NO327740B1 - Farmasoytisk sammensetning og anvendelse av farmasoytiske effektive mengder av en forbindelse som har anti-Xa-aktivitet og en plateaggregeringsantagonistforbindelse. - Google Patents
Farmasoytisk sammensetning og anvendelse av farmasoytiske effektive mengder av en forbindelse som har anti-Xa-aktivitet og en plateaggregeringsantagonistforbindelse. Download PDFInfo
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- NO327740B1 NO327740B1 NO19992555A NO992555A NO327740B1 NO 327740 B1 NO327740 B1 NO 327740B1 NO 19992555 A NO19992555 A NO 19992555A NO 992555 A NO992555 A NO 992555A NO 327740 B1 NO327740 B1 NO 327740B1
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- Prior art keywords
- platelet aggregation
- compound
- antagonist compound
- enoxaparin
- activity
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Hematology (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3187896P | 1996-11-27 | 1996-11-27 | |
| PCT/US1997/021440 WO1998023279A1 (en) | 1996-11-27 | 1997-11-24 | PHARMACEUTICAL COMPOSITION COMPRISING A COMPOUND HAVING ANTI-Xa ACTIVITY AND A PLATELET AGGREGATION ANTAGONIST COMPOUND |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO992555L NO992555L (no) | 1999-05-27 |
| NO992555D0 NO992555D0 (no) | 1999-05-27 |
| NO327740B1 true NO327740B1 (no) | 2009-09-14 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19992555A NO327740B1 (no) | 1996-11-27 | 1999-05-27 | Farmasoytisk sammensetning og anvendelse av farmasoytiske effektive mengder av en forbindelse som har anti-Xa-aktivitet og en plateaggregeringsantagonistforbindelse. |
Country Status (27)
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|---|---|
| US (2) | US6103705A (https=) |
| EP (1) | EP0946185B2 (https=) |
| JP (1) | JP4498471B2 (https=) |
| KR (1) | KR100512671B1 (https=) |
| CN (1) | CN1121224C (https=) |
| AP (1) | AP1390A (https=) |
| AT (1) | ATE283062T1 (https=) |
| AU (1) | AU754936B2 (https=) |
| BG (1) | BG64542B1 (https=) |
| BR (1) | BR9713141A (https=) |
| CA (1) | CA2272317C (https=) |
| CZ (1) | CZ298552B6 (https=) |
| DE (1) | DE69731763T3 (https=) |
| DK (1) | DK0946185T4 (https=) |
| EA (1) | EA002475B1 (https=) |
| ES (1) | ES2230624T5 (https=) |
| HU (1) | HUP9903496A3 (https=) |
| IL (1) | IL129877A (https=) |
| NO (1) | NO327740B1 (https=) |
| OA (1) | OA11049A (https=) |
| PL (1) | PL189116B1 (https=) |
| PT (1) | PT946185E (https=) |
| SI (1) | SI0946185T2 (https=) |
| SK (1) | SK286024B6 (https=) |
| UA (1) | UA63929C2 (https=) |
| WO (1) | WO1998023279A1 (https=) |
| ZA (1) | ZA9710691B (https=) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA63929C2 (uk) * | 1996-11-27 | 2004-02-16 | Aventis Pharm Prod Inc | Фармацевтична композиція та продукт, що містить сполуки з анти-ха активністю і антагоніст агрегації тромбоцитів, спосіб і набір для лікування або профілактики захворювань, які супроводжують тромбоутворення |
| FR2764511B1 (fr) | 1997-06-13 | 2000-09-08 | Sanofi Sa | Compositions pour le traitement et la prevention de la thrombose arterielle et utilisation d'un inhibiteur du facteur xa seul et/ou en combinaison avec un antiagregant plaquettaire |
| US6136794A (en) * | 1998-02-02 | 2000-10-24 | Merck & Co., Inc. | Platelet aggregation inhibition using low molecular weight heparin in combination with a GP IIb/IIIa antagonist |
| WO2000029019A1 (en) * | 1998-11-18 | 2000-05-25 | G.D. Searle & Co. | Restoration of platelet aggregation by antibody administration after gpiib/iiia antagonist treatment |
| CA2377734A1 (en) * | 1999-06-30 | 2001-01-11 | Hamilton Civic Hospitals Research Development, Inc. | Heparin compositions that inhibit clot associated coagulation factors |
| ES2161615B1 (es) * | 1999-07-23 | 2003-03-16 | Rovi Lab Farmaceut Sa | Composiciones de heparinas de muy bajo peso molecular. |
| US6969705B2 (en) * | 2000-07-21 | 2005-11-29 | Aventis Pharma S.A. | Compositions of polysaccharides derived from heparin, their preparation and pharmaceutical compositions containing them |
| CA2420890A1 (en) * | 2000-09-08 | 2002-03-14 | Hamilton Civic Hospitals Research Development, Inc. | Antithrombotic compositions |
