NO984082D0 - Pyrimido£5,4-d|pyrimidiner, medikamenter inneholdende disse forbindelser, deres anvendelse og fremgangsmÕte for fremstilling derav - Google Patents

Pyrimido£5,4-d|pyrimidiner, medikamenter inneholdende disse forbindelser, deres anvendelse og fremgangsmÕte for fremstilling derav

Info

Publication number
NO984082D0
NO984082D0 NO984082A NO984082A NO984082D0 NO 984082 D0 NO984082 D0 NO 984082D0 NO 984082 A NO984082 A NO 984082A NO 984082 A NO984082 A NO 984082A NO 984082 D0 NO984082 D0 NO 984082D0
Authority
NO
Norway
Prior art keywords
pyrimido
pyrimidines
compounds
preparation
drugs containing
Prior art date
Application number
NO984082A
Other languages
English (en)
Other versions
NO984082L (no
NO311522B1 (no
Inventor
Frank Himmelsbach
Georg Dahmann
Den Thomas Von R
Thomas Metz
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of NO984082L publication Critical patent/NO984082L/no
Publication of NO984082D0 publication Critical patent/NO984082D0/no
Publication of NO311522B1 publication Critical patent/NO311522B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO19984082A 1996-03-06 1998-09-04 Pyrimido[5,4-d]pyrimidiner, legemiddel inneholdende disse forbindelser, deres anvendelse og fremgangsmåte for fremstillingderav NO311522B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19608588A DE19608588A1 (de) 1996-03-06 1996-03-06 Pyrimido [5,4-d]pyrimidine, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
PCT/EP1997/001047 WO1997032880A1 (de) 1996-03-06 1997-03-03 PYRIMIDO[5,4-d]PYRIMIDINE, DIESE VERBINDUNGEN ENTHALTENDE ARZNEIMITTEL, DEREN VERWENDUNG UND VERFAHREN ZU IHRER HERSTELLUNG

Publications (3)

Publication Number Publication Date
NO984082L NO984082L (no) 1998-09-04
NO984082D0 true NO984082D0 (no) 1998-09-04
NO311522B1 NO311522B1 (no) 2001-12-03

Family

ID=7787345

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19984082A NO311522B1 (no) 1996-03-06 1998-09-04 Pyrimido[5,4-d]pyrimidiner, legemiddel inneholdende disse forbindelser, deres anvendelse og fremgangsmåte for fremstillingderav

Country Status (30)

Country Link
US (1) US5821240A (no)
EP (1) EP0888351B1 (no)
JP (1) JP2000506151A (no)
KR (1) KR19990087504A (no)
CN (1) CN1064362C (no)
AR (1) AR006108A1 (no)
AT (1) ATE252101T1 (no)
AU (1) AU730376B2 (no)
BG (1) BG63163B1 (no)
BR (1) BR9707839A (no)
CA (1) CA2248720A1 (no)
CO (1) CO4650043A1 (no)
CZ (1) CZ281598A3 (no)
DE (2) DE19608588A1 (no)
EE (1) EE9800278A (no)
HK (1) HK1018450A1 (no)
HU (1) HUP9902049A3 (no)
IL (1) IL125342A0 (no)
MX (1) MX9807073A (no)
NO (1) NO311522B1 (no)
NZ (1) NZ331545A (no)
PL (1) PL328719A1 (no)
RU (1) RU2195461C2 (no)
SK (1) SK120898A3 (no)
TR (1) TR199801755T2 (no)
TW (1) TW454008B (no)
UA (1) UA54421C2 (no)
UY (1) UY24474A1 (no)
WO (1) WO1997032880A1 (no)
ZA (1) ZA971887B (no)

