IS2640B - Kristall fyrir lyf á föstu formi til inntöku og lyf á föstu formi til inntöku sem inniheldur kristalinn til að meðhöndla þvaglátstregðu. - Google Patents
Kristall fyrir lyf á föstu formi til inntöku og lyf á föstu formi til inntöku sem inniheldur kristalinn til að meðhöndla þvaglátstregðu.Info
- Publication number
- IS2640B IS2640B IS7785A IS7785A IS2640B IS 2640 B IS2640 B IS 2640B IS 7785 A IS7785 A IS 7785A IS 7785 A IS7785 A IS 7785A IS 2640 B IS2640 B IS 2640B
- Authority
- IS
- Iceland
- Prior art keywords
- oral
- solid
- crystals
- crystal
- treatment
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Urology & Nephrology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Indole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2002262157 | 2002-09-06 | ||
PCT/JP2003/011345 WO2004022538A1 (ja) | 2002-09-06 | 2003-09-05 | 経口用固形医薬用結晶およびそれを含む排尿障害治療用経口用固形医薬 |
Publications (2)
Publication Number | Publication Date |
---|---|
IS7785A IS7785A (is) | 2005-04-05 |
IS2640B true IS2640B (is) | 2010-06-15 |
Family
ID=31973150
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IS7785A IS2640B (is) | 2002-09-06 | 2005-04-05 | Kristall fyrir lyf á föstu formi til inntöku og lyf á föstu formi til inntöku sem inniheldur kristalinn til að meðhöndla þvaglátstregðu. |
Country Status (24)
Country | Link |
---|---|
US (1) | US20060142374A1 (is) |
EP (1) | EP1541554B1 (is) |
JP (1) | JP4532274B2 (is) |
KR (1) | KR100670592B1 (is) |
CN (1) | CN1321111C (is) |
AT (1) | ATE416159T1 (is) |
AU (1) | AU2003264385B2 (is) |
BR (1) | BR0314338A (is) |
CA (1) | CA2496780C (is) |
DE (1) | DE60325074D1 (is) |
ES (1) | ES2316858T3 (is) |
HK (1) | HK1084396A1 (is) |
HR (1) | HRP20050214B1 (is) |
IL (1) | IL167168A (is) |
IS (1) | IS2640B (is) |
MX (1) | MXPA05002549A (is) |
NO (2) | NO329855B1 (is) |
NZ (1) | NZ538598A (is) |
PL (1) | PL375701A1 (is) |
RU (1) | RU2347774C2 (is) |
TW (1) | TW200407126A (is) |
UA (1) | UA78854C2 (is) |
WO (1) | WO2004022538A1 (is) |
ZA (1) | ZA200501884B (is) |
Families Citing this family (40)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2402010A1 (en) * | 2002-12-16 | 2012-01-04 | Kissei Pharmaceutical Co., Ltd. | Solid drug for oral use |
ES2436608T3 (es) * | 2004-03-05 | 2014-01-03 | Kissei Pharmaceutical Co., Ltd. | Composición medicinal para la prevención o el tratamiento de la vejiga hiperactiva asociada a un trastorno nervioso |
KR100965205B1 (ko) * | 2004-10-05 | 2010-06-24 | 깃세이 야쿠힌 고교 가부시키가이샤 | 하부요로 폐색 질환에 따른 축뇨장해의 예방 및/또는치료제 |
PL1806136T3 (pl) * | 2004-10-06 | 2012-04-30 | Kissei Pharmaceutical | Kompozycja medyczna do zapobiegania przejściu na leczenie operacyjne łagodnego rozrostu gruczołu krokowego |
RU2419638C2 (ru) * | 2005-02-02 | 2011-05-27 | Тева Фармасьютикал Индастриз, Лтд. | Способ получения полипептидных смесей с использованием гидрогенолиза |
CA2596664A1 (en) * | 2005-02-17 | 2006-08-24 | Teva Pharmaceutical Industries Ltd. | Combination therapy with glatiramer acetate and rasagiline for the treatment of multiple sclerosis |
