KR850000969B1 - 안드로스탄 카보티오에이트의 제조방법 - Google Patents
안드로스탄 카보티오에이트의 제조방법 Download PDFInfo
- Publication number
- KR850000969B1 KR850000969B1 KR1019810000442A KR810000442A KR850000969B1 KR 850000969 B1 KR850000969 B1 KR 850000969B1 KR 1019810000442 A KR1019810000442 A KR 1019810000442A KR 810000442 A KR810000442 A KR 810000442A KR 850000969 B1 KR850000969 B1 KR 850000969B1
- Authority
- KR
- South Korea
- Prior art keywords
- hydroxy
- diene
- solution
- methyl
- ethyl acetate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 0 CCCCC(C=C(C1)[C@@]2(*)*C11C(*)CC3(C)C(*)(*)C(*)CC3C1C2)O Chemical compound CCCCC(C=C(C1)[C@@]2(*)*C11C(*)CC3(C)C(*)(*)C(*)CC3C1C2)O 0.000 description 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/0026—Oxygen-containing hetero ring cyclic ketals
- C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
- C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0038—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 with an androstane skeleton, including 18- or 19-substituted derivatives, 18-nor derivatives and also derivatives where position 17-beta is substituted by a carbon atom not directly bonded to a further carbon atom and not being part of an amide group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
- C07J71/0015—Oxiranes at position 9(11)
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8005174 | 1980-02-15 | ||
| GB8005174 | 1980-02-15 | ||
| GB8013339 | 1980-04-23 | ||
| GB8013339 | 1981-04-23 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR830005262A KR830005262A (ko) | 1983-08-03 |
| KR850000969B1 true KR850000969B1 (ko) | 1985-07-02 |
Family
ID=26274505
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019810000442A Expired KR850000969B1 (ko) | 1980-02-15 | 1981-02-13 | 안드로스탄 카보티오에이트의 제조방법 |
Country Status (23)
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA817929B (en) * | 1980-12-22 | 1982-10-27 | Upjohn Co | 5alpha-and 5beta-androstane-17beta-carboxylates |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1436549A (en) * | 1972-06-15 | 1976-05-19 | Glaxo Lab Ltd | 17beta-mercaptocarbonyl-3alpha-hydroxy-steroids and their esters |
| GB1438940A (en) * | 1972-07-19 | 1976-06-09 | Glaxo Lab Ltd | 17beta-haloalkoxycarbonyl-17alpha-oxysteroids |
| GB1514476A (en) * | 1974-08-30 | 1978-06-14 | Glaxo Lab Ltd | Alkyl and haloalkyl androst-4-ene and androsta-1,4-diene-17beta-carboxylates |
| US4188385A (en) * | 1978-04-05 | 1980-02-12 | Syntex (U.S.A.) Inc. | Thioetianic acid derivatives |
| GB1580517A (en) * | 1978-04-06 | 1980-12-03 | Fowler I | Crutches |
-
1981
- 1981-02-13 KR KR1019810000442A patent/KR850000969B1/ko not_active Expired
- 1981-02-13 ES ES499394A patent/ES499394A0/es active Granted
- 1981-02-13 AT AT0067481A patent/AT395427B/de not_active IP Right Cessation
- 1981-02-13 AU AU67298/81A patent/AU544517B2/en not_active Expired
- 1981-02-13 NL NL8100707A patent/NL191792C/xx not_active IP Right Cessation
- 1981-02-13 FI FI810444A patent/FI70904C/fi not_active IP Right Cessation
- 1981-02-13 CH CH3890/84A patent/CH651307A5/de not_active IP Right Cessation
- 1981-02-13 DE DE3153379A patent/DE3153379C2/de not_active Expired - Lifetime
- 1981-02-13 IE IE282/81A patent/IE51394B1/en active Protection Beyond IP Right Term
- 1981-02-13 CH CH98281A patent/CH644615A5/de not_active IP Right Cessation
- 1981-02-13 DE DE19813105307 patent/DE3105307A1/de active Granted
- 1981-02-13 IT IT47792/81A patent/IT1170717B/it active Protection Beyond IP Right Term
- 1981-02-13 FR FR8102818A patent/FR2477156A1/fr active Granted
- 1981-02-13 SE SE8101010A patent/SE452468B/sv not_active IP Right Cessation
- 1981-02-13 NZ NZ196260A patent/NZ196260A/xx unknown
- 1981-02-13 PT PT72502A patent/PT72502B/pt unknown
- 1981-02-13 DK DK62381A patent/DK147022C/da not_active IP Right Cessation
- 1981-08-17 FR FR8115812A patent/FR2485542A1/fr active Granted
-
1982
- 1982-02-12 ES ES509539A patent/ES8305379A1/es not_active Expired
- 1982-12-14 ES ES518161A patent/ES8402317A1/es not_active Expired
-
1983
- 1983-08-16 ES ES524985A patent/ES524985A0/es active Granted
-
1984
- 1984-04-30 ES ES532055A patent/ES532055A0/es active Granted
-
1985
- 1985-05-13 KE KE3526A patent/KE3526A/xx unknown
- 1985-05-16 SG SG368/85A patent/SG36885G/en unknown
- 1985-08-08 HK HK583/85A patent/HK58385A/xx not_active IP Right Cessation
- 1985-12-30 MY MY757/85A patent/MY8500757A/xx unknown
