX349470B (cg-RX-API-DMAC7.html)
MY (1) MY165908A (cg-RX-API-DMAC7.html)
NZ (1) NZ607593A (cg-RX-API-DMAC7.html)
PE (1) PE20131116A1 (cg-RX-API-DMAC7.html)
PH (1) PH12013500247A1 (cg-RX-API-DMAC7.html)
PL (1) PL2603513T3 (cg-RX-API-DMAC7.html)
PT (1) PT2603513T (cg-RX-API-DMAC7.html)
RS (1) RS60311B1 (cg-RX-API-DMAC7.html)
SG (1) SG187656A1 (cg-RX-API-DMAC7.html)
SI (1) SI2603513T1 (cg-RX-API-DMAC7.html)
TW (1) TWI504604B (cg-RX-API-DMAC7.html)
UA (1) UA111594C2 (cg-RX-API-DMAC7.html)
UY (1) UY33551A (cg-RX-API-DMAC7.html)
WO (1) WO2012020848A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA201301120B (cg-RX-API-DMAC7.html)

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CN110312712B (zh) 2016-12-21 2023-06-23 Fmc公司 硝酮除草剂
CN107892697B (zh) 2016-12-26 2020-11-03 郑州泰基鸿诺医药股份有限公司 一种[1,3]噻嗪-2-胺类化合物及应用,药物组合物
JP7201609B2 (ja) 2017-03-21 2023-01-10 エフ エム シー コーポレーション ピロリジノン及びこれらを調製するためのプロセス
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EP3693360B1 (en) * 2017-10-06 2023-12-13 Takeda Pharmaceutical Company Limited Heterocyclic compounds
EP3693368B1 (en) * 2017-10-06 2023-12-06 Takeda Pharmaceutical Company Limited Heterocyclic compound
PL4031552T3 (pl) 2019-09-16 2025-03-17 Takeda Pharmaceutical Company Limited Pochodne azolowo-skondensowanych pirydazyn-3(2h)-onów
JP2023526249A (ja) * 2020-05-15 2023-06-21 武田薬品工業株式会社 うつ病の処置
CN113943294A (zh) * 2020-07-15 2022-01-18 成都海博为药业有限公司 一种作为btk抑制剂的化合物及其制备方法与用途
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Also Published As

Publication number Publication date
US20150353578A1 (en) 2015-12-10
NZ607593A (en) 2015-01-30
US20170022222A1 (en) 2017-01-26
MY165908A (en) 2018-05-18
WO2012020848A1 (en) 2012-02-16
BR112013002250A2 (pt) 2016-05-24
GEP20156216B (en) 2015-01-12
TW201217386A (en) 2012-05-01
EP2603513B1 (en) 2020-03-11
MA34509B1 (fr) 2013-09-02
AU2011290126A1 (en) 2013-03-07
MX2013001614A (es) 2013-07-05
HUE049460T2 (hu) 2020-09-28
US20190263832A1 (en) 2019-08-29
SI2603513T1 (sl) 2020-07-31
UA111594C2 (uk) 2016-05-25
CN103180326A (zh) 2013-06-26
KR101852215B1 (ko) 2018-04-25
DK2603513T3 (da) 2020-06-15
US8575154B2 (en) 2013-11-05
US20130184266A1 (en) 2013-07-18
US20240360156A1 (en) 2024-10-31
CN104926837A (zh) 2015-09-23
US20130190291A1 (en) 2013-07-25
CR20130066A (es) 2013-05-03
CA2807460C (en) 2018-09-18
US8778934B2 (en) 2014-07-15
ES2793723T3 (es) 2020-11-16
HRP20200844T1 (hr) 2020-08-21
US11279713B2 (en) 2022-03-22
US20150073137A1 (en) 2015-03-12
PE20131116A1 (es) 2013-10-24
SG187656A1 (en) 2013-03-28
TWI504604B (zh) 2015-10-21
US9499568B2 (en) 2016-11-22
PL2603513T3 (pl) 2020-07-27
CL2013000380A1 (es) 2013-05-31
PH12013500247A1 (en) 2013-03-11
ECSP13012478A (es) 2013-04-30
US9884875B2 (en) 2018-02-06
RS60311B1 (sr) 2020-07-31
KR20130138738A (ko) 2013-12-19
JP5788496B2 (ja) 2015-09-30
CY1123507T1 (el) 2022-03-24
US20180162875A1 (en) 2018-06-14
CO6680700A2 (es) 2013-05-31
US20200317692A1 (en) 2020-10-08
DOP2013000030A (es) 2013-03-15
EA201390222A1 (ru) 2013-08-30
EA022078B1 (ru) 2015-10-30
JP2016006080A (ja) 2016-01-14
US20120077799A1 (en) 2012-03-29
LT2603513T (lt) 2020-05-25
AR082618A1 (es) 2012-12-19
JP6113789B2 (ja) 2017-04-12
BR112013002250B1 (pt) 2020-10-27
ZA201301120B (en) 2014-04-30
MX349470B (es) 2017-07-31
CA2807460A1 (en) 2012-02-16
AU2011290126B2 (en) 2016-01-07
WO2012020848A8 (en) 2012-09-27
UY33551A (es) 2012-03-30
IL224452A (en) 2017-11-30
US20140080817A1 (en) 2014-03-20
EP2603513A1 (en) 2013-06-19
JP2013535408A (ja) 2013-09-12
US8916551B2 (en) 2014-12-23
US10654874B2 (en) 2020-05-19
CN103180326B (zh) 2015-06-10
US9150591B2 (en) 2015-10-06

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