KR20150119848A - 친수성 자기-희생 링커 및 그것의 포합체 - Google Patents

친수성 자기-희생 링커 및 그것의 포합체 Download PDF

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KR20150119848A
KR20150119848A KR1020157019681A KR20157019681A KR20150119848A KR 20150119848 A KR20150119848 A KR 20150119848A KR 1020157019681 A KR1020157019681 A KR 1020157019681A KR 20157019681 A KR20157019681 A KR 20157019681A KR 20150119848 A KR20150119848 A KR 20150119848A
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linker
self
compound
bond
formula
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Korean (ko)
Inventor
롱-화 린
쉬-야오 린
유-차이 흐시에
치우-첸 후앙
Original Assignee
바이오얼라이언스 씨.브이.
어브게노믹스 인터내셔널 인코포레이티드
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Application filed by 바이오얼라이언스 씨.브이., 어브게노믹스 인터내셔널 인코포레이티드 filed Critical 바이오얼라이언스 씨.브이.
Priority to KR1020217034685A priority Critical patent/KR20210132742A/ko
Publication of KR20150119848A publication Critical patent/KR20150119848A/ko
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    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
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KR1020157019681A 2012-12-21 2013-12-20 친수성 자기-희생 링커 및 그것의 포합체 Abandoned KR20150119848A (ko)

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Application Number Priority Date Filing Date Title
KR1020217034685A KR20210132742A (ko) 2012-12-21 2013-12-20 친수성 자기-희생 링커 및 그것의 포합체

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US201261745448P 2012-12-21 2012-12-21
US61/745,448 2012-12-21
US201361785027P 2013-03-14 2013-03-14
US61/785,027 2013-03-14
PCT/US2013/077306 WO2014100762A1 (en) 2012-12-21 2013-12-20 Hydrophilic self-immolative linkers and conjugates thereof

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