IL144668A - Use of a 4-h-1-benzopyran-4-one derivative for the preparation of a medicament for inhibiting smooth muscle cell proliferation - Google Patents

Use of a 4-h-1-benzopyran-4-one derivative for the preparation of a medicament for inhibiting smooth muscle cell proliferation

Info

Publication number
IL144668A
IL144668A IL14466800A IL14466800A IL144668A IL 144668 A IL144668 A IL 144668A IL 14466800 A IL14466800 A IL 14466800A IL 14466800 A IL14466800 A IL 14466800A IL 144668 A IL144668 A IL 144668A
Authority
IL
Israel
Prior art keywords
benzopyran
medicament
derivative
preparation
cell proliferation
Prior art date
Application number
IL14466800A
Other languages
English (en)
Other versions
IL144668A0 (en
Original Assignee
Aventis Pharma Inc
Univ Texas
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Inc, Univ Texas filed Critical Aventis Pharma Inc
Publication of IL144668A0 publication Critical patent/IL144668A0/xx
Publication of IL144668A publication Critical patent/IL144668A/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/453Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL14466800A 1999-02-01 2000-01-18 Use of a 4-h-1-benzopyran-4-one derivative for the preparation of a medicament for inhibiting smooth muscle cell proliferation IL144668A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24338099A 1999-02-01 1999-02-01
US09/468,665 US6399633B1 (en) 1999-02-01 1999-12-21 Use of 4-H-1-benzopryan-4-one derivatives as inhibitors of smooth muscle cell proliferation
PCT/US2000/001104 WO2000044362A2 (en) 1999-02-01 2000-01-18 The use of 4-h-1-benzopyran-4-one derivatives as inhibitors of smooth muscle cell proliferation

Publications (2)

Publication Number Publication Date
IL144668A0 IL144668A0 (en) 2002-05-23
IL144668A true IL144668A (en) 2005-06-19

Family

ID=22918541

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14466800A IL144668A (en) 1999-02-01 2000-01-18 Use of a 4-h-1-benzopyran-4-one derivative for the preparation of a medicament for inhibiting smooth muscle cell proliferation

Country Status (38)

Country Link
US (1) US6399633B1 (enExample)
EP (1) EP1150746B1 (enExample)
JP (1) JP4755759B2 (enExample)
KR (1) KR100793047B1 (enExample)
CN (1) CN1219556C (enExample)
AP (1) AP1469A (enExample)
AR (1) AR042569A1 (enExample)
AT (1) ATE275428T1 (enExample)
AU (1) AU777368B2 (enExample)
BG (1) BG65151B1 (enExample)
BR (1) BR0007911A (enExample)
CA (1) CA2360668C (enExample)
CR (1) CR6448A (enExample)
CZ (1) CZ300395B6 (enExample)
DE (1) DE60013555T2 (enExample)
DK (1) DK1150746T3 (enExample)
EA (1) EA004786B1 (enExample)
EE (1) EE04851B1 (enExample)
ES (1) ES2226792T3 (enExample)
HK (1) HK1042445B (enExample)
HR (1) HRP20010521A2 (enExample)
HU (1) HU229263B1 (enExample)
ID (1) ID30180A (enExample)
IL (1) IL144668A (enExample)
ME (1) MEP10508A (enExample)
NO (1) NO330512B1 (enExample)
NZ (1) NZ512822A (enExample)
OA (1) OA11755A (enExample)
PL (1) PL197693B1 (enExample)
PT (1) PT1150746E (enExample)
RS (1) RS50242B (enExample)
SI (1) SI1150746T1 (enExample)
SK (1) SK286747B6 (enExample)
TR (1) TR200102223T2 (enExample)
TW (1) TWI273907B (enExample)
UA (1) UA73110C2 (enExample)
WO (1) WO2000044362A2 (enExample)
ZA (1) ZA200105596B (enExample)

