MX342164B - Derivados de pirimidina fusionados novedosos para la inhibicion de la actividad de tirosina cinasa. - Google Patents

Derivados de pirimidina fusionados novedosos para la inhibicion de la actividad de tirosina cinasa.

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Publication number
MX342164B
MX342164B MX2014005025A MX2014005025A MX342164B MX 342164 B MX342164 B MX 342164B MX 2014005025 A MX2014005025 A MX 2014005025A MX 2014005025 A MX2014005025 A MX 2014005025A MX 342164 B MX342164 B MX 342164B
Authority
MX
Mexico
Prior art keywords
inhibition
tyrosine kinase
fused pyrimidine
kinase activity
novel fused
Prior art date
Application number
MX2014005025A
Other languages
English (en)
Inventor
Young Cha Mi
Jong Kang Seok
Ra Kim Mi
Yeon Lee Ju
Young Jeon Ji
Gi Jo Myoung
Joo Kwak Eun
Ok Lee Kwang
Hee Ha Tae
Hyun Suh Kwee
Sup Kim Maeng
Original Assignee
Hanmi Science Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45371929&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX342164(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hanmi Science Co Ltd filed Critical Hanmi Science Co Ltd
Publication of MX342164B publication Critical patent/MX342164B/es

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    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • C07D491/044Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

La presente invención se refiere a un derivado de pirimidina fusionada novedosa que tiene una actividad inhibidora de tirosinas cinasas, y una composición farmacéutica para prevenir o tratar cánceres, tumores, enfermedades inflamatorias, enfermedades autoinmunes, o enfermedades mediadas inmunológicamente que comprenden el mismo como un ingrediente activo.
MX2014005025A 2010-06-23 2011-06-20 Derivados de pirimidina fusionados novedosos para la inhibicion de la actividad de tirosina cinasa. MX342164B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR20100059686 2010-06-23
PCT/KR2011/004482 WO2011162515A2 (en) 2010-06-23 2011-06-20 Novel fused pyrimidine derivatives for inhd3ition of tyrosine kinase activity

Publications (1)

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MX342164B true MX342164B (es) 2016-09-19

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