PL197693B1 - Zastosowanie pochodnych 4-H-1 benzopiran-4-onu - Google Patents

Zastosowanie pochodnych 4-H-1 benzopiran-4-onu

Info

Publication number
PL197693B1
PL197693B1 PL350735A PL35073500A PL197693B1 PL 197693 B1 PL197693 B1 PL 197693B1 PL 350735 A PL350735 A PL 350735A PL 35073500 A PL35073500 A PL 35073500A PL 197693 B1 PL197693 B1 PL 197693B1
Authority
PL
Poland
Prior art keywords
alkyl
flavopiridol
alkylamino
proliferation
smc
Prior art date
Application number
PL350735A
Other languages
English (en)
Polish (pl)
Other versions
PL350735A1 (en
Inventor
Winston Campbell Patterson
Jennifer A. Dumont
Original Assignee
Aventis Pharma Inc
Univ Texas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Inc, Univ Texas filed Critical Aventis Pharma Inc
Publication of PL350735A1 publication Critical patent/PL350735A1/xx
Publication of PL197693B1 publication Critical patent/PL197693B1/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/453Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL350735A 1999-02-01 2000-01-18 Zastosowanie pochodnych 4-H-1 benzopiran-4-onu PL197693B1 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24338099A 1999-02-01 1999-02-01
US09/468,665 US6399633B1 (en) 1999-02-01 1999-12-21 Use of 4-H-1-benzopryan-4-one derivatives as inhibitors of smooth muscle cell proliferation
PCT/US2000/001104 WO2000044362A2 (en) 1999-02-01 2000-01-18 The use of 4-h-1-benzopyran-4-one derivatives as inhibitors of smooth muscle cell proliferation

Publications (2)

Publication Number Publication Date
PL350735A1 PL350735A1 (en) 2003-01-27
PL197693B1 true PL197693B1 (pl) 2008-04-30

Family

ID=22918541

Family Applications (1)

Application Number Title Priority Date Filing Date
PL350735A PL197693B1 (pl) 1999-02-01 2000-01-18 Zastosowanie pochodnych 4-H-1 benzopiran-4-onu

Country Status (38)

Country Link
US (1) US6399633B1 (enExample)
EP (1) EP1150746B1 (enExample)
JP (1) JP4755759B2 (enExample)
KR (1) KR100793047B1 (enExample)
CN (1) CN1219556C (enExample)
AP (1) AP1469A (enExample)
AR (1) AR042569A1 (enExample)
AT (1) ATE275428T1 (enExample)
AU (1) AU777368B2 (enExample)
BG (1) BG65151B1 (enExample)
BR (1) BR0007911A (enExample)
CA (1) CA2360668C (enExample)
CR (1) CR6448A (enExample)
CZ (1) CZ300395B6 (enExample)
DE (1) DE60013555T2 (enExample)
DK (1) DK1150746T3 (enExample)
EA (1) EA004786B1 (enExample)
EE (1) EE04851B1 (enExample)
ES (1) ES2226792T3 (enExample)
HK (1) HK1042445B (enExample)
HR (1) HRP20010521A2 (enExample)
HU (1) HU229263B1 (enExample)
ID (1) ID30180A (enExample)
IL (1) IL144668A (enExample)
ME (1) MEP10508A (enExample)
NO (1) NO330512B1 (enExample)
NZ (1) NZ512822A (enExample)
OA (1) OA11755A (enExample)
PL (1) PL197693B1 (enExample)
PT (1) PT1150746E (enExample)
RS (1) RS50242B (enExample)
SI (1) SI1150746T1 (enExample)
SK (1) SK286747B6 (enExample)
TR (1) TR200102223T2 (enExample)
TW (1) TWI273907B (enExample)
UA (1) UA73110C2 (enExample)
WO (1) WO2000044362A2 (enExample)
ZA (1) ZA200105596B (enExample)

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Also Published As

Publication number Publication date
SI1150746T1 (en) 2005-02-28
JP2002535356A (ja) 2002-10-22
MEP10508A (en) 2010-06-10
NZ512822A (en) 2005-01-28
CZ20012804A3 (cs) 2002-08-14
DE60013555T2 (de) 2005-09-29
US6399633B1 (en) 2002-06-04
CR6448A (es) 2004-03-17
YU54401A (sh) 2004-05-12
HK1042445B (zh) 2006-01-13
DE60013555D1 (de) 2004-10-14
DK1150746T3 (da) 2005-01-10
HRP20010521A2 (en) 2002-08-31
EE200100385A (et) 2002-12-16
SK286747B6 (sk) 2009-04-06
NO20013335D0 (no) 2001-07-05
AP1469A (en) 2005-09-26
EP1150746A2 (en) 2001-11-07
WO2000044362A2 (en) 2000-08-03
BG65151B1 (bg) 2007-04-30
BR0007911A (pt) 2001-10-16
EA004786B1 (ru) 2004-08-26
AP2001002218A0 (en) 2001-09-30
WO2000044362A3 (en) 2001-04-05
ID30180A (id) 2001-11-08
ES2226792T3 (es) 2005-04-01
BG105751A (en) 2002-02-28
AR042569A1 (es) 2005-06-29
CN1338958A (zh) 2002-03-06
UA73110C2 (en) 2005-06-15
KR20010093309A (ko) 2001-10-27
TWI273907B (en) 2007-02-21
HUP0200804A2 (hu) 2002-12-28
TR200102223T2 (tr) 2004-12-21
OA11755A (en) 2005-07-19
CN1219556C (zh) 2005-09-21
NO20013335L (no) 2001-09-25
PT1150746E (pt) 2004-12-31
AU777368B2 (en) 2004-10-14
HK1042445A1 (en) 2002-08-16
EP1150746B1 (en) 2004-09-08
RS50242B (sr) 2009-07-15
ZA200105596B (en) 2002-10-07
HU229263B1 (en) 2013-10-28
CA2360668C (en) 2009-03-17
KR100793047B1 (ko) 2008-01-10
SK10862001A3 (sk) 2002-07-02
CA2360668A1 (en) 2000-08-03
HUP0200804A3 (en) 2004-03-29
NO330512B1 (no) 2011-05-09
EA200100742A1 (ru) 2001-12-24
ATE275428T1 (de) 2004-09-15
JP4755759B2 (ja) 2011-08-24
CZ300395B6 (cs) 2009-05-06
IL144668A0 (en) 2002-05-23
PL350735A1 (en) 2003-01-27
AU3209800A (en) 2000-08-18
EE04851B1 (et) 2007-06-15
IL144668A (en) 2005-06-19

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