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US20130225530A1 (en) 2010-07-12 2013-08-29 Dkfz Deutsches Krebsforschungszentrum Wogonin for the prevention and therapy of cardiac hypertrophy
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DK2877493T3 (en) 2012-07-25 2018-06-14 Celldex Therapeutics Inc ANTI-KIT ANTIBODIES AND APPLICATIONS THEREOF
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WO2014080290A2 (en) 2012-11-21 2014-05-30 Rvx Therapeutics Inc. Cyclic amines as bromodomain inhibitors
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CA2895905A1 (en) 2012-12-21 2014-06-26 Zenith Epigenetics Corp. Novel heterocyclic compounds as bromodomain inhibitors
NZ714765A (en) 2013-06-06 2021-12-24 Pf Medicament Anti-c10orf54 antibodies and uses thereof
HUE056325T2 (hu) 2013-08-26 2022-02-28 Biontech Res And Development Inc SIALYL-LEWIS A elleni humán antitesteket kódoló nukleinsavak
GB201403775D0 (en) 2014-03-04 2014-04-16 Kymab Ltd Antibodies, uses & methods
PT3154583T (pt) 2014-06-04 2021-03-24 Biontech Res And Development Inc Anticorpos monoclonais humanos para o gangliósido gd2
TN2017000246A1 (en) 2014-12-11 2018-10-19 Pf Medicament Anti-c10orf54 antibodies and uses thereof
KR20250005465A (ko) 2015-03-03 2025-01-09 키맵 리미티드 항체, 용도 및 방법
EP3268007B1 (en) 2015-03-13 2022-11-09 Resverlogix Corp. Compositions and therapeutic methods for the treatment of complement-associated diseases
RU2717829C2 (ru) 2015-04-20 2020-03-26 Толеро Фармасьютикалз, Инк. Прогнозирование ответа на альвоцидиб с помощью анализа профиля митохондрий
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Also Published As

Publication number Publication date
SI1150746T1 (en) 2005-02-28
JP2002535356A (ja) 2002-10-22
MEP10508A (en) 2010-06-10
NZ512822A (en) 2005-01-28
CZ20012804A3 (cs) 2002-08-14
DE60013555T2 (de) 2005-09-29
US6399633B1 (en) 2002-06-04
PL197693B1 (pl) 2008-04-30
CR6448A (es) 2004-03-17
YU54401A (sh) 2004-05-12
HK1042445B (zh) 2006-01-13
DE60013555D1 (de) 2004-10-14
DK1150746T3 (da) 2005-01-10
HRP20010521A2 (en) 2002-08-31
EE200100385A (et) 2002-12-16
SK286747B6 (sk) 2009-04-06
NO20013335D0 (no) 2001-07-05
AP1469A (en) 2005-09-26
EP1150746A2 (en) 2001-11-07
WO2000044362A2 (en) 2000-08-03
BG65151B1 (bg) 2007-04-30
BR0007911A (pt) 2001-10-16
EA004786B1 (ru) 2004-08-26
AP2001002218A0 (en) 2001-09-30
WO2000044362A3 (en) 2001-04-05
ID30180A (id) 2001-11-08
ES2226792T3 (es) 2005-04-01
BG105751A (en) 2002-02-28
AR042569A1 (es) 2005-06-29
CN1338958A (zh) 2002-03-06
UA73110C2 (en) 2005-06-15
KR20010093309A (ko) 2001-10-27
TWI273907B (en) 2007-02-21
HUP0200804A2 (hu) 2002-12-28
TR200102223T2 (tr) 2004-12-21
OA11755A (en) 2005-07-19
CN1219556C (zh) 2005-09-21
NO20013335L (no) 2001-09-25
PT1150746E (pt) 2004-12-31
AU777368B2 (en) 2004-10-14
HK1042445A1 (en) 2002-08-16
EP1150746B1 (en) 2004-09-08
RS50242B (sr) 2009-07-15
ZA200105596B (en) 2002-10-07
HU229263B1 (en) 2013-10-28
CA2360668C (en) 2009-03-17
KR100793047B1 (ko) 2008-01-10
SK10862001A3 (sk) 2002-07-02
CA2360668A1 (en) 2000-08-03
HUP0200804A3 (en) 2004-03-29
NO330512B1 (no) 2011-05-09
EA200100742A1 (ru) 2001-12-24
ATE275428T1 (de) 2004-09-15
JP4755759B2 (ja) 2011-08-24
CZ300395B6 (cs) 2009-05-06
IL144668A0 (en) 2002-05-23
PL350735A1 (en) 2003-01-27
AU3209800A (en) 2000-08-18
EE04851B1 (et) 2007-06-15

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