PL142909B1 - Method of obtaining novel derivatives of thiazolidine - Google Patents
Method of obtaining novel derivatives of thiazolidine Download PDFInfo
- Publication number
- PL142909B1 PL142909B1 PL1984252129A PL25212984A PL142909B1 PL 142909 B1 PL142909 B1 PL 142909B1 PL 1984252129 A PL1984252129 A PL 1984252129A PL 25212984 A PL25212984 A PL 25212984A PL 142909 B1 PL142909 B1 PL 142909B1
- Authority
- PL
- Poland
- Prior art keywords
- ppm
- compound
- indomethacin
- thiazolidine
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/10—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/18—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU83888A HU188852B (en) | 1983-03-16 | 1983-03-16 | Process for producing thiazolidine derivatives active against gastric ulcer and intestinal ulcer |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PL252129A1 PL252129A1 (en) | 1985-11-19 |
| PL142909B1 true PL142909B1 (en) | 1987-12-31 |
Family
ID=10951891
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL1984252129A PL142909B1 (en) | 1983-03-16 | 1984-03-13 | Method of obtaining novel derivatives of thiazolidine |
| PL1984246683A PL142749B1 (en) | 1983-03-16 | 1984-03-15 | Method of obtaining novel thiazolydine derivatives |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL1984246683A PL142749B1 (en) | 1983-03-16 | 1984-03-15 | Method of obtaining novel thiazolydine derivatives |
Country Status (32)
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6051184A (ja) * | 1983-08-30 | 1985-03-22 | Fujimoto Seiyaku Kk | Ν−シアノイミノチアゾリジン誘導体およびその製造法 |
| JPH0730070B2 (ja) * | 1985-10-03 | 1995-04-05 | 日本バイエルアグロケム株式会社 | 新規複素環式化合物 |
| JPH066585B2 (ja) * | 1985-02-04 | 1994-01-26 | 日本バイエルアグロケム株式会社 | ニトロメチレン誘導体、その製法及び殺虫剤 |
| US5204360A (en) * | 1985-02-04 | 1993-04-20 | Nihon Bayer Agrochem K.K. | Heterocyclic compounds |
| ATE67493T1 (de) * | 1985-02-04 | 1991-10-15 | Bayer Agrochem Kk | Heterocyclische verbindungen. |
| JPH0649699B2 (ja) * | 1985-02-04 | 1994-06-29 | 日本バイエルアグロケム株式会社 | ニトロメチレン誘導体、その製法及び殺虫剤 |
| US5001138B1 (en) * | 1985-02-04 | 1998-01-20 | Bayer Agrochem Kk | Heterocyclic compounds |
| USRE39130E1 (en) | 1986-03-07 | 2006-06-13 | Bayer Cropscience K.K. | Heterocyclic compounds |
| JPH0717621B2 (ja) * | 1986-03-07 | 1995-03-01 | 日本バイエルアグロケム株式会社 | 新規ヘテロ環式化合物 |
| JP2607369B2 (ja) * | 1987-02-20 | 1997-05-07 | 興和株式会社 | 新規な複素環化合物 |
| US5122522A (en) * | 1989-06-21 | 1992-06-16 | The Trustees Of The University Of Pennsylvania | Treatment and control of ocular development |
| DE69029734T2 (de) * | 1989-06-21 | 1997-05-28 | Univ Pennsylvania | Verwendung von Pirenzepine, Telenzepine oder O-Methoxy -sila-hexocyclium zur Herstellung eines Medikaments zur BEHANDLUNG UND REGULIERUNG DER AUGENENTWICKLUNG |
| HU207047B (en) * | 1989-11-07 | 1993-03-01 | Richter Gedeon Vegyeszet | Process for producing new pyridine derivatives and pharmaceutical copositions comprising same |
| US5240918A (en) * | 1992-03-24 | 1993-08-31 | Egis Gyogyszergyar | 2-(substituted imino)-thiazolidines and process for the preparation thereof |
| JP2721805B2 (ja) * | 1994-07-22 | 1998-03-04 | 日本バイエルアグロケム株式会社 | 新規ヘテロ環式化合物 |
| DE4427539A1 (de) * | 1994-08-04 | 1996-02-08 | Sueddeutsche Kalkstickstoff | Verfahren zur Herstellung von 2-Cyaniminothiazolidin |
| DE4427569A1 (de) * | 1994-08-04 | 1996-02-08 | Bayer Ag | Verfahren zur Herstellung von Cyanimino-1,3-thiazolidin |
| DE19904310A1 (de) | 1999-01-28 | 2000-08-03 | Bayer Ag | Verfahren zur Herstellung heterocyclischer Verbindungen |
| CN1198803C (zh) * | 1999-03-05 | 2005-04-27 | 第一三得利制药株式会社 | 具有激活烟碱性乙酰胆碱α4β2受体作用的杂环化合物 |
| US6667401B2 (en) * | 2000-01-19 | 2003-12-23 | Bayer Aktiengesellschaft | Method for producing heterocyclic compounds |
| JP2004531569A (ja) * | 2001-05-25 | 2004-10-14 | ヴァリー フォージ ファーマスーティカルズ、インコーポレイテッド | ピレンゼピン眼科用ゲル剤 |
| ES2315566T3 (es) * | 2002-11-22 | 2009-04-01 | Smithkline Beecham Corporation | Tiazolidin-4-onas para inhibir proteinas hyak3. |