EA016820B1 (ru) * | 2006-12-14 | 2012-07-30 | Тева Фармасьютикал Индастриз, Лтд. | Кристаллическое твердое основание разагилина |
US20100076010A1 (en) * | 2007-02-26 | 2010-03-25 | Concert Pharmaceuticals, Inc. | Alpha 1a-adrenoceptor antagonists |
WO2008106125A2 (en) * | 2007-02-26 | 2008-09-04 | Concert Pharmaceuticals, Inc. | Deuterated derivatives of silodosin as alpha la-adrenoceptor antagonists |
US20080242717A1 (en) * | 2007-02-28 | 2008-10-02 | Fumiyasu Sato | Methods for treating benign prostatic hyperplasia |
JP2011525489A (ja) * | 2008-06-19 | 2011-09-22 | テバ ファーマシューティカル インダストリーズ リミティド | ラサリジン塩基の精製方法 |
ES2471076T3 (es) | 2010-06-28 | 2014-06-25 | Ratiopharm Gmbh | Compuestos de inclusión de silodoxina-ciclodextrina |
EP2595607A2 (de) | 2010-07-23 | 2013-05-29 | Ratiopharm GmbH | Arzneimittel zur oralen verabreichung umfassend ein gemisch aus silodosin und einem basischen copolymer |
WO2012014186A1 (en) | 2010-07-30 | 2012-02-02 | Ranbaxy Laboratories Limited | Process for the preparation of silodosin and its novel intermediates |
CN102229558B (zh) * | 2010-08-05 | 2013-05-08 | 南京海纳医药科技有限公司 | 西洛多辛的晶型δ、它的制备方法和包含它的药物组合物 |
CN102229557B (zh) * | 2010-08-05 | 2013-03-27 | 南京海纳医药科技有限公司 | 西洛多辛的半水合物晶体、制备方法和包含它的药物组合物 |
CN102010359B (zh) * | 2010-09-10 | 2013-01-23 | 北京阳光诺和药物研究有限公司 | β晶型西洛多辛的制备方法 |
WO2012077138A1 (en) | 2010-12-09 | 2012-06-14 | Panacea Biotec Limited | Methods of crystallizing (r) -1- (3 -hydroxypropyl) -5- [2- [2- [2- ( 2, 2, 2 - trifluoroethoxy) phenoxy] ethylamino] propyl] indoline-7 -carboxamide |
SI2474529T1 (sl) * | 2010-12-23 | 2014-12-31 | Sandoz Ag | Kristalne oblike aktivne farmacevtske učinkovine |
CN102283816B (zh) * | 2011-08-05 | 2013-09-11 | 北京海步国际医药科技发展有限公司 | 西洛多辛缓释片剂及其制备方法 |
WO2013061338A1 (en) * | 2011-08-24 | 2013-05-02 | Cadila Healthcare Limited | Pharmaceutical compositions of silodosin |
WO2013072935A2 (en) | 2011-10-10 | 2013-05-23 | Cadila Healthcare Limited | Process for the preparation of silodosin |
US20160045446A1 (en) * | 2013-03-26 | 2016-02-18 | Kissei Pharmaceutical Co., Ltd. | Oral administration preparation with masked bitterness of silodosin |
CN103159664B (zh) * | 2013-03-29 | 2016-03-23 | 深圳市海滨制药有限公司 | 一种赛洛多辛原料药及其制备方法、药物组合物 |
WO2015015512A2 (en) * | 2013-07-29 | 2015-02-05 | Ind-Swift Laboratories Limited | Process for the preparation of silodosin and its gamma form |
JP2015117192A (ja) * | 2013-12-17 | 2015-06-25 | 東和薬品株式会社 | シロドシンγ型結晶及びその製造方法 |
CN105960394B (zh) | 2014-02-06 | 2019-03-15 | 宇部兴产株式会社 | 二氢吲哚化合物的制造方法 |
KR20150127996A (ko) * | 2014-05-08 | 2015-11-18 | 한미정밀화학주식회사 | 실로도신 감마형 결정의 제조방법 |
KR101725393B1 (ko) * | 2014-07-24 | 2017-04-27 | 주식회사 경보제약 | 실로도신의 제조 방법 및 신규 중간체 |
KR101673160B1 (ko) | 2014-10-24 | 2016-11-07 | 보령제약 주식회사 | 실로도신 γ 결정형의 제조방법 |
JP2016147811A (ja) * | 2015-02-10 | 2016-08-18 | ダイト株式会社 | シロドシンγ型結晶の製造方法 |
ES2607639B1 (es) | 2015-09-30 | 2018-02-28 | Urquima, S.A | Sal de ácido maleico de un intermedio de silodosina |
