NZ518094A - Process for preparing N-acylamino compounds - Google Patents

Process for preparing N-acylamino compounds

Info

Publication number
NZ518094A
NZ518094A NZ518094A NZ51809496A NZ518094A NZ 518094 A NZ518094 A NZ 518094A NZ 518094 A NZ518094 A NZ 518094A NZ 51809496 A NZ51809496 A NZ 51809496A NZ 518094 A NZ518094 A NZ 518094A
Authority
NZ
New Zealand
Prior art keywords
group
independently selected
optionally
substituted
mimosa
Prior art date
Application number
NZ518094A
Other languages
English (en)
Inventor
Mark J Batchelor
David Bebbington
Wolf Herman Fridman
Roger J Gillespie
Julian M C Golec
Yong Gu
David J Lauffer
David J Livingston
Saroop S Matharu
Michael D Mullican
Mark A Murcko
Robert Murdoch
Philip L Nyce
Andrea L C Robidoux
Michael Su
M Woods Wannamaker
Keith P Wilson
Robert E Zelle
Guy W Bemis
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27534345&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ518094(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/575,641 external-priority patent/US6008217A/en
Priority claimed from US08/598,332 external-priority patent/US5874424A/en
Priority claimed from US08/712,878 external-priority patent/US5985863A/en
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NZ518094A publication Critical patent/NZ518094A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/12—1,5-Benzodiazepines; Hydrogenated 1,5-benzodiazepines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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US08/712,878 US5985863A (en) 1996-09-12 1996-09-12 Compositions and methods for decreasing IGIF and IFN-γ production by administering an ICE inhibitor
US3149596P 1996-11-26 1996-11-26
US08/761,483 US6204261B1 (en) 1995-12-20 1996-12-06 Inhibitors of interleukin-1β Converting enzyme inhibitors

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IL124850A (en) 2006-08-20
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