ES2001794A6 - Un procedimiento para la preparacion de derivados de quinolina - Google Patents
Un procedimiento para la preparacion de derivados de quinolinaInfo
- Publication number
- ES2001794A6 ES2001794A6 ES8602086A ES8602086A ES2001794A6 ES 2001794 A6 ES2001794 A6 ES 2001794A6 ES 8602086 A ES8602086 A ES 8602086A ES 8602086 A ES8602086 A ES 8602086A ES 2001794 A6 ES2001794 A6 ES 2001794A6
- Authority
- ES
- Spain
- Prior art keywords
- quinoline derivatives
- iii
- compounds
- formula
- salts
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Treatment And Processing Of Natural Fur Or Leather (AREA)
- Polyurethanes Or Polyureas (AREA)
- Detergent Compositions (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
SE DESCRIBE UN PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE QUINOLINA DE LA FORMULA (I) Y QUE PUEDE UTILIZARSE EN LA TERAPIA Y PROFILAXIS DE ENFERMEDADES, ESPECIALMENTE EN INFECCIONES BACTERIANAS. EL PROCEDIMIENTO SE CARACTERIZA PORQUE LOS COMPUESTOS DE FORMULA (I) PUEDEN PREPARARSE POR VARIOS PROCEDIMIENTOS, CITANDO ENTRE ELLOS EL DE LA SAPONIFICACION DE UN ESTER DE ALQUILO INFERIOR CORRESPONDIENTE AL ACIDO DE LA FORMULA (I) HACIENDO REACCIONAR CON UNA BASE INORGANICA, EN PRESENCIA DE UN ALCANOL INFERIOR, MIENTRAS SE CALIENTA A LA TEMPERATURA DE REFLUJO. SI SE DESEA, EL ACIDO OBTENIDO PUEDE AISLARSE EN FORMA DE UNA SAL.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH412085 | 1985-09-24 | ||
CH317786 | 1986-08-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2001794A6 true ES2001794A6 (es) | 1988-06-16 |
Family
ID=25692381
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES8602086A Expired ES2001794A6 (es) | 1985-09-24 | 1986-09-23 | Un procedimiento para la preparacion de derivados de quinolina |
Country Status (16)
Country | Link |
---|---|
US (3) | US4806541A (es) |
EP (1) | EP0216345B1 (es) |
CN (1) | CN1013865B (es) |
AT (1) | ATE72668T1 (es) |
AU (1) | AU603549B2 (es) |
DE (1) | DE3683922D1 (es) |
DK (1) | DK454086A (es) |
ES (1) | ES2001794A6 (es) |
FI (1) | FI863836A (es) |
HU (1) | HU196411B (es) |
IL (1) | IL80114A0 (es) |
MC (1) | MC1772A1 (es) |
NO (1) | NO863790L (es) |
NZ (1) | NZ217650A (es) |
PH (1) | PH24627A (es) |
PT (1) | PT83423B (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5153204A (en) * | 1986-03-01 | 1992-10-06 | Bayer Aktiengesellschaft | 7-(1-Pyrrolidinyl)-quinolonecarboxylic acid derivatives |
US5147871A (en) * | 1986-07-03 | 1992-09-15 | Hoffmann La-Roche, Inc. | Anti-bacterial cephalosporin compounds |
CS273349B2 (en) * | 1988-03-31 | 1991-03-12 | Hoffmann La Roche | Method of cephalosporin's new derivatives production |
US5336768A (en) * | 1988-05-24 | 1994-08-09 | Hoffmann-La Roche Inc. | Antibacterial cephalosporin compounds |
CA2001203C (en) * | 1988-10-24 | 2001-02-13 | Thomas P. Demuth, Jr. | Novel antimicrobial dithiocarbamoyl quinolones |
EP0366189A3 (en) * | 1988-10-24 | 1992-01-02 | Norwich Eaton Pharmaceuticals, Inc. | Novel antimicrobial lactam-quinolones |
US5162523A (en) * | 1989-07-21 | 1992-11-10 | Hoffmann-La Roche Inc. | Cephalosporin antibacterial compounds |
US5159077A (en) * | 1989-07-21 | 1992-10-27 | Hoffmann-La Roche Inc. | Penam antibacterial compounds |
AR054608A1 (es) * | 2005-08-08 | 2007-06-27 | Actelion Pharmaceuticals Ltd | Derivados de oxazolidinona enlazados a quinolonas como antibacterianos |
US8124623B2 (en) * | 2006-11-10 | 2012-02-28 | Actelion Pharmaceuticals Ltd. | 5-hydroxymethyl-oxazolidin-2-one-derivatives and their uses as antibacterials |
CL2007003332A1 (es) * | 2006-11-24 | 2008-06-20 | Actelion Pharmaceuticals Ltd | Compuestos derivados de heterociclos condensados; compuestos intermediarios; composicion farmaceutica; y uso en la prevencion o tratamiento de infecciones bacterianas. |
WO2008131415A1 (en) * | 2007-04-23 | 2008-10-30 | Achillion Pharmaceuticals, Inc. | 4-substituted-1h-isothiazolo[5,4-b][1,4]oxazino[2,3,4-ij]quinoline-7,8(2h,9h)-diones and related compounds as anti-infective agents |
