PL218764B1 - Związek będacy antagonistą receptora adenozynowego A<sub>2a</sub>, zawierająca go kompozycja farmaceutyczna i jego zastosowanie oraz sposób wytwarzania związków pośrednich - Google Patents
Związek będacy antagonistą receptora adenozynowego A<sub>2a</sub>, zawierająca go kompozycja farmaceutyczna i jego zastosowanie oraz sposób wytwarzania związków pośrednichInfo
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- PL218764B1 PL218764B1 PL360472A PL36047201A PL218764B1 PL 218764 B1 PL218764 B1 PL 218764B1 PL 360472 A PL360472 A PL 360472A PL 36047201 A PL36047201 A PL 36047201A PL 218764 B1 PL218764 B1 PL 218764B1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US20714300P | 2000-05-26 | 2000-05-26 | |
| PCT/US2001/016954 WO2001092264A1 (en) | 2000-05-26 | 2001-05-24 | Adenosine a2a receptor antagonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL360472A1 PL360472A1 (en) | 2004-09-06 |
| PL218764B1 true PL218764B1 (pl) | 2015-01-30 |
Family
ID=22769372
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL360472A PL218764B1 (pl) | 2000-05-26 | 2001-05-24 | Związek będacy antagonistą receptora adenozynowego A<sub>2a</sub>, zawierająca go kompozycja farmaceutyczna i jego zastosowanie oraz sposób wytwarzania związków pośrednich |
Country Status (31)
| Country | Link |
|---|---|
| US (4) | US6630475B2 (https=) |
| EP (1) | EP1283839B1 (https=) |
| JP (3) | JP4574112B2 (https=) |
| KR (1) | KR100520907B1 (https=) |
| CN (2) | CN100384847C (https=) |
| AR (1) | AR028621A1 (https=) |
| AT (1) | ATE293627T1 (https=) |
| AU (2) | AU2001268089C1 (https=) |
| BR (1) | BRPI0111015B8 (https=) |
| CA (1) | CA2410237C (https=) |
| CZ (1) | CZ303790B6 (https=) |
| DE (1) | DE60110219T2 (https=) |
| DK (1) | DK1283839T3 (https=) |
| EC (1) | ECSP024364A (https=) |
| ES (1) | ES2237576T3 (https=) |
| HK (1) | HK1049007B (https=) |
| HU (1) | HU230420B1 (https=) |
| IL (3) | IL152726A0 (https=) |
| MX (1) | MXPA02011625A (https=) |
| MY (1) | MY132006A (https=) |
| NO (1) | NO325008B1 (https=) |
| NZ (1) | NZ522326A (https=) |
| PE (1) | PE20020062A1 (https=) |
| PL (1) | PL218764B1 (https=) |
| PT (1) | PT1283839E (https=) |
| RU (1) | RU2315053C2 (https=) |
| SI (1) | SI1283839T1 (https=) |
| SK (1) | SK287748B6 (https=) |
| TW (1) | TWI288137B (https=) |
| WO (1) | WO2001092264A1 (https=) |
| ZA (1) | ZA200208898B (https=) |
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| ES2273599B1 (es) | 2005-10-14 | 2008-06-01 | Universidad De Barcelona | Compuestos para el tratamiento de la fibrilacion auricular. |
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| CA2468649C (en) * | 2001-11-30 | 2009-03-10 | Schering Corporation | Adenosine a2a receptor antagonists |
| JP2006514697A (ja) * | 2002-12-19 | 2006-05-11 | シェーリング コーポレイション | アデノシンＡ２ａレセプターアンタゴニストの使用 |
| CN1898246B (zh) * | 2003-10-28 | 2010-10-27 | 先灵公司 | 制备取代的5-氨基-吡唑并[4，3-e]-1，2，4-三唑并[1，5-c]嘧啶的方法 |
| WO2005054245A2 (en) * | 2003-12-01 | 2005-06-16 | Schering Corporation | Process for preparing substituted 5-amino-pyrazolo-[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines |
| EP1745047B1 (en) * | 2004-04-21 | 2010-03-24 | Schering Corporation | Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine adenosine-a2a- receptor antagonists |
| ATE538123T1 (de) * | 2005-09-19 | 2012-01-15 | Schering Corp | 2-heteroarylpyrazoloä4,3-eü-1, 2, 4-triazolo-ä1,5-cü-pyrimidine als antagonisten des adenosin-a2a- rezeptors |
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2001
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