HK1018450A1 - Pyrimido [5,4-d] [pyrimidines, medicaments containing these compounds, their use and process for their production - Google Patents

Pyrimido [5,4-d] [pyrimidines, medicaments containing these compounds, their use and process for their production

Info

Publication number
HK1018450A1
HK1018450A1 HK99103458A HK99103458A HK1018450A1 HK 1018450 A1 HK1018450 A1 HK 1018450A1 HK 99103458 A HK99103458 A HK 99103458A HK 99103458 A HK99103458 A HK 99103458A HK 1018450 A1 HK1018450 A1 HK 1018450A1
Authority
HK
Hong Kong
Prior art keywords
pyrimido
pyrimidines
compounds
production
medicaments containing
Prior art date
Application number
HK99103458A
Other languages
English (en)
Inventor
Frank Himmelsbach
Georg Dahmann
Ruden Thomas Von
Thomas Metz
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of HK1018450A1 publication Critical patent/HK1018450A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HK99103458A 1996-03-06 1999-08-10 Pyrimido [5,4-d] [pyrimidines, medicaments containing these compounds, their use and process for their production HK1018450A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19608588A DE19608588A1 (de) 1996-03-06 1996-03-06 Pyrimido [5,4-d]pyrimidine, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
PCT/EP1997/001047 WO1997032880A1 (de) 1996-03-06 1997-03-03 PYRIMIDO[5,4-d]PYRIMIDINE, DIESE VERBINDUNGEN ENTHALTENDE ARZNEIMITTEL, DEREN VERWENDUNG UND VERFAHREN ZU IHRER HERSTELLUNG

Publications (1)

Publication Number Publication Date
HK1018450A1 true HK1018450A1 (en) 1999-12-24

Family

ID=7787345

Family Applications (1)

Application Number Title Priority Date Filing Date
HK99103458A HK1018450A1 (en) 1996-03-06 1999-08-10 Pyrimido [5,4-d] [pyrimidines, medicaments containing these compounds, their use and process for their production

Country Status (30)

Country Link
US (1) US5821240A (xx)
EP (1) EP0888351B1 (xx)
JP (1) JP2000506151A (xx)
KR (1) KR19990087504A (xx)
CN (1) CN1064362C (xx)
AR (1) AR006108A1 (xx)
AT (1) ATE252101T1 (xx)
AU (1) AU730376B2 (xx)
BG (1) BG63163B1 (xx)
BR (1) BR9707839A (xx)
CA (1) CA2248720A1 (xx)
CO (1) CO4650043A1 (xx)
CZ (1) CZ281598A3 (xx)
DE (2) DE19608588A1 (xx)
EE (1) EE9800278A (xx)
HK (1) HK1018450A1 (xx)
HU (1) HUP9902049A3 (xx)
IL (1) IL125342A0 (xx)
MX (1) MX9807073A (xx)
NO (1) NO311522B1 (xx)
NZ (1) NZ331545A (xx)
PL (1) PL328719A1 (xx)
RU (1) RU2195461C2 (xx)
SK (1) SK120898A3 (xx)
TR (1) TR199801755T2 (xx)
TW (1) TW454008B (xx)
UA (1) UA54421C2 (xx)
UY (1) UY24474A1 (xx)
WO (1) WO1997032880A1 (xx)
ZA (1) ZA971887B (xx)

