NO20100078L - (2S,3R)-N-(2-((3-pyridinyl)metyl)-1-azabicyklo[2.2.2]oct-3-yl)benzofuran-2-karboksamid, nye saltformer og deres anvendelse - Google Patents

(2S,3R)-N-(2-((3-pyridinyl)metyl)-1-azabicyklo[2.2.2]oct-3-yl)benzofuran-2-karboksamid, nye saltformer og deres anvendelse

Info

Publication number
NO20100078L
NO20100078L NO20100078A NO20100078A NO20100078L NO 20100078 L NO20100078 L NO 20100078L NO 20100078 A NO20100078 A NO 20100078A NO 20100078 A NO20100078 A NO 20100078A NO 20100078 L NO20100078 L NO 20100078L
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NO
Norway
Prior art keywords
azabicyclo
benzofuran
pyridinyl
carboxamide
oct
Prior art date
Application number
NO20100078A
Other languages
English (en)
Norwegian (no)
Inventor
Gary Maurice Dull
Anatoly A Mazurov
Gregory J Gatto
Julio A Munoz
John Genus
Lan Miao
Merouane Bencherif
Lisa Benson
Nikolai Fedorov
Kristen G Jordan
Jacob Mathew
Inigo Pfeiffer
Sondra Pfeiffer
Teresa Y Phillips
Original Assignee
Targacept Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39945177&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20100078(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Targacept Inc filed Critical Targacept Inc
Publication of NO20100078L publication Critical patent/NO20100078L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • A—HUMAN NECESSITIES
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

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  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20100078A 2007-08-02 2010-01-18 (2S,3R)-N-(2-((3-pyridinyl)metyl)-1-azabicyklo[2.2.2]oct-3-yl)benzofuran-2-karboksamid, nye saltformer og deres anvendelse NO20100078L (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US95361407P 2007-08-02 2007-08-02
US95361307P 2007-08-02 2007-08-02
US95361007P 2007-08-02 2007-08-02
US97165407P 2007-09-12 2007-09-12
PCT/US2008/071872 WO2009018505A1 (en) 2007-08-02 2008-08-01 (2s,3r)-n-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofuran-2-carboxamide, novel salt forms, and methods of use thereof

Publications (1)

Publication Number Publication Date
NO20100078L true NO20100078L (no) 2010-02-26

Family

ID=39945177

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20100078A NO20100078L (no) 2007-08-02 2010-01-18 (2S,3R)-N-(2-((3-pyridinyl)metyl)-1-azabicyklo[2.2.2]oct-3-yl)benzofuran-2-karboksamid, nye saltformer og deres anvendelse
NO20100077A NO20100077L (no) 2007-08-02 2010-01-18 Behandling med alfa7-selektive ligander

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NO20100077A NO20100077L (no) 2007-08-02 2010-01-18 Behandling med alfa7-selektive ligander

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