KR920009279A - 광학 활성 피리도벤즈옥사진 유도체의 제조방법 - Google Patents

광학 활성 피리도벤즈옥사진 유도체의 제조방법

Info

Publication number
KR920009279A
KR920009279A KR1019900017517A KR900017517A KR920009279A KR 920009279 A KR920009279 A KR 920009279A KR 1019900017517 A KR1019900017517 A KR 1019900017517A KR 900017517 A KR900017517 A KR 900017517A KR 920009279 A KR920009279 A KR 920009279A
Authority
KR
South Korea
Prior art keywords
optically active
derivatives
preparing
pyridobenzoxazin
preparing optically
Prior art date
Application number
KR1019900017517A
Other languages
English (en)
Other versions
KR940003757B1 (ko
Inventor
이사오 하야가와
쇼오고 아다라시
슈이찌 요고하마
마사즈미 이마무라
가쯔이찌 사가노
노부유끼 히가시하시
마사유끼 오오시마
Original Assignee
다이이찌 세이야꾸 가부시끼가이샤
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27281433&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR920009279(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from JP60226499A external-priority patent/JPH0720946B2/ja
Application filed by 다이이찌 세이야꾸 가부시끼가이샤 filed Critical 다이이찌 세이야꾸 가부시끼가이샤
Priority to KR1019900017517A priority Critical patent/KR940003757B1/ko
Publication of KR920009279A publication Critical patent/KR920009279A/ko
Application granted granted Critical
Publication of KR940003757B1 publication Critical patent/KR940003757B1/ko

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR1019900017517A 1985-06-20 1990-10-31 광학 활성 피리도벤즈옥사진 유도체의 제조방법 KR940003757B1 (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019900017517A KR940003757B1 (ko) 1985-06-20 1990-10-31 광학 활성 피리도벤즈옥사진 유도체의 제조방법

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
JP134712/85 1985-06-20
JP13471285 1985-06-20
JP226499/85 1985-10-11
JP60226499A JPH0720946B2 (ja) 1985-10-11 1985-10-11 光学活性３−メチルベンゾオキサジン誘導体およびその製法
JP16496/86 1986-01-28
JP1649686 1986-01-28
KR1019860004934A KR920010048B1 (ko) 1985-06-20 1986-06-20 광학 활성 피리도벤즈옥사진 유도체 및 이의 중간체의 제조방법
KR1019900017517A KR940003757B1 (ko) 1985-06-20 1990-10-31 광학 활성 피리도벤즈옥사진 유도체의 제조방법

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1019860004934A Division KR920010048B1 (ko) 1985-06-20 1986-06-20 광학 활성 피리도벤즈옥사진 유도체 및 이의 중간체의 제조방법

Publications (2)

Publication Number Publication Date
KR920009279A true KR920009279A (ko) 1992-05-28
KR940003757B1 KR940003757B1 (ko) 1994-04-30

Family

ID=27281433

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1019860004934A KR920010048B1 (ko) 1985-06-20 1986-06-20 광학 활성 피리도벤즈옥사진 유도체 및 이의 중간체의 제조방법
KR1019900017517A KR940003757B1 (ko) 1985-06-20 1990-10-31 광학 활성 피리도벤즈옥사진 유도체의 제조방법

Family Applications Before (1)

Application Number Title Priority Date Filing Date
KR1019860004934A KR920010048B1 (ko) 1985-06-20 1986-06-20 광학 활성 피리도벤즈옥사진 유도체 및 이의 중간체의 제조방법

Country Status (16)

Country Link
US (3) US5053407A (ko)
EP (1) EP0206283B1 (ko)
KR (2) KR920010048B1 (ko)
AT (1) ATE85057T1 (ko)
BG (1) BG60527B2 (ko)
CA (1) CA1304080C (ko)
DE (2) DE3687599T2 (ko)
DK (1) DK170473B1 (ko)
ES (1) ES8801251A1 (ko)
FI (1) FI90241C (ko)
GR (1) GR861625B (ko)
HK (1) HK91793A (ko)
IE (1) IE59463B1 (ko)
NL (1) NL980016I2 (ko)
NO (1) NO166131C (ko)
YU (3) YU44918B (ko)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20010103346A (ko) * 2000-05-09 2001-11-23 이후근 패각 입자와 접착제 그리고 물감을 혼합하여 그림 밑칠용재료를 제조하는 방법

