NO304408B1 - Farmas°ytisk sammensetning med antagonistisk virkning for oral anvendelse - Google Patents
Farmas°ytisk sammensetning med antagonistisk virkning for oral anvendelse Download PDFInfo
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- NO304408B1 NO304408B1 NO924417A NO924417A NO304408B1 NO 304408 B1 NO304408 B1 NO 304408B1 NO 924417 A NO924417 A NO 924417A NO 924417 A NO924417 A NO 924417A NO 304408 B1 NO304408 B1 NO 304408B1
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Cardiology (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cosmetics (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Investigating Or Analysing Biological Materials (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP30492491 | 1991-11-20 |
Publications (3)
Publication Number | Publication Date |
---|---|
NO924417D0 NO924417D0 (no) | 1992-11-16 |
NO924417L NO924417L (no) | 1993-05-21 |
NO304408B1 true NO304408B1 (no) | 1998-12-14 |
Family
ID=17938952
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO924417A NO304408B1 (no) | 1991-11-20 | 1992-11-16 | Farmas°ytisk sammensetning med antagonistisk virkning for oral anvendelse |
Country Status (18)
Country | Link |
---|---|
US (1) | US5534534A (ja) |
EP (3) | EP0782852B1 (ja) |
KR (1) | KR100256633B1 (ja) |
CN (1) | CN1047518C (ja) |
AT (2) | ATE157248T1 (ja) |
AU (1) | AU659691B2 (ja) |
BR (1) | BR1100336A (ja) |
CA (1) | CA2083305C (ja) |
DE (2) | DE69233424T2 (ja) |
DK (1) | DK0546358T3 (ja) |
ES (1) | ES2104797T3 (ja) |
FI (2) | FI111604B (ja) |
GR (1) | GR3025338T3 (ja) |
HU (1) | HU211608A9 (ja) |
MX (1) | MX9206634A (ja) |
NO (1) | NO304408B1 (ja) |
NZ (1) | NZ245175A (ja) |
TW (1) | TW284688B (ja) |
Families Citing this family (51)
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TW284688B (ja) * | 1991-11-20 | 1996-09-01 | Takeda Pharm Industry Co Ltd | |
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AU679616B2 (en) * | 1994-04-19 | 1997-07-03 | Tanabe Seiyaku Co., Ltd. | Imidazopyridine derivatives and process for preparing the same |
US5753672A (en) * | 1994-04-19 | 1998-05-19 | Tanabe Seiyaku Co., Ltd. | Imidazopyridine derivatives and process for preparing the same |
TW418204B (en) * | 1997-03-28 | 2001-01-11 | Dev Center Biotechnology | Novel 1,2,4-triazine-5-ketonyl benzene derivatives and the analogs, the preparation, and the pharmaceutical compositions as angiotension II receptor antogonists |
US6297239B1 (en) | 1997-10-08 | 2001-10-02 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
AU2745199A (en) * | 1998-03-04 | 1999-09-20 | Takeda Chemical Industries Ltd. | Sustained-release preparation for aii antagonist, production and use thereof |
US7115644B2 (en) * | 2002-09-13 | 2006-10-03 | Boehringer Ingelheim Pharmaceuticals Inc. | Heterocyclic compounds |
US20050031683A1 (en) * | 2003-08-04 | 2005-02-10 | Ashish Kapoor | Solid pharmaceutical composition |
PT1685126E (pt) * | 2003-10-16 | 2007-04-30 | Teva Pharma | Preparação de candesartan cilexetil |
US20050175689A1 (en) * | 2003-10-27 | 2005-08-11 | Yamanouchi Pharmaceutical Co., Ltd. | Coated fine particles containing drug for intrabuccally fast disintegrating tablet |
WO2005070398A2 (en) * | 2004-01-23 | 2005-08-04 | Ranbaxy Laboratories Limited | Pharmaceutical compositions of candesartan cilexetil stabilized with co-solvents |
WO2005079751A2 (en) * | 2004-01-23 | 2005-09-01 | Ranbaxy Laboratories Limited | Oral pharmaceutical compositions of candesartan cilexetil |