EP2250171A2 (en) * | 2008-02-12 | 2010-11-17 | Achaogen, Inc. | Antibacterial fluoroquinolone analogs |
WO2011031740A1 (en) * | 2009-09-09 | 2011-03-17 | Achaogen, Inc. | Antibacterial fluoroquinolone analogs |
WO2011031744A1 (en) * | 2009-09-09 | 2011-03-17 | Achaogen, Inc. | Antibacterial fluoroquinolone analogs |
WO2011031745A1 (en) * | 2009-09-09 | 2011-03-17 | Achaogen, Inc. | Antibacterial fluoroquinolone analogs |
WO2011031743A1 (en) * | 2009-09-09 | 2011-03-17 | Achaogen, Inc. | Antibacterial fluoroquinolone analogs |
US10087171B2 (en) | 2016-12-19 | 2018-10-02 | Actelion Pharmaceuticals Ltd | Crystalline forms of cadazolid |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5270014A (en) * | 1975-12-05 | 1977-06-10 | Senju Pharma Co | Stabilization of pyrido*3*22a*phenoxadine compounds |
DE3306772A1 (de) * | 1983-02-25 | 1984-08-30 | Bayer Ag, 5090 Leverkusen | Chinolonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
DE3308909A1 (de) * | 1983-03-12 | 1984-09-13 | Bayer Ag, 5090 Leverkusen | Bakterizide mittel auf chinoloncarbonsaeure-basis |
AU553415B2 (en) * | 1983-09-19 | 1986-07-17 | Abbott Japan Co., Ltd. | 6-fluoro-1-4-dihydro-4-oxo-7-substituted piperazinyl- quinoline-3-carboxylic acids |
DE3409922A1 (de) * | 1984-03-17 | 1985-09-26 | Bayer Ag, 5090 Leverkusen | 1,7-diamino-1,4-dihydro-4-oxo-3-(aza)chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie ihre verwendung bei der bekaempfung bakterieller erkrankungen |
DE3420798A1 (de) * | 1984-06-04 | 1985-12-05 | Bayer Ag, 5090 Leverkusen | 7-(3-aryl-l-piperazinyl)- sowie 7-(3-cyclohexyl-l-piperazinyl)-3-chinoloncarbonsaeuren |
US4689325A (en) * | 1985-12-23 | 1987-08-25 | Abbott Laboratories | Isoxazolo-pyrido-phenoxazine and isothiazolo-pyrido-phenoxazine derivatives |
-
1986
- 1986-09-22 DE DE8686113036T patent/DE3683922D1/de not_active Expired - Fee Related
- 1986-09-22 HU HU864007A patent/HU196411B/hu unknown
- 1986-09-22 AT AT86113036T patent/ATE72668T1/de not_active IP Right Cessation
- 1986-09-22 US US06/910,566 patent/US4806541A/en not_active Expired - Fee Related
- 1986-09-22 NZ NZ217650A patent/NZ217650A/xx unknown
- 1986-09-22 IL IL80114A patent/IL80114A0/xx unknown
- 1986-09-22 EP EP86113036A patent/EP0216345B1/de not_active Expired - Lifetime
- 1986-09-23 FI FI863836A patent/FI863836A/fi not_active IP Right Cessation
- 1986-09-23 AU AU63075/86A patent/AU603549B2/en not_active Ceased
- 1986-09-23 DK DK454086A patent/DK454086A/da not_active Application Discontinuation
- 1986-09-23 CN CN86106372A patent/CN1013865B/zh not_active Expired
- 1986-09-23 NO NO863790A patent/NO863790L/no unknown
- 1986-09-23 MC MC861850A patent/MC1772A1/xx unknown
- 1986-09-23 PH PH34279A patent/PH24627A/en unknown
- 1986-09-23 PT PT83423A patent/PT83423B/pt unknown
- 1986-09-23 ES ES8602086A patent/ES2001794A6/es not_active Expired
-
1988
- 1988-11-21 US US07/274,162 patent/US4946847A/en not_active Expired - Fee Related
-
1990
- 1990-06-15 US US07/524,196 patent/US4977265A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP0216345A2 (de) | 1987-04-01 |
HU196411B (en) | 1988-11-28 |
US4977265A (en) | 1990-12-11 |
DE3683922D1 (de) | 1992-03-26 |
PT83423A (en) | 1986-10-01 |
US4806541A (en) | 1989-02-21 |
FI863836A (fi) | 1987-03-25 |
HUT45538A (en) | 1988-07-28 |
EP0216345A3 (en) | 1988-07-06 |
EP0216345B1 (de) | 1992-02-19 |
MC1772A1 (fr) | 1987-07-17 |
NO863790L (no) | 1987-03-25 |
FI863836A0 (fi) | 1986-09-23 |
CN86106372A (zh) | 1987-03-18 |
DK454086A (da) | 1987-03-25 |
AU6307586A (en) | 1987-03-26 |
NO863790D0 (no) | 1986-09-23 |
ATE72668T1 (de) | 1992-03-15 |
DK454086D0 (da) | 1986-09-23 |
PH24627A (en) | 1990-08-17 |
NZ217650A (en) | 1989-09-27 |
AU603549B2 (en) | 1990-11-22 |
US4946847A (en) | 1990-08-07 |
CN1013865B (zh) | 1991-09-11 |
IL80114A0 (en) | 1986-12-31 |
PT83423B (en) | 1988-10-24 |
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