NO2011011I1 - Silodosin (Indolinforbindelse representert ved strukturformelen vist i krav 1 i norsk patent 329855) - Google Patents

Silodosin (Indolinforbindelse representert ved strukturformelen vist i krav 1 i norsk patent 329855)

Info

Publication number
NO2011011I1
NO2011011I1 NO2011011C NO2011011C NO2011011I1 NO 2011011 I1 NO2011011 I1 NO 2011011I1 NO 2011011 C NO2011011 C NO 2011011C NO 2011011 C NO2011011 C NO 2011011C NO 2011011 I1 NO2011011 I1 NO 2011011I1
Authority
NO
Norway
Prior art keywords
silodosin
compound represented
structural formula
formula shown
indoline compound
Prior art date
Application number
NO2011011C
Other languages
English (en)
Other versions
NO2011011I2 (no
Original Assignee
Kissei Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31973150&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO2011011(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kissei Pharmaceutical filed Critical Kissei Pharmaceutical
Publication of NO2011011I1 publication Critical patent/NO2011011I1/no
Publication of NO2011011I2 publication Critical patent/NO2011011I2/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO2011011C 2002-09-06 2011-07-11 Silodosin (Indolinforbindelse representert ved strukturformelen vist i krav 1 i norsk patent 329855) NO2011011I1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002262157 2002-09-06
PCT/JP2003/011345 WO2004022538A1 (ja) 2002-09-06 2003-09-05 経口用固形医薬用結晶およびそれを含む排尿障害治療用経口用固形医薬

Publications (2)

Publication Number Publication Date
NO2011011I1 true NO2011011I1 (no) 2011-07-25
NO2011011I2 NO2011011I2 (no) 2012-10-01

Family

ID=31973150

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20051709A NO329855B1 (no) 2002-09-06 2005-04-06 Kystallforbindelse for fast oralt medikament samt fast oralt medikament omfattende denne til behandling av dysuria
NO2011011C NO2011011I1 (no) 2002-09-06 2011-07-11 Silodosin (Indolinforbindelse representert ved strukturformelen vist i krav 1 i norsk patent 329855)

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO20051709A NO329855B1 (no) 2002-09-06 2005-04-06 Kystallforbindelse for fast oralt medikament samt fast oralt medikament omfattende denne til behandling av dysuria

Country Status (24)

Country Link
US (1) US20060142374A1 (no)
EP (1) EP1541554B1 (no)
JP (1) JP4532274B2 (no)
KR (1) KR100670592B1 (no)
CN (1) CN1321111C (no)
AT (1) ATE416159T1 (no)
AU (1) AU2003264385B2 (no)
BR (1) BR0314338A (no)
CA (1) CA2496780C (no)
DE (1) DE60325074D1 (no)
ES (1) ES2316858T3 (no)
HK (1) HK1084396A1 (no)
HR (1) HRP20050214B1 (no)
IL (1) IL167168A (no)
IS (1) IS2640B (no)
MX (1) MXPA05002549A (no)
NO (2) NO329855B1 (no)
NZ (1) NZ538598A (no)
PL (1) PL375701A1 (no)
RU (1) RU2347774C2 (no)
TW (1) TW200407126A (no)
UA (1) UA78854C2 (no)
WO (1) WO2004022538A1 (no)
ZA (1) ZA200501884B (no)