EP1713795A2 (en) * | 2004-02-11 | 2006-10-25 | Teva Pharmaceutical Industries Ltd. | Candesartan cilexetil polymorphs |
US20070298108A1 (en) | 2004-03-01 | 2007-12-27 | Peter Svete | Pharmaceutical Formulation |
CZ23088U1 (cs) * | 2004-03-25 | 2011-12-19 | Astellas Pharma Inc. | Kompozice pevného farmaceutického prípravku solifenacinu nebo jeho soli |
CN1953973A (zh) * | 2004-05-05 | 2007-04-25 | 特瓦制药工业有限公司 | 高纯度坎地沙坦酯的制备 |
US7588779B2 (en) * | 2004-05-28 | 2009-09-15 | Andrx Labs, Llc | Pharmaceutical formulation containing a biguanide and an angiotensin antagonist |
AU2005320672B2 (en) * | 2004-12-27 | 2011-01-06 | Astellas Pharma Inc. | Stable particulate pharmaceutical composition of solifenacin or salt thereof |
KR20070118224A (ko) * | 2005-01-06 | 2007-12-14 | 엘란 파마 인터내셔널 리미티드 | 나노입자형 칸데사르탄 제제 |
JP2007527925A (ja) * | 2005-01-14 | 2007-10-04 | テバ ファーマシューティカル インダストリーズ リミティド | 粗カンデサルタンシレキセチルの調製 |
PL1843754T3 (pl) * | 2005-01-26 | 2011-12-30 | Lek Pharmaceuticals | Nowa kompozycja farmaceutyczna zawierająca cyleksetyl kandesartanu jako lipofilową substancję krystaliczną |
CA2599415C (en) * | 2005-05-10 | 2011-07-19 | Teva Pharmaceutical Industries Ltd. | Stable micronized candesartan cilexetil and methods for preparing thereof |
US7815939B2 (en) * | 2005-07-20 | 2010-10-19 | Astellas Pharma Inc. | Coated fine particles containing drug for intrabuccally fast disintegrating dosage forms |
TW200800299A (en) * | 2006-04-27 | 2008-01-01 | Takeda Pharmaceutical | Pharmaceutical composition |
CN102813635A (zh) * | 2006-08-10 | 2012-12-12 | 武田药品工业株式会社 | 药物组合物 |
WO2008045006A1 (en) * | 2006-10-11 | 2008-04-17 | Fako Ilaclari A. S. | Formulations of candesartan |
ES2301401B1 (es) * | 2006-11-28 | 2009-06-08 | Laboratorios Liconsa S.A. | Composicion farmaceutica solida estabilizada de candesartan cilexetilo. |
EP1952806A1 (en) | 2007-02-01 | 2008-08-06 | Helm AG | Process for the preparation of adsorbates of candesartan |
ATE479427T1 (de) * | 2007-03-08 | 2010-09-15 | Teva Pharma | Pharmazeutische zusammensetzung mit candesartan- cilexetil |
US9066936B2 (en) * | 2007-03-28 | 2015-06-30 | Takeda Pharmaceutical Company Limited | Solid pharmaceutical composition comprising a benzimidazole-7-carboxylate derivative and a pH control agent |
MX2009011493A (es) | 2007-04-25 | 2009-11-09 | Teva Pharma | Complejo de excipiente farmaceutico. |
WO2008149338A2 (en) * | 2007-06-06 | 2008-12-11 | Dexcel Ltd. | Process for forming solid oral dosage forms of angiotensin ii receptor antagonists |
DE102007052070A1 (de) | 2007-10-30 | 2009-05-07 | Tiefenbacher Pharmachemikalien Alfred E. Tiefenbacher Gmbh & Co. Kg | Candesartancilexetil |
EP2165702B1 (en) | 2008-09-17 | 2011-11-16 | Helm AG | Stable and readily dissolved compositions of candesartan cilexetil prepared with wet granulation |
US9387249B2 (en) | 2008-12-23 | 2016-07-12 | Takeda Pharmaceutical Company Limited | Methods of treating hypertension with at least one angiotensin II receptor blocker and chlorthalidone |
ES2364011B1 (es) | 2009-11-20 | 2013-01-24 | Gp Pharm, S.A. | Cápsulas de principios activos farmacéuticos y ésteres de ácidos grasos poliinsaturados para el tratamiento de enfermedades cardiovasculares. |
EP2624696B1 (en) | 2010-10-06 | 2016-12-21 | Glaxosmithkline LLC | Benzimidazole derivatives as pi3 kinase inhibitors |
