IL124850A0 - Inhibitors of interleukin-1beta converting enzyme and processes for their production - Google Patents

Inhibitors of interleukin-1beta converting enzyme and processes for their production

Info

Publication number
IL124850A0
IL124850A0 IL12485096A IL12485096A IL124850A0 IL 124850 A0 IL124850 A0 IL 124850A0 IL 12485096 A IL12485096 A IL 12485096A IL 12485096 A IL12485096 A IL 12485096A IL 124850 A0 IL124850 A0 IL 124850A0
Authority
IL
Israel
Prior art keywords
interleukin
inhibitors
processes
production
converting enzyme
Prior art date
Application number
IL12485096A
Other languages
English (en)
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27534345&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL124850(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/575,641 external-priority patent/US6008217A/en
Priority claimed from US08/598,332 external-priority patent/US5874424A/en
Priority claimed from US08/712,878 external-priority patent/US5985863A/en
Application filed by Vertex Pharma filed Critical Vertex Pharma
Priority to IL14513296A priority Critical patent/IL145132A0/xx
Publication of IL124850A0 publication Critical patent/IL124850A0/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/12—1,5-Benzodiazepines; Hydrogenated 1,5-benzodiazepines
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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IL12485096A 1995-12-20 1996-12-20 Inhibitors of interleukin-1beta converting enzyme and processes for their production IL124850A0 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IL14513296A IL145132A0 (en) 1995-12-20 1996-12-20 N-acyl amio derivatives, pharmaceutical compositions containing the same and processes for their production

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US08/575,641 US6008217A (en) 1995-12-20 1995-12-20 Inhibitors of interleukin-1β converting enzyme
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US08/712,878 US5985863A (en) 1996-09-12 1996-09-12 Compositions and methods for decreasing IGIF and IFN-γ production by administering an ICE inhibitor
US3149596P 1996-11-26 1996-11-26
US08/761,483 US6204261B1 (en) 1995-12-20 1996-12-06 Inhibitors of interleukin-1β Converting enzyme inhibitors
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US20030225269A1 (en) 2003-12-04
TR200201217T2 (tr) 2002-12-23
JP2003137896A (ja) 2003-05-14
CZ190698A3 (cs) 1998-10-14
BRPI9612258B1 (xx) 2011-05-31
NO982597L (no) 1998-08-12
AU735075B2 (en) 2001-06-28
SK84298A3 (en) 1999-03-12
US20080039449A1 (en) 2008-02-14
US7790713B2 (en) 2010-09-07
JP2002507961A (ja) 2002-03-12
GEP20022638B (en) 2002-02-25
KR20040096550A (ko) 2004-11-16
WO1997022619A3 (en) 1997-10-16
CZ300171B6 (cs) 2009-03-04
EP0869967A2 (en) 1998-10-14
US8119631B2 (en) 2012-02-21
AP0202539A0 (en) 1998-06-20
US6423840B1 (en) 2002-07-23
NZ518094A (en) 2004-01-30
KR100561504B1 (ko) 2006-03-20
NO982597D0 (no) 1998-06-05
NZ326610A (en) 2000-08-25
CZ298171B6 (cs) 2007-07-11
IS4771A (is) 1998-06-12
AP0202538A0 (en) 1998-06-20
US20050143436A1 (en) 2005-06-30
TR200201216T2 (tr) 2002-09-23
JP4205762B2 (ja) 2009-01-07
EP2083014A3 (en) 2010-01-06
PL190736B1 (pl) 2005-12-30
BG64465B1 (bg) 2005-03-31
AU1522297A (en) 1997-07-14
CA2239904C (en) 2010-01-19
BR9612258A (pt) 1999-07-13
CN1229412A (zh) 1999-09-22
EP2295442A2 (en) 2011-03-16
US6258948B1 (en) 2001-07-10
BRPI9612258B8 (pt) 2018-04-17
UA66337C2 (uk) 2004-04-15
EP2295442A3 (en) 2011-04-06
HK1089435A1 (en) 2006-12-01
IL124850A (en) 2006-08-20

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