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EP0273399B1 (en) * 1986-12-25 1994-08-17 Daiichi Pharmaceutical Co., Ltd. Optically active 2,3-dihydrobenzoaxine derivatives and process for preparing the same
NO172846C (no) * 1987-12-25 1993-09-15 Daiichi Seiyaku Co Fremgangsmaate for fremstilling av 7,8-dihalogen-3-metyl-2,3-dihydro-2m-benzoksazinderivater og propoksybenzenderivater for utoevelse av fremgangsmaaten.
US5175160A (en) * 1988-08-09 1992-12-29 Daiichi Pharmaceutical Co., Ltd. Antimicrobial agent for animals
MY104139A (en) * 1988-08-09 1994-02-28 Daiichi Seiyaku Co Antimicrobial agent for animals
AU4376589A (en) * 1988-11-07 1990-05-10 Gist-Brocades N.V. Optically active benzoxazines and benzothiazines
FI94339C (fi) 1989-07-21 1995-08-25 Warner Lambert Co Menetelmä farmaseuttisesti käyttökelpoisen /R-(R*,R*)/-2-(4-fluorifenyyli)- , -dihydroksi-5-(1-metyylietyyli)-3-fenyyli-4-/(fenyyliamino)karbonyyli/-1H-pyrroli-1-heptaanihapon ja sen farmaseuttisesti hyväksyttävien suolojen valmistamiseksi
FR2655545B1 (fr) * 1989-12-11 1994-06-10 Rhone Poulenc Sante Nouvelle application therapeutique des derives des fluoroquinolones.
TW208013B (ko) * 1990-03-01 1993-06-21 Daiichi Co Ltd
NO179912C (no) * 1990-11-28 1997-01-08 Daiichi Seiyaku Co Analogifremgangsmåte for fremstilling av et terapeutisk virksomt optisk aktivt pyridobenzoksazinderivat
US5521310A (en) * 1992-10-07 1996-05-28 Derivados Del Etilo, S.A. Process to obtain benzoxazines to be used for the synthesis of ofloxazine, levofloxazine and derivatives
ES2055656B1 (es) * 1992-10-07 1995-11-16 Etilo Derivados Procedimiento para la obtencion de benzoxazinas utiles para sintesis de ofloxacina, levofloxacina y derivados.
US5532239A (en) * 1993-08-02 1996-07-02 Assistance Publique - Hopitaux De Paris Therapeutic application of fluoroquinolone derivatives
ZA946853B (en) * 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
US5686095A (en) * 1995-10-23 1997-11-11 Price, Jr.; Francis W. Method of treating canker sores
KR100491282B1 (ko) 1996-07-24 2005-05-24 워너-램버트 캄파니 엘엘씨 통증 치료용 이소부틸가바 및 그의 유도체
US6248343B1 (en) 1998-01-20 2001-06-19 Ethicon, Inc. Therapeutic antimicrobial compositions
US5972358A (en) * 1998-01-20 1999-10-26 Ethicon, Inc. Low tack lotion, gels and creams
US5997893A (en) * 1998-01-20 1999-12-07 Ethicon, Inc. Alcohol based anti-microbial compositions with cosmetic appearance
US6022551A (en) * 1998-01-20 2000-02-08 Ethicon, Inc. Antimicrobial composition
KR100309871B1 (ko) 1999-02-24 2001-10-29 윤종용 (-)피리도벤즈옥사진 카르복실산 유도체의 제조방법
JP2003527308A (ja) 1998-12-04 2003-09-16 インフラックス，インコーポレイテッド 多剤輸送体の阻害剤
KR100617952B1 (ko) * 1999-03-04 2006-08-30 보령제약 주식회사 광학활성 피리도 벤즈옥사진 유도체의 제조방법
EP2360160B1 (en) * 1999-09-08 2013-07-24 Daiichi Sankyo Company, Limited Intermediates and their use for producing benzoxazine derivative
ATE319710T1 (de) 2000-12-21 2006-03-15 Pharmacia & Upjohn Co Llc Antimikrobielle chinolonderivate und ihre verwendung zur behandlung bakterieller infektionen
ES2329554T3 (es) 2001-03-07 2009-11-27 Daiichi Sankyo Company, Limited Procesos para producir derivados de propoxianilina opticamente activos.
KR100444248B1 (ko) 2001-04-27 2004-08-16 한국산업기술평가원 열간가공성이 우수한 고망간 듀플렉스 스텐레스강과 그제조방법
WO2003028665A2 (en) 2001-10-03 2003-04-10 Teva Pharmaceutical Industries Ltd. Methods for the purification of levofloxacin
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AU2002365416A1 (en) * 2001-11-29 2003-06-10 Teva Pharmaceutical Industries Ltd. Methods for the purification of levofloxacin
EP2172192A1 (en) * 2001-12-24 2010-04-07 Teva Pharmaceutical Industries Ltd. Dosage form with a core tablet of active ingredient sheathed in a compressed annular body of powder of granular material, and process and tooling for producing it
US20040052843A1 (en) * 2001-12-24 2004-03-18 Lerner E. Itzhak Controlled release dosage forms
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FR2859471B1 (fr) 2003-09-09 2006-02-03 Solvay Procede pour la fabrication d'un compose enantiopur
EP1852431A4 (en) 2005-02-07 2009-11-04 Mitsubishi Tanabe Pharma Corp OPTICALLY ACTIVE TETRAHYDRONAPHTALENE DERIVATIVE
US8546423B2 (en) 2005-05-18 2013-10-01 Mpex Pharmaceuticals, Inc. Aerosolized fluoroquinolones and uses thereof
US7838532B2 (en) * 2005-05-18 2010-11-23 Mpex Pharmaceuticals, Inc. Aerosolized fluoroquinolones and uses thereof
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US7964723B2 (en) 2008-08-02 2011-06-21 Apeloa-Kangyu And practical process for exclusively producing (S)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido-[1,2,3,de][1,4]benzoxazine-6-carboxylic acid hemihydrate
NO2344129T3 (ko) 2008-10-07 2018-07-21
PT2346509T (pt) 2008-10-07 2020-08-05 Horizon Orphan Llc Inalação de levofloxacina para redução da inflamação pulmonar
AU2010247141A1 (en) 2009-05-15 2011-12-15 Redx Pharma Plc Redox drug derivatives
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CN101659669B (zh) * 2009-09-04 2011-07-20 诚达药业股份有限公司 左旋氧氟沙星的制备方法
CN102775424A (zh) * 2012-07-09 2012-11-14 浙江司太立制药股份有限公司 一种左氧氟沙星杂质的制备方法
CN106413713B (zh) * 2014-05-09 2020-07-14 特克尼梅德医疗技术股份公司 用作药物的吡吲哚对映异构体的药学上可接受的盐
CN105037388A (zh) * 2015-08-28 2015-11-11 安徽环球药业股份有限公司 一种安妥沙星的制备方法
CN105367585B (zh) * 2015-12-02 2017-11-17 山东齐都药业有限公司 左氧氟沙星杂质的制备方法
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20010103346A (ko) * 2000-05-09 2001-11-23 이후근 패각 입자와 접착제 그리고 물감을 혼합하여 그림 밑칠용재료를 제조하는 방법