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KR101072909B1 (ko) * 2002-12-16 2011-10-17 깃세이 야쿠힌 고교 가부시키가이샤 경구고형의약
US20070167511A1 (en) * 2004-03-05 2007-07-19 Kissei Pharmaceutical Co,. Ltd. Medicinal composition for prevention or treatment of overactive bladder accompanying nervous disorder
CN101027052A (zh) * 2004-10-05 2007-08-29 橘生药品工业株式会社 用于伴下尿路梗阻的集尿障碍的预防和/或治疗剂
ES2378240T3 (es) * 2004-10-06 2012-04-10 Kissei Pharmaceutical Co., Ltd. Composición medicinal para evitar la transición al tratamiento operatorio de la hipertrofia prostática
NZ556156A (en) * 2005-02-02 2010-03-26 Teva Pharma Process for producing acetate salts of polypeptides using hydrogenolysis
PT1848415E (pt) * 2005-02-17 2013-06-27 Teva Pharma Terapia de combinação com acetato de glatirâmero e rasagilina para o tratamento da esclerose múltipla
ES2375761T3 (es) * 2006-12-14 2012-03-06 Teva Pharmaceutical Industries Ltd. Base de rasagilina cristalina sólida.
US20100076010A1 (en) * 2007-02-26 2010-03-25 Concert Pharmaceuticals, Inc. Alpha 1a-adrenoceptor antagonists
US8013007B2 (en) * 2007-02-26 2011-09-06 Concert Pharmaceuticals, Inc. Alpha 1A-adrenoceptor antagonists
MX2009009230A (es) * 2007-02-28 2009-11-26 Kissei Pharmaceutical Uso de silodosina en una administracion diaria para tratar hiperplasia prostatica benigna.
JP2011525489A (ja) * 2008-06-19 2011-09-22 テバ ファーマシューティカル インダストリーズ リミティド ラサリジン塩基の精製方法
ES2471076T3 (es) 2010-06-28 2014-06-25 Ratiopharm Gmbh Compuestos de inclusión de silodoxina-ciclodextrina
JP2013532651A (ja) 2010-07-23 2013-08-19 ラティオファルム ゲー・エム・ベー・ハー シロドシンと塩基性コポリマーとの混合物を含む経口投与用医薬品
WO2012014186A1 (en) 2010-07-30 2012-02-02 Ranbaxy Laboratories Limited Process for the preparation of silodosin and its novel intermediates
CN102229557B (zh) * 2010-08-05 2013-03-27 南京海纳医药科技有限公司 西洛多辛的半水合物晶体、制备方法和包含它的药物组合物
CN102229558B (zh) * 2010-08-05 2013-05-08 南京海纳医药科技有限公司 西洛多辛的晶型δ、它的制备方法和包含它的药物组合物
CN102010359B (zh) * 2010-09-10 2013-01-23 北京阳光诺和药物研究有限公司 β晶型西洛多辛的制备方法
WO2012077138A1 (en) 2010-12-09 2012-06-14 Panacea Biotec Limited Methods of crystallizing (r) -1- (3 -hydroxypropyl) -5- [2- [2- [2- ( 2, 2, 2 - trifluoroethoxy) phenoxy] ethylamino] propyl] indoline-7 -carboxamide
SI2474529T1 (sl) 2010-12-23 2014-12-31 Sandoz Ag Kristalne oblike aktivne farmacevtske učinkovine
CN102283816B (zh) * 2011-08-05 2013-09-11 北京海步国际医药科技发展有限公司 西洛多辛缓释片剂及其制备方法
WO2013061338A1 (en) * 2011-08-24 2013-05-02 Cadila Healthcare Limited Pharmaceutical compositions of silodosin
WO2013072935A2 (en) 2011-10-10 2013-05-23 Cadila Healthcare Limited Process for the preparation of silodosin
TWI659752B (zh) * 2013-03-26 2019-05-21 日商橘生藥品工業股份有限公司 經遮蔽西羅多辛（Ｓｉｌｏｄｏｓｉｎ）苦味之經口投與製劑
CN103159664B (zh) * 2013-03-29 2016-03-23 深圳市海滨制药有限公司 一种赛洛多辛原料药及其制备方法、药物组合物
WO2015015512A2 (en) * 2013-07-29 2015-02-05 Ind-Swift Laboratories Limited Process for the preparation of silodosin and its gamma form
JP2015117192A (ja) * 2013-12-17 2015-06-25 東和薬品株式会社 シロドシンγ型結晶及びその製造方法
JP6225998B2 (ja) 2014-02-06 2017-11-08 宇部興産株式会社 インドリン化合物の製造方法
KR20150127996A (ko) * 2014-05-08 2015-11-18 한미정밀화학주식회사 실로도신 감마형 결정의 제조방법
KR101725393B1 (ko) * 2014-07-24 2017-04-27 주식회사 경보제약 실로도신의 제조 방법 및 신규 중간체
KR101673160B1 (ko) 2014-10-24 2016-11-07 보령제약 주식회사 실로도신 γ 결정형의 제조방법
JP2016147811A (ja) * 2015-02-10 2016-08-18 ダイト株式会社 シロドシンγ型結晶の製造方法
ES2607639B1 (es) 2015-09-30 2018-02-28 Urquima, S.A Sal de ácido maleico de un intermedio de silodosina
KR101733084B1 (ko) 2016-07-27 2017-05-08 (주)다산메디켐 실로도신의 결정형의 제조방법
EP3354283B1 (en) 2017-06-20 2019-08-07 Alfred E. Tiefenbacher (GmbH & Co. KG) Pharmaceutical capsule composition comprising silodosin
JP2018035199A (ja) * 2017-12-07 2018-03-08 東和薬品株式会社 シロドシンγ型結晶及びその製造方法
CN107903201B (zh) * 2017-12-27 2020-09-25 浙江天宇药业股份有限公司 一种β晶型西洛多辛的制备方法
CN111410626B (zh) * 2019-01-04 2022-11-04 上海汇伦医药股份有限公司 赛洛多辛α-晶型的制备方法
CN109824569B (zh) * 2019-04-04 2022-09-20 重庆医药高等专科学校 一种西罗多辛晶型i及其制备方法
WO2020237643A1 (zh) * 2019-05-31 2020-12-03 上海汇伦生命科技有限公司 赛洛多辛α-晶型的制备方法
CN114601826B (zh) * 2022-03-31 2024-06-04 乐泰药业有限公司 一种用于治疗前列腺增生的药物制剂及其制备方法和质量检测方法

