NL8400099A - Gesubstitueerde carboxy-thiazolo3,2-apyrimidinederivaten, werkwijze ter bereiding daarvan en farmaceutische samenstellingen, die deze derivaten bevatten. - Google Patents

Gesubstitueerde carboxy-thiazolo3,2-apyrimidinederivaten, werkwijze ter bereiding daarvan en farmaceutische samenstellingen, die deze derivaten bevatten. Download PDF

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Publication number
NL8400099A
NL8400099A NL8400099A NL8400099A NL8400099A NL 8400099 A NL8400099 A NL 8400099A NL 8400099 A NL8400099 A NL 8400099A NL 8400099 A NL8400099 A NL 8400099A NL 8400099 A NL8400099 A NL 8400099A
Authority
NL
Netherlands
Prior art keywords
oxo
trans
thiazolo
carboxylic acid
pyrimidine
Prior art date
Application number
NL8400099A
Other languages
English (en)
Dutch (nl)
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NL8400099A publication Critical patent/NL8400099A/nl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NL8400099A 1983-01-12 1984-01-11 Gesubstitueerde carboxy-thiazolo3,2-apyrimidinederivaten, werkwijze ter bereiding daarvan en farmaceutische samenstellingen, die deze derivaten bevatten. NL8400099A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8300728 1983-01-12
GB838300728A GB8300728D0 (en) 1983-01-12 1983-01-12 Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives

Publications (1)

Publication Number Publication Date
NL8400099A true NL8400099A (nl) 1984-08-01

Family

ID=10536219

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8400099A NL8400099A (nl) 1983-01-12 1984-01-11 Gesubstitueerde carboxy-thiazolo3,2-apyrimidinederivaten, werkwijze ter bereiding daarvan en farmaceutische samenstellingen, die deze derivaten bevatten.

Country Status (27)

Country Link
US (2) US4558046A (pt)
JP (1) JPS59130891A (pt)
KR (1) KR840007420A (pt)
AT (1) AT386601B (pt)
AU (1) AU568527B2 (pt)
BE (1) BE898641A (pt)
CA (1) CA1232604A (pt)
CH (1) CH660011A5 (pt)
CS (1) CS27984A2 (pt)
DE (1) DE3400733A1 (pt)
DK (1) DK12084A (pt)
ES (1) ES528662A0 (pt)
FI (1) FI77869C (pt)
FR (1) FR2539131B1 (pt)
GB (1) GB8300728D0 (pt)
GR (1) GR81735B (pt)
HU (1) HU190945B (pt)
IL (1) IL70651A (pt)
IT (1) IT1185050B (pt)
NL (1) NL8400099A (pt)
NO (1) NO840092L (pt)
NZ (1) NZ206816A (pt)
PH (1) PH22448A (pt)
PT (1) PT77946B (pt)
SE (1) SE456996B (pt)
SU (1) SU1355131A3 (pt)
ZA (1) ZA84227B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4921854A (en) * 1986-12-30 1990-05-01 Egis Gyogyszergyar Condensed thiazolopyrimidine, pyrimido-thiazine or thiazepine pyrimidine compounds
US6121300A (en) * 1998-11-10 2000-09-19 Wagle; Dilip R. Reversing advanced glycosylation cross-links using heterocyclic-substituted thiazolium salts
NZ595781A (en) * 2008-01-11 2013-07-26 Glenmark Pharmaceuticals Sa Fused pyrimidine derivatives as trpv3 modulators
US8119647B2 (en) * 2008-04-23 2012-02-21 Glenmark Pharmaceuticals S.A. Fused pyrimidineone compounds as TRPV3 modulators