| WO2004089927A1 (en) * | 2003-04-07 | 2004-10-21 | Cortical Pty Ltd | Novel methods for the treatment of inflammatory diseases |
| US8309733B2 (en) | 2008-07-01 | 2012-11-13 | Meji Seika Pharma Co., Ltd. | Imino derivatives, methods for producing the same and insecticides containing the same |
| DK2751100T3 (en) * | 2011-09-02 | 2016-01-18 | Bayer Ip Gmbh | METHOD FOR PREPARING [3 - [(6-CHLOR-3-PYRIDINYL) METHYL] -2-THIAZOLIDINYLIDE] CYANAMIDE |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3264316A (en) * | 1963-09-18 | 1966-08-02 | Res Lab Dr C Janssen N V | Certain 2-acylimino-3-substitutedthiazoline-4 compounds |
| DE2205745A1 (de) * | 1972-02-08 | 1973-08-23 | Thomae Gmbh Dr K | Neue durch den n-cyaniminorest substituierten heterocyclen und verfahren zu ihrer herstellung |
| US4006156A (en) * | 1975-06-27 | 1977-02-01 | Shell Oil Company | 3-Alkyl-2-(nitromethylene) thiazolidine |
| DK173777A (da) * | 1976-05-03 | 1977-11-04 | Merck & Co Inc | Fremgangsmade til fremstilling af derivater af 2-iminothiazolidiner og thiazoliner |
| JPS57171986A (en) * | 1981-04-14 | 1982-10-22 | Taiho Yakuhin Kogyo Kk | Heterocylic ring compound containing sulfur |
| JPS5823682A (ja) * | 1981-08-03 | 1983-02-12 | Santen Pharmaceut Co Ltd | 複素五員環化合物 |
| DE3133918A1 (de) * | 1981-08-27 | 1983-03-17 | Bayer Ag, 5090 Leverkusen | 2-arylhydrazino-2-thiazoline, acylderivate derselben, 2-arylazo-2-thiazoline, herstellungsverfahren und ihre verwendung zur bekaempfung von ekto- und endoparasiten |
| JPS58222886A (ja) * | 1982-06-19 | 1983-12-24 | Ricoh Co Ltd | 感熱記録シ−ト |
| JPS5933267A (ja) * | 1982-08-19 | 1984-02-23 | Fujimoto Seiyaku Kk | グアニジン誘導体およびその製造法 |
-
1983
- 1983-03-16 HU HU83888A patent/HU188852B/hu not_active IP Right Cessation
-
1984
- 1984-02-29 DK DK143284A patent/DK143284A/da not_active Application Discontinuation
- 1984-03-12 BE BE1/10980A patent/BE899132A/fr not_active IP Right Cessation
- 1984-03-12 CH CH1211/84A patent/CH660592A5/de not_active IP Right Cessation
- 1984-03-13 PL PL1984252129A patent/PL142909B1/pl unknown
- 1984-03-14 LU LU85248A patent/LU85248A1/fr unknown
- 1984-03-15 NL NL8400817A patent/NL8400817A/nl not_active Application Discontinuation
- 1984-03-15 FR FR8403985A patent/FR2542740B1/fr not_active Expired
- 1984-03-15 DD DD84260939A patent/DD216929A5/de not_active IP Right Cessation
- 1984-03-15 SE SE8401463A patent/SE455945B/sv not_active IP Right Cessation
- 1984-03-15 CS CS841885A patent/CS241074B2/cs unknown
- 1984-03-15 JP JP59048270A patent/JPS59196877A/ja active Pending
- 1984-03-15 PL PL1984246683A patent/PL142749B1/pl unknown
- 1984-03-15 IL IL71249A patent/IL71249A/xx unknown
- 1984-03-15 GR GR74119A patent/GR81883B/el unknown
- 1984-03-15 AT AT0088284A patent/AT383596B/de not_active IP Right Cessation
- 1984-03-15 PT PT78260A patent/PT78260B/pt not_active IP Right Cessation
- 1984-03-15 NO NO841002A patent/NO162858C/no unknown
- 1984-03-15 CA CA000449688A patent/CA1273933A/en not_active Expired - Lifetime
- 1984-03-15 IN IN186/CAL/84A patent/IN157738B/en unknown
- 1984-03-15 GB GB08406790A patent/GB2140412B/en not_active Expired
- 1984-03-15 ZA ZA841938A patent/ZA841938B/xx unknown
- 1984-03-15 NZ NZ207516A patent/NZ207516A/en unknown
- 1984-03-15 IE IE655/84A patent/IE57101B1/en unknown
- 1984-03-15 IT IT20057/84A patent/IT1196048B/it active
- 1984-03-16 ES ES530738A patent/ES530738A0/es active Granted
- 1984-03-16 DE DE3409801A patent/DE3409801A1/de not_active Withdrawn
- 1984-03-16 YU YU00473/84A patent/YU47384A/xx unknown
- 1984-03-16 KR KR1019840001360A patent/KR840008001A/ko not_active Ceased
- 1984-03-16 US US06/590,486 patent/US4616025A/en not_active Expired - Fee Related
- 1984-03-16 SU SU843713458A patent/SU1240355A3/ru active
- 1984-03-16 FI FI841066A patent/FI79843C/fi not_active IP Right Cessation
- 1984-03-16 AU AU25833/84A patent/AU559753B2/en not_active Ceased
- 1984-10-17 SU SU843799805A patent/SU1240356A3/ru active
-
1985
- 1985-06-17 ES ES544286A patent/ES8604179A1/es not_active Expired
Also Published As
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