| US6982251B2 (en) * | 2000-12-20 | 2006-01-03 | Schering Corporation | Substituted 2-azetidinones useful as hypocholesterolemic agents |
| AR035533A1 (es) | 2001-01-26 | 2004-06-02 | Schering Corp | Uso de por lo menos un inhibidor de la absorcion de los esteroles o sus sales, solvatos, prodrogas farmaceuticamente aceptables o mezclas de los mismos para la preparacion de un medicamento para el tratamiento de la sitosterolemia, composiciones farmaceuticas, el uso de dichas composiciones para la |
| US7071181B2 (en) | 2001-01-26 | 2006-07-04 | Schering Corporation | Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors |
| IL156445A0 (en) | 2001-01-26 | 2004-01-04 | Schering Corp | Combinations of peroxisome proliferator-activated receptor (ppar) activator(s) and sterol absorption inhibitor(s) and treatments for vascular indications |
| DE10141106A1 (de) * | 2001-08-22 | 2003-03-13 | Aventis Pharma Gmbh | Verwendung von Heparinoid-Derivaten zur Behandlung und Diagnose von mit Heparinoiden behandelbaren Erkrankungen |
| US7053080B2 (en) | 2001-09-21 | 2006-05-30 | Schering Corporation | Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors |
| MXPA04002573A (es) | 2001-09-21 | 2004-06-18 | Schering Corp | Tratamiento de xantoma con derivados de azetidinona como inhibidores de la absorcion de esterol. |
| US20040171819A1 (en) * | 2002-10-10 | 2004-09-02 | Aventis Pharma S.A. | Mixtures of polysaccharides derived from heparin, their preparation and pharmaceutical compositions containing them |
| WO2004043457A1 (en) | 2002-11-06 | 2004-05-27 | Schering Corporation | Cholesterol absorptions inhibitors for the treatment of autoimmune disorders |
| EP1601668B1 (en) | 2003-03-07 | 2008-08-27 | Schering Corporation | Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia |
| JP2006519869A (ja) | 2003-03-07 | 2006-08-31 | シェーリング コーポレイション | 置換アゼチジノン化合物、置換アゼチジノン化合物を調製するためのプロセス、それらの処方物および使用 |
| US7459442B2 (en) | 2003-03-07 | 2008-12-02 | Schering Corporation | Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof |
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1997
- 1997-11-24 UA UA99063586A patent/UA63929C2/uk unknown
- 1997-11-24 JP JP52478398A patent/JP4498471B2/ja not_active Expired - Fee Related
- 1997-11-24 DE DE69731763T patent/DE69731763T3/de not_active Expired - Lifetime
- 1997-11-24 ES ES97948482T patent/ES2230624T5/es not_active Expired - Lifetime
- 1997-11-24 AP APAP/P/1999/001517A patent/AP1390A/en active
- 1997-11-24 IL IL12987797A patent/IL129877A/en not_active IP Right Cessation
- 1997-11-24 PT PT97948482T patent/PT946185E/pt unknown
- 1997-11-24 BR BR9713141-5A patent/BR9713141A/pt not_active Application Discontinuation
- 1997-11-24 SK SK673-99A patent/SK286024B6/sk not_active IP Right Cessation
- 1997-11-24 KR KR10-1999-7004656A patent/KR100512671B1/ko not_active Expired - Fee Related
- 1997-11-24 CN CN97180019A patent/CN1121224C/zh not_active Expired - Fee Related
- 1997-11-24 AU AU54546/98A patent/AU754936B2/en not_active Ceased
- 1997-11-24 CZ CZ0174299A patent/CZ298552B6/cs not_active IP Right Cessation
- 1997-11-24 SI SI9730691T patent/SI0946185T2/sl unknown
- 1997-11-24 WO PCT/US1997/021440 patent/WO1998023279A1/en not_active Ceased
- 1997-11-24 EA EA199900499A patent/EA002475B1/ru not_active IP Right Cessation
- 1997-11-24 AT AT97948482T patent/ATE283062T1/de active
- 1997-11-24 CA CA002272317A patent/CA2272317C/en not_active Expired - Fee Related
- 1997-11-24 PL PL97333665A patent/PL189116B1/pl not_active IP Right Cessation
- 1997-11-24 EP EP97948482A patent/EP0946185B2/en not_active Expired - Lifetime
- 1997-11-24 HU HU9903496A patent/HUP9903496A3/hu unknown
- 1997-11-24 DK DK97948482.1T patent/DK0946185T4/da active
- 1997-11-27 ZA ZA9710691A patent/ZA9710691B/xx unknown
-
1998
- 1998-11-16 US US09/192,710 patent/US6103705A/en not_active Expired - Lifetime
-
1999
- 1999-04-29 BG BG103372A patent/BG64542B1/bg unknown
- 1999-05-19 OA OA9900105A patent/OA11049A/en unknown
- 1999-05-27 NO NO19992555A patent/NO327740B1/no not_active IP Right Cessation
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2000
- 2000-03-01 US US09/516,981 patent/US20020032214A1/en not_active Abandoned
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