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KR19990082463A (ko) 1996-02-13 1999-11-25 돈 리사 로얄 혈관 내피 성장 인자 억제제로서의 퀴나졸린유도체
CN1116286C (zh) 1996-03-05 2003-07-30 曾尼卡有限公司 4－苯胺基喹唑啉衍生物
US6028183A (en) 1997-11-07 2000-02-22 Gilead Sciences, Inc. Pyrimidine derivatives and oligonucleotides containing same
JP3270834B2 (ja) * 1999-01-27 2002-04-02 ファイザー・プロダクツ・インク 抗がん剤として有用なヘテロ芳香族二環式誘導体
PT1244647E (pt) 1999-11-05 2006-10-31 Astrazeneca Ab Derivados de quinazolina como inibidores de vegf
EP1170011A1 (en) * 2000-07-06 2002-01-09 Boehringer Ingelheim International GmbH Novel use of inhibitors of the epidermal growth factor receptor
DE10115921A1 (de) * 2001-03-30 2002-10-02 Boehringer Ingelheim Pharma Verfahren zur Herstellung von 4,6-Diaminopyrimido[5,4-d]pyrimidinen
EP1300146A1 (en) * 2001-10-03 2003-04-09 Boehringer Ingelheim International GmbH Pharmaceutical composition for the treatment of animal mammary tumors
WO2003055858A1 (fr) * 2001-12-27 2003-07-10 Toray Fine Chemicals Co., Ltd. Processus de production de derive heterocyclique sature azote 1-alcoxycarbonyle
EP1608652A1 (en) * 2003-03-31 2005-12-28 Vernalis (Cambridge) Limited Pyrazolopyrimidine compounds and their use in medicine
CA2549869C (en) * 2003-12-18 2015-05-05 Janssen Pharmaceutica N.V. Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents
JO3088B1 (ar) * 2004-12-08 2017-03-15 Janssen Pharmaceutica Nv مشتقات كوينازولين كبيرة الحلقات و استعمالها بصفتها موانع كينيز متعددة الاهداف
NI200700147A (es) 2004-12-08 2019-05-10 Janssen Pharmaceutica Nv Derivados de quinazolina inhibidores de cinasas dirigidos a multip
KR101139038B1 (ko) 2005-06-28 2012-05-02 삼성전자주식회사 피리미도피리미딘 유도체 및 이를 이용한 유기 박막 트랜지스터
AU2007274284B2 (en) 2006-07-13 2012-04-26 Janssen Pharmaceutica N.V. Mtki quinazoline derivatives
DK2170827T3 (da) * 2007-06-21 2013-11-18 Janssen Pharmaceutica Nv Indolin-2-oner og aza-indolin-2-oner
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Family Cites Families (3)

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Publication number Priority date Publication date Assignee Title
DE3049207A1 (de) * 1980-12-27 1982-07-29 Dr. Karl Thomae Gmbh, 7950 Biberach Neue trisubstituierte pyrimido (5,4-d) pyrimidine, ihre herstellung und ihre verwendung als arzneimittel
TW414798B (en) * 1994-09-07 2000-12-11 Thomae Gmbh Dr K Pyrimido (5,4-d) pyrimidines, medicaments comprising these compounds, their use and processes for their preparation
DE4431867A1 (de) * 1994-09-07 1996-03-14 Thomae Gmbh Dr K Pyrimido[5,4-d]pyrimidine, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
NO311522B1 (no) 2001-12-03
CZ281598A3 (cs) 1999-02-17
TW454008B (en) 2001-09-11
DE59710864D1 (de) 2003-11-20
UA54421C2 (uk) 2003-03-17
EP0888351A1 (de) 1999-01-07
JP2000506151A (ja) 2000-05-23
NZ331545A (en) 2000-03-27
CO4650043A1 (es) 1998-09-03
MX9807073A (es) 1998-12-31
NO984082D0 (no) 1998-09-04
AU2094597A (en) 1997-09-22
RU2195461C2 (ru) 2002-12-27
BR9707839A (pt) 1999-07-27
HUP9902049A3 (en) 2000-03-28
HUP9902049A2 (hu) 1999-10-28
ATE252101T1 (de) 2003-11-15
AR006108A1 (es) 1999-08-11
KR19990087504A (ko) 1999-12-27
EP0888351B1 (de) 2003-10-15
CN1064362C (zh) 2001-04-11
SK120898A3 (en) 1999-02-11
CA2248720A1 (en) 1997-09-12
NO984082L (no) 1998-09-04
ZA971887B (en) 1998-09-07
UY24474A1 (es) 2000-09-29
BG63163B1 (bg) 2001-05-31
EE9800278A (et) 1999-02-15
TR199801755T2 (xx) 1998-12-21
CN1212694A (zh) 1999-03-31
PL328719A1 (en) 1999-02-15
AU730376B2 (en) 2001-03-08
WO1997032880A1 (de) 1997-09-12
BG102789A (en) 1999-09-30
US5821240A (en) 1998-10-13
DE19608588A1 (de) 1997-09-11
IL125342A0 (en) 1999-03-12

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