KR101733084B1 (ko) | 2016-07-27 | 2017-05-08 | (주)다산메디켐 | 실로도신의 결정형의 제조방법 |
EP3354283B1 (en) | 2017-06-20 | 2019-08-07 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Pharmaceutical capsule composition comprising silodosin |
JP2018035199A (ja) * | 2017-12-07 | 2018-03-08 | 東和薬品株式会社 | シロドシンγ型結晶及びその製造方法 |
CN107903201B (zh) * | 2017-12-27 | 2020-09-25 | 浙江天宇药业股份有限公司 | 一种β晶型西洛多辛的制备方法 |
CN111410626B (zh) * | 2019-01-04 | 2022-11-04 | 上海汇伦医药股份有限公司 | 赛洛多辛α-晶型的制备方法 |
CN109824569B (zh) * | 2019-04-04 | 2022-09-20 | 重庆医药高等专科学校 | 一种西罗多辛晶型i及其制备方法 |
WO2020237643A1 (zh) * | 2019-05-31 | 2020-12-03 | 上海汇伦生命科技有限公司 | 赛洛多辛α-晶型的制备方法 |
CN114601826B (zh) * | 2022-03-31 | 2024-06-04 | 乐泰药业有限公司 | 一种用于治疗前列腺增生的药物制剂及其制备方法和质量检测方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69319551T2 (de) * | 1992-12-02 | 1998-10-29 | Kissei Pharmaceutical | Indolin Verbindungen zur Behandlung von Dysurien |
JP3331048B2 (ja) * | 1994-06-01 | 2002-10-07 | キッセイ薬品工業株式会社 | インドール誘導体 |
WO1999015202A1 (fr) * | 1997-09-22 | 1999-04-01 | Kissei Pharmaceutical Co., Ltd. | Medicaments contre la dysurie resultant d'une hypertrophie de la prostate |
WO1999048530A1 (en) * | 1998-03-23 | 1999-09-30 | Merck & Co., Inc. | Combination therapy for the treatment of benign prostatic hyperplasia |
JP4324266B2 (ja) * | 1999-02-26 | 2009-09-02 | キッセイ薬品工業株式会社 | α1Aアドレナリン受容体の変異体、当該変異体を用いた測定方法及び前立腺肥大に伴う排尿困難症治療剤 |
JP4921646B2 (ja) * | 2001-03-08 | 2012-04-25 | キッセイ薬品工業株式会社 | 1−(3−ベンジルオキシプロピル)−5−(2−置換プロピル)インドリン誘導体およびその使用方法 |
MX2007005126A (es) * | 2004-10-27 | 2007-07-04 | Kissei Pharmaceutical | Compuesto de indolina y proceso para producir el mismo. |
-
2003
- 2003-05-09 UA UAA200503153A patent/UA78854C2/uk unknown
- 2003-09-05 CN CNB038247968A patent/CN1321111C/zh not_active Expired - Lifetime
- 2003-09-05 RU RU2005109930/04A patent/RU2347774C2/ru active
- 2003-09-05 AT AT03794249T patent/ATE416159T1/de not_active IP Right Cessation
- 2003-09-05 DE DE60325074T patent/DE60325074D1/de not_active Expired - Lifetime
- 2003-09-05 KR KR1020057003768A patent/KR100670592B1/ko active IP Right Grant
- 2003-09-05 JP JP2004534170A patent/JP4532274B2/ja not_active Expired - Lifetime
- 2003-09-05 US US10/526,898 patent/US20060142374A1/en not_active Abandoned
- 2003-09-05 WO PCT/JP2003/011345 patent/WO2004022538A1/ja active Application Filing
- 2003-09-05 PL PL03375701A patent/PL375701A1/xx not_active Application Discontinuation
- 2003-09-05 NZ NZ538598A patent/NZ538598A/en not_active IP Right Cessation
- 2003-09-05 AU AU2003264385A patent/AU2003264385B2/en active Active
- 2003-09-05 EP EP03794249A patent/EP1541554B1/en not_active Expired - Lifetime
- 2003-09-05 MX MXPA05002549A patent/MXPA05002549A/es active IP Right Grant
- 2003-09-05 ES ES03794249T patent/ES2316858T3/es not_active Expired - Lifetime
- 2003-09-05 BR BR0314338-4A patent/BR0314338A/pt not_active Application Discontinuation
- 2003-09-05 CA CA2496780A patent/CA2496780C/en not_active Expired - Lifetime