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US6028183A (en) 1997-11-07 2000-02-22 Gilead Sciences, Inc. Pyrimidine derivatives and oligonucleotides containing same
JP3270834B2 (ja) * 1999-01-27 2002-04-02 ファイザー・プロダクツ・インク 抗がん剤として有用なヘテロ芳香族二環式誘導体
UA72946C2 (uk) 1999-11-05 2005-05-16 Астразенека Аб Похідні хіназоліну як інгібітори васкулярного ендотеліального фактора росту (vegf)
EP1170011A1 (en) * 2000-07-06 2002-01-09 Boehringer Ingelheim International GmbH Novel use of inhibitors of the epidermal growth factor receptor
DE10115921A1 (de) 2001-03-30 2002-10-02 Boehringer Ingelheim Pharma Verfahren zur Herstellung von 4,6-Diaminopyrimido[5,4-d]pyrimidinen
EP1300146A1 (en) * 2001-10-03 2003-04-09 Boehringer Ingelheim International GmbH Pharmaceutical composition for the treatment of animal mammary tumors
EP1460061A4 (en) * 2001-12-27 2006-05-31 Toray Finechemicals Co Ltd PROCESS FOR PRODUCING 1-ALCOXYCARBONYL SATURATED NITROGENIC HETEROCYCLIC DERIVATIVE
US20070179161A1 (en) * 2003-03-31 2007-08-02 Vernalis (Cambridge) Limited. Pyrazolopyrimidine compounds and their use in medicine
EA013904B1 (ru) * 2003-12-18 2010-08-30 Янссен Фармацевтика Н.В. Пиридо- и пиримидопиримидиновые производные в качестве антипролиферативных агентов
JO3088B1 (ar) * 2004-12-08 2017-03-15 Janssen Pharmaceutica Nv مشتقات كوينازولين كبيرة الحلقات و استعمالها بصفتها موانع كينيز متعددة الاهداف
NI200700147A (es) 2004-12-08 2019-05-10 Janssen Pharmaceutica Nv Derivados de quinazolina inhibidores de cinasas dirigidos a multip
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EP2044084B1 (en) 2006-07-13 2016-02-17 Janssen Pharmaceutica NV Mtki quinazoline derivatives
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Family Cites Families (3)

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DE3049207A1 (de) * 1980-12-27 1982-07-29 Dr. Karl Thomae Gmbh, 7950 Biberach Neue trisubstituierte pyrimido (5,4-d) pyrimidine, ihre herstellung und ihre verwendung als arzneimittel
TW414798B (en) * 1994-09-07 2000-12-11 Thomae Gmbh Dr K Pyrimido (5,4-d) pyrimidines, medicaments comprising these compounds, their use and processes for their preparation
DE4431867A1 (de) * 1994-09-07 1996-03-14 Thomae Gmbh Dr K Pyrimido[5,4-d]pyrimidine, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
PL328719A1 (en) 1999-02-15
AR006108A1 (es) 1999-08-11
BG102789A (en) 1999-09-30
NO984082L (no) 1998-09-04
CN1212694A (zh) 1999-03-31
HUP9902049A2 (hu) 1999-10-28
JP2000506151A (ja) 2000-05-23
CO4650043A1 (es) 1998-09-03
US5821240A (en) 1998-10-13
EE9800278A (et) 1999-02-15
BR9707839A (pt) 1999-07-27
MX9807073A (es) 1998-12-31
EP0888351A1 (de) 1999-01-07
TW454008B (en) 2001-09-11
HUP9902049A3 (en) 2000-03-28
TR199801755T2 (xx) 1998-12-21
AU730376B2 (en) 2001-03-08
KR19990087504A (ko) 1999-12-27
CZ281598A3 (cs) 1999-02-17
HK1018450A1 (en) 1999-12-24
WO1997032880A1 (de) 1997-09-12
ATE252101T1 (de) 2003-11-15
CA2248720A1 (en) 1997-09-12
NO311522B1 (no) 2001-12-03
UY24474A1 (es) 2000-09-29
AU2094597A (en) 1997-09-22
UA54421C2 (uk) 2003-03-17
DE59710864D1 (de) 2003-11-20
CN1064362C (zh) 2001-04-11
EP0888351B1 (de) 2003-10-15
BG63163B1 (bg) 2001-05-31
IL125342A0 (en) 1999-03-12
SK120898A3 (en) 1999-02-11
DE19608588A1 (de) 1997-09-11
RU2195461C2 (ru) 2002-12-27
NZ331545A (en) 2000-03-27
ZA971887B (en) 1998-09-07

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