-
1991
- 1991-12-23 CZ CS914034A patent/CZ281275B6/cs unknown
- 1991-12-23 SK SK4034-91A patent/SK403491A3/sk unknown
-
1992
- 1992-06-05 MX MX9202717A patent/MX9202717A/es unknown
-
1993
- 1993-08-20 BG BG098060A patent/BG60700B2/bg unknown
-
1996
- 1996-10-29 NL NL960029C patent/NL960029I2/nl unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CA1201114A (en) | Androstane carbothioates | |
| US4377575A (en) | Corticoid-17-(alkyl carbonates) and process for their manufacture | |
| GB2088877A (en) | Androstane 17 beta carbothioates | |
| FI78111B (fi) | Foerfarande foer framstaellning av terapeutiskt aktiva 3,20-dioxo-1,4-pregnadien-17 -ol 17-aromatisk- heterocykliska karboxylater. | |
| EP0004773B1 (en) | 17-beta-thiocarboxylic acid esters of 4-halo-3-oxoandrost-4-enes, their pharmaceutical use and processes for their preparation | |
| US4187301A (en) | 17 Beta-thiocarboxylic acid esters of 6 alpha, 6 beta-difluoro-3-oxoandrost-4-enes | |
| DK147735B (da) | Analogifremgangsmaade til fremstilling af 3-oxo-androst-4-en-17beta-thiocarboxylsyreestere | |
| KR100290225B1 (ko) | △ 9,11 스테로이드의 레지오 선택적 제조방법 | |
| US4650610A (en) | Androstane carbothioic acids | |
| JP3346873B2 (ja) | ６α，９α−二弗素化ステロイドの新製造法及び新規な中間体 | |
| KR850000969B1 (ko) | 안드로스탄 카보티오에이트의 제조방법 | |
| EP0097328B1 (en) | Process for preparation of steroids | |
| JP3037508B2 (ja) | プレグナ−１，４−ジエン−３，２０−ジオンの新規な置換された１６−メチルステロイド誘導体、それらの製造法、それらの１６−メチレンステロイドの製造への用途及び新規な中間体 | |
| JP2005530679A (ja) | ６α−フルオロコルチコステロイドの調製方法 | |
| DK146017B (da) | Analogifremgangsmaade til fremstilling af 17alfa-acyloxy-9alfa,21-dihalogen-11beta-hydroxy-6alfa-fluor-16beta-methyl-pregna-1,4-dien-3,20-dion-forbindelser | |
| GB2137206A (en) | Androstane 17-carbothioc acid derivatives | |
| US4427592A (en) | Androstene-17-dithioketals | |
| GB2079754A (en) | Production of 16-methyl-17 -acyloxy corticoids by selective solvolysis of 11-trihaloacetoxy and 21-acyloxy groups | |
| JPS632280B2 (enrdf_load_stackoverflow) | ||
| IE51395B1 (en) | Steroids of the androstane series | |
| KR830000084B1 (ko) | 코르티코이드-17-(알킬 카보네이트)의 제조방법 | |
| US3980680A (en) | Process for the preparation of 21-desoxy-17-acyloxy-4-pregnenes and of 21-iodo-21-desoxy-17-acyl oxy-4-pregnene intermediates useful therein | |
| US3814751A (en) | Process for preparing 6,6-difluoro-17alpha,21-dihydroxy 16alpha-methyl-4-pregnene-3,20-dione | |
| NO132189B (enrdf_load_stackoverflow) | ||
| NO791144L (no) | 4-halogenetansyre og derivater derav, samt fremgangsmaate til deres fremstilling |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0109 | Patent application |
Patent event code: PA01091R01D Comment text: Patent Application Patent event date: 19810213 |
|
| PG1501 | Laying open of application | ||
| PE0902 | Notice of grounds for rejection |
Comment text: Notification of reason for refusal Patent event date: 19850130 Patent event code: PE09021S01D |
|
| PG1605 | Publication of application before grant of patent |
Comment text: Decision on Publication of Application Patent event code: PG16051S01I Patent event date: 19850605 |
|
| PE0701 | Decision of registration |
Patent event code: PE07011S01D Comment text: Decision to Grant Registration Patent event date: 19850923 |
|
| PR0701 | Registration of establishment |
Comment text: Registration of Establishment Patent event date: 19851011 Patent event code: PR07011E01D |
|
| PR1002 | Payment of registration fee |
Payment date: 19851011 End annual number: 3 Start annual number: 1 |
|
| PR1001 | Payment of annual fee |
Payment date: 19880624 Start annual number: 4 End annual number: 4 |
|
| PR1001 | Payment of annual fee |
Payment date: 19890628 Start annual number: 5 End annual number: 5 |
|
| PR1001 | Payment of annual fee |
Payment date: 19900622 Start annual number: 6 End annual number: 6 |
|
| PR1001 | Payment of annual fee |
Payment date: 19910619 Start annual number: 7 End annual number: 7 |
|
| PR1001 | Payment of annual fee |
Payment date: 19920617 Start annual number: 8 End annual number: 8 |
|
| PR1001 | Payment of annual fee |
Payment date: 19930622 Start annual number: 9 End annual number: 9 |
|
| PR1001 | Payment of annual fee |
Payment date: 19940621 Start annual number: 10 End annual number: 10 |
|
| PR1001 | Payment of annual fee |
Payment date: 19950623 Start annual number: 11 End annual number: 11 |
|
| PC1801 | Expiration of term |