- 2003-09-05 TW TW092124775A patent/TW200407126A/zh not_active IP Right Cessation
-
2005
- 2005-03-01 IL IL167168A patent/IL167168A/en unknown
- 2005-03-04 HR HRP20050214AA patent/HRP20050214B1/hr not_active IP Right Cessation
- 2005-03-04 ZA ZA2005/01884A patent/ZA200501884B/en unknown
- 2005-04-05 IS IS7785A patent/IS2640B/is unknown
- 2005-04-06 NO NO20051709A patent/NO329855B1/no not_active IP Right Cessation
-
2006
- 2006-04-20 HK HK06104721A patent/HK1084396A1/xx not_active IP Right Cessation
-
2011
- 2011-07-11 NO NO2011011C patent/NO2011011I1/no not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IS2640B (is) | Kristall fyrir lyf á föstu formi til inntöku og lyf á föstu formi til inntöku sem inniheldur kristalinn til að meðhöndla þvaglátstregðu. | |
EP1400529A4 (en) | GLUCOPYRANOSYLOXYPYRAZOLE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL AND INTERMEDIARY USE THEREOF | |
HK1050369A1 (en) | Glucopyranosyloxypyrazole derivatives, medicinal compositions containing the same and intermediates in the production thereof. | |
WO2005044192A3 (en) | Triazole compounds and uses related thereto | |
AU2003225617A1 (en) | Thiadiazolylpiperazine derivatives useful for treating or preventing pain | |
NO20082445L (no) | Neuropeptid-2 reseptor-agonister | |
MXPA04012998A (es) | Modulares de receptores nucleares de hormonas esteroideas triciclicos. | |
NO20052182L (no) | Nye forbindelser | |
NO20052699L (no) | 4(fenylpiperazinyl-metyl)benzamid-derivater og deres anvendelse ved behandling av smerte og gastrointestinale lidelser. | |
EP1491187A4 (en) | PREVENTIVE OR THERAPEUTIC AGENT FOR RENAL DISEASES | |
WO2004041802A8 (en) | 4(phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain or gastrointestinal disorders | |
NO20044531L (no) | Imidazolinylmetyl-aralkylsulfonamider, blandinger omfattende slike, fremgangsmate for fremstilling av slike, slike forbindelser som medikament samt anvendelse av slike forbindelser for fremstilling av medikamenter for behandling av sykdom | |
GB0212410D0 (en) | Organic compounds | |
SE0201837D0 (sv) | Chemical compounds | |
DE60013560D1 (de) | Malto-oligosaccharid-derivate und ihre anwendungen | |
NO20013601L (no) | Nye morfolinobenzamidsalter | |
NO20045353L (no) | Orto-substituerte benzosyrederivater for behandling av insulinresistens | |
NO20045223L (no) | Orto-substituerte benzosyrederivater for behandling av insulinresistens | |
DE60106246D1 (de) | Malto-oligosaccharide und deren verwendung | |
GEP20084343B (en) | Use of indole derivatives for the treatment of neuropathic pain | |
SE0103272D0 (sv) | Chemical compounds | |
MXPA05013732A (es) | Proceso para preparacion de sensibilizador de insulina y compuesto intermediario del mismo. | |
EP1238971A4 (en) | SUBSTITUTED GUANIDINE DERIVATIVES | |
TH53156A3 (th) | สารประกอบเฮทเทอโรไซคลิกและการใช้สารประกอบเฮทเทอโร-ไซคลิกในการรักษาโรค | |
TH53868A3 (th) | สารประกอบอะซาโพลีไซคลิกที่ถูกเชื่อมประสานของอะรีล |