CN102138920A (zh) * | 2011-02-24 | 2011-08-03 | 海南中济医药科技有限公司 | 一种含有坎地沙坦酯和氢氯噻嗪的药物组合物及其制备方法 |
CN102357095A (zh) * | 2011-07-12 | 2012-02-22 | 迪沙药业集团有限公司 | 稳定的药物组合物 |
WO2013068875A1 (en) | 2011-11-11 | 2013-05-16 | Pfizer Inc. | 2-thiopyrimidinones |
EP2928468A4 (en) * | 2012-12-05 | 2016-07-27 | Sawai Seiyaku Kk | PREPARATION CONTAINING CANDÉSARTAN CILEXÉTIL |
PL236001B1 (pl) | 2012-12-21 | 2020-11-30 | Adamed Spolka Z Ograniczona Odpowiedzialnoscia | Złożona kompozycja farmaceutyczna zawierająca kandesartan cyleksetylu oraz amlodypinę, sposób jej wytwarzania oraz jednostkowa postać dawkowania zawierająca tę kompozycję |
ES2768651T3 (es) | 2013-04-25 | 2020-06-23 | Kyorin Seiyaku Kk | Composición farmacéutica sólida |
WO2014199315A1 (en) * | 2013-06-11 | 2014-12-18 | Universidade Federal De Minas Gerais - Ufmg | Process for preparing amphiphilic peptide derivatives |
FI3263110T3 (fi) | 2015-02-26 | 2023-07-25 | Takeda Pharmaceuticals Co | Tabletti, joka käsittää metoksiureajohdannaista ja mannitolipartikkeleita |
CR20170498A (es) | 2015-05-05 | 2018-01-26 | Pfizer | 2-tiopirimidinonas |
KR102684436B1 (ko) | 2015-10-16 | 2024-07-15 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | Ep4 길항제 |
CN111617046A (zh) * | 2020-07-09 | 2020-09-04 | 浙江诺得药业有限公司 | 阿齐沙坦分散片及其制备工艺 |
CN112957336A (zh) * | 2021-03-03 | 2021-06-15 | 广州白云山天心制药股份有限公司 | 一种稳定的坎地沙坦酯药物固体组合物及其制备方法 |
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TW284688B (ja) * | 1991-11-20 | 1996-09-01 | Takeda Pharm Industry Co Ltd |
-
1992
- 1992-11-09 TW TW081108934A patent/TW284688B/zh not_active IP Right Cessation
- 1992-11-13 AU AU28391/92A patent/AU659691B2/en not_active Expired
- 1992-11-16 NO NO924417A patent/NO304408B1/no not_active IP Right Cessation
- 1992-11-18 MX MX9206634A patent/MX9206634A/es unknown
- 1992-11-18 US US07/978,290 patent/US5534534A/en not_active Expired - Lifetime
- 1992-11-18 NZ NZ24517592A patent/NZ245175A/en not_active IP Right Cessation
- 1992-11-19 AT AT92119705T patent/ATE157248T1/de active
- 1992-11-19 EP EP96118520A patent/EP0782852B1/en not_active Expired - Lifetime
- 1992-11-19 DK DK92119705.9T patent/DK0546358T3/da active
- 1992-11-19 ES ES92119705T patent/ES2104797T3/es not_active Expired - Lifetime
- 1992-11-19 EP EP04013762A patent/EP1468683A3/en not_active Withdrawn
- 1992-11-19 CA CA002083305A patent/CA2083305C/en not_active Expired - Lifetime
- 1992-11-19 FI FI925270A patent/FI111604B/fi not_active IP Right Cessation
- 1992-11-19 AT AT96118520T patent/ATE277602T1/de active
- 1992-11-19 CN CN92113172A patent/CN1047518C/zh not_active Expired - Lifetime
- 1992-11-19 DE DE69233424T patent/DE69233424T2/de not_active Expired - Lifetime
- 1992-11-19 EP EP92119705A patent/EP0546358B1/en not_active Expired - Lifetime
- 1992-11-19 DE DE69221831T patent/DE69221831T2/de not_active Expired - Lifetime
- 1992-11-20 KR KR1019920021902A patent/KR100256633B1/ko not_active IP Right Cessation
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1995
- 1995-06-29 HU HU95P/P00534P patent/HU211608A9/hu unknown
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1997
- 1997-04-23 BR BR1100336-7A patent/BR1100336A/pt active IP Right Grant
- 1997-11-11 GR GR970402980T patent/GR3025338T3/el unknown
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2003
- 2003-02-12 FI FI20030210A patent/FI20030210A/fi unknown
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