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EP0600675B1 (en) * 1992-12-02 1998-07-08 Kissei Pharmaceutical Co., Ltd. Indoline compounds for the treatment of dysuria
JP3331048B2 (ja) * 1994-06-01 2002-10-07 キッセイ薬品工業株式会社 インドール誘導体
WO1999015202A1 (fr) * 1997-09-22 1999-04-01 Kissei Pharmaceutical Co., Ltd. Medicaments contre la dysurie resultant d'une hypertrophie de la prostate
WO1999048530A1 (en) * 1998-03-23 1999-09-30 Merck & Co., Inc. Combination therapy for the treatment of benign prostatic hyperplasia
JP4324266B2 (ja) * 1999-02-26 2009-09-02 キッセイ薬品工業株式会社 α１Ａアドレナリン受容体の変異体、当該変異体を用いた測定方法及び前立腺肥大に伴う排尿困難症治療剤
JP4921646B2 (ja) * 2001-03-08 2012-04-25 キッセイ薬品工業株式会社 １−（３−ベンジルオキシプロピル）−５−（２−置換プロピル）インドリン誘導体およびその使用方法
ES2362788T3 (es) * 2004-10-27 2011-07-13 Kissei Pharmaceutical Co., Ltd. Compuesto de indolina y proceso para la producción del mismo.

Also Published As

Publication number Publication date
UA78854C2 (en) 2007-04-25
JPWO2004022538A1 (ja) 2005-12-22
TW200407126A (en) 2004-05-16
CA2496780C (en) 2011-03-15
NZ538598A (en) 2007-08-31
HK1084396A1 (en) 2006-07-28
IS7785A (is) 2005-04-05
CN1321111C (zh) 2007-06-13
US20060142374A1 (en) 2006-06-29
TWI305148B (no) 2009-01-11
HRP20050214A2 (en) 2006-05-31
MXPA05002549A (es) 2005-06-03
AU2003264385A1 (en) 2004-03-29
PL375701A1 (en) 2005-12-12
CN1694867A (zh) 2005-11-09
NO329855B1 (no) 2011-01-10
CA2496780A1 (en) 2004-03-18
WO2004022538A1 (ja) 2004-03-18
NO20051709L (no) 2005-06-06
JP4532274B2 (ja) 2010-08-25
HRP20050214B1 (hr) 2013-09-30
IS2640B (is) 2010-06-15
IL167168A (en) 2010-11-30
ATE416159T1 (de) 2008-12-15
BR0314338A (pt) 2005-07-05
RU2005109930A (ru) 2006-01-20
KR20050057181A (ko) 2005-06-16
AU2003264385B2 (en) 2009-12-17
DE60325074D1 (de) 2009-01-15
NO2011011I2 (no) 2012-10-01
RU2347774C2 (ru) 2009-02-27
ZA200501884B (en) 2006-05-31
EP1541554A1 (en) 2005-06-15
EP1541554A4 (en) 2006-11-08
KR100670592B1 (ko) 2007-01-17
EP1541554B1 (en) 2008-12-03
ES2316858T3 (es) 2009-04-16

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