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3594378A (en) * 1969-10-24 1971-07-20 Ayerst Mckenna & Harrison Thiazolopyrimidine derivatives and preparation thereof
US3888983A (en) * 1970-08-14 1975-06-10 Seperic Derivatives of thiazolino-pyrimidin-6-ones, in inducing analgesia
GB1334628A (en) * 1972-02-02 1973-10-24 Seperic Thiazolino-pyrimidinone derivatives their preparation and appli cations
DE2557425A1 (de) * 1975-12-19 1977-06-30 Boehringer Sohn Ingelheim Chinazolonderivate
US4041163A (en) * 1976-03-29 1977-08-09 Pfizer Inc. N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents
US4168380A (en) * 1978-04-21 1979-09-18 Hoffmann-La Roche Inc. 7-Methoxy-5-oxo-5H-thiazolo[2,3-b]quinazoline-2-carboxylic acid
US4223031A (en) * 1978-05-05 1980-09-16 Mead Johnson & Company Azolopyrimidinones
IL59802A (en) * 1979-05-08 1983-07-31 Erba Farmitalia Substituted pyrido(1,2-a)pyrimidine carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
US4282360A (en) * 1979-10-12 1981-08-04 Hoffmann-La Roche Inc. 7-Methylthio or methylsulfinyl-5-oxo-5H-thiazolo[2,3-b]quinazoline-2-carboxylic acid
DK151811C (da) * 1979-11-23 1988-06-06 Pfizer Analogifremgangsmaade til fremstilling af n-(5-tetrazolyl)-1-oxo-1h-thiazolooe3,2-aaa-pyrimidin-2-carboxamider eller farmaceutisk acceptable kationsalte deraf samt 1-oxo-1h-thiazolooe3,2-aaapyrimidin-2-carboxylsyrer til anvendelse som udgangsmaterialer ved fremgangsmaaden
PL129612B1 (en) * 1980-07-24 1984-05-31 Rhone Poulenc Ind Process for preparing novel derivatives of 2,3,6,7-tetrahydrothiazole/3,2-a/pirymidin-5-one
US4340734A (en) * 1980-11-14 1982-07-20 American Cyanamid Company 3-(α-Substituted-benzyl)-2,3-dihydrothiazolo [3,2-a][1,3]diazacyclan-3-ol derivatives
US4443451A (en) * 1981-07-15 1984-04-17 Janssen Pharmaceutica N.V. Bicyclic pyrimidin-5-one derivatives
US4347248A (en) * 1981-03-23 1982-08-31 American Cyanamid Company 2,3-Disubstituted-thiazolo[3,2-a]pyrimidines
US4325955A (en) * 1981-03-23 1982-04-20 American Cyanamid Company Substituted 3-benzhydrylthiazolo(3,2-a)pyrimidines
NL8202706A (nl) * 1981-07-15 1983-02-01 Erba Farmitalia Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.
US4537962A (en) * 1982-02-04 1985-08-27 Farmitalia Carlo Erba, S.P.A. Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them

Also Published As

Publication number Publication date
FI77869B (fi) 1989-01-31
ES8505357A1 (es) 1985-05-16
FI840088A (fi) 1984-07-13
SE456996B (sv) 1988-11-21
NZ206816A (en) 1985-09-13
DK12084A (da) 1984-07-13
CS27984A2 (en) 1991-03-12
PT77946B (en) 1986-04-16
DK12084D0 (da) 1984-01-11
PH22448A (en) 1988-09-12
JPS59130891A (ja) 1984-07-27
AU2322184A (en) 1984-07-19
IT1185050B (it) 1987-11-04
GB8300728D0 (en) 1983-02-16
SU1355131A3 (ru) 1987-11-23
US4609660A (en) 1986-09-02
FI840088A0 (fi) 1984-01-11
SE8400118L (sv) 1984-07-13
CA1232604A (en) 1988-02-09
NO840092L (no) 1984-07-13
ATA8084A (de) 1988-02-15
AT386601B (de) 1988-09-26
ES528662A0 (es) 1985-05-16
BE898641A (fr) 1984-07-10
US4558046A (en) 1985-12-10
IT8419085A0 (it) 1984-01-10
AU568527B2 (en) 1988-01-07
HU190945B (en) 1986-12-28
DE3400733A1 (de) 1984-07-12
KR840007420A (ko) 1984-12-07
CH660011A5 (de) 1987-03-13
GR81735B (pt) 1984-12-12
SE8400118D0 (sv) 1984-01-11
FR2539131A1 (fr) 1984-07-13
FI77869C (fi) 1989-05-10
FR2539131B1 (fr) 1987-01-30
IL70651A0 (en) 1984-04-30
IL70651A (en) 1986-10-31
PT77946A (en) 1984-02-01
ZA84227B (en) 1984-08-29

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A85 Still pending on 85-01-01
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BA A request for search or an international-type search has been filed
BB A search report has been drawn up
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