Also Published As

Publication number Publication date
ATE85057T1 (de) 1993-02-15
NO862426D0 (no) 1986-06-18
NO862426L (no) 1986-12-22
EP0206283A3 (en) 1988-08-10
ES556292A0 (es) 1988-01-01
ES8801251A1 (es) 1988-01-01
DE19875012I2 (de) 2006-06-29
CA1304080C (en) 1992-06-23
YU45512B (en) 1992-05-28
NO166131C (no) 1991-06-05
IE861631L (en) 1986-12-20
YU209889A (en) 1990-04-30
YU107386A (en) 1988-02-29
DE3687599T2 (de) 1993-05-19
NL980016I1 (nl) 1998-07-01
NO166131B (no) 1991-02-25
KR940003757B1 (ko) 1994-04-30
YU186788A (en) 1989-04-30
FI862643A0 (fi) 1986-06-19
US4985557A (en) 1991-01-15
IE59463B1 (en) 1994-02-23
US5142046A (en) 1992-08-25
KR920010048B1 (ko) 1992-11-13
FI90241C (fi) 1994-01-10
DK285086D0 (da) 1986-06-18
YU45524B (en) 1992-05-28
EP0206283A2 (en) 1986-12-30
DK170473B1 (da) 1995-09-11
DE3687599D1 (de) 1993-03-11
BG60527B2 (bg) 1995-07-28
KR870000340A (ko) 1987-02-17
FI862643A (fi) 1986-12-21
FI90241B (fi) 1993-09-30
YU44918B (en) 1991-04-30
NL980016I2 (nl) 1998-08-03
GR861625B (en) 1986-10-21
US5053407A (en) 1991-10-01
EP0206283B1 (en) 1993-01-27
HK91793A (en) 1993-09-10
DK285086A (da) 1986-12-21

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