KR102329186B1 - 페남을 제조하기 위한 방법 - Google Patents

페남을 제조하기 위한 방법 Download PDF

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KR102329186B1
KR102329186B1 KR1020167032608A KR20167032608A KR102329186B1 KR 102329186 B1 KR102329186 B1 KR 102329186B1 KR 1020167032608 A KR1020167032608 A KR 1020167032608A KR 20167032608 A KR20167032608 A KR 20167032608A KR 102329186 B1 KR102329186 B1 KR 102329186B1
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KR20170002466A (ko
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안드레아 파이니
마르코 포르자띠
지오반니 포그리아토
스테파노 비온디
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알레크라 테라퓨틱스 에스에이에스
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/18Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1896Compounds having one or more Si-O-acyl linkages
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/87Compounds being unsubstituted in position 3 or with substituents other than only two methyl radicals attached in position 3, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Feed For Specific Animals (AREA)
KR1020167032608A 2014-05-15 2015-05-14 페남을 제조하기 위한 방법 Active KR102329186B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB1408649.0 2014-05-15
GBGB1408649.0A GB201408649D0 (en) 2014-05-15 2014-05-15 Method
PCT/EP2015/060733 WO2015173378A2 (en) 2014-05-15 2015-05-14 Method

Publications (2)

Publication Number Publication Date
KR20170002466A KR20170002466A (ko) 2017-01-06
KR102329186B1 true KR102329186B1 (ko) 2021-11-22

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KR1020167032608A Active KR102329186B1 (ko) 2014-05-15 2015-05-14 페남을 제조하기 위한 방법

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US (1) US9963465B2 (enExample)
EP (3) EP3143028B1 (enExample)
JP (1) JP6613303B2 (enExample)
KR (1) KR102329186B1 (enExample)
CN (1) CN106459086B (enExample)
AU (1) AU2015261416B2 (enExample)
BR (1) BR112016026074B1 (enExample)
CA (1) CA2945900C (enExample)
CL (2) CL2016002880A1 (enExample)
CR (1) CR20160580A (enExample)
CY (2) CY1120957T1 (enExample)
DK (2) DK3143028T3 (enExample)
EA (2) EA033494B1 (enExample)
EC (1) ECSP16085143A (enExample)
ES (2) ES2699644T3 (enExample)
GB (1) GB201408649D0 (enExample)
HR (2) HRP20182065T1 (enExample)
HU (1) HUE044511T2 (enExample)
IL (1) IL248834B (enExample)
LT (2) LT3143028T (enExample)
MX (1) MX378875B (enExample)
PE (1) PE20161433A1 (enExample)
PL (2) PL3231806T3 (enExample)
PT (2) PT3143028T (enExample)
RS (2) RS58748B1 (enExample)
SG (1) SG11201609494YA (enExample)
SI (2) SI3231806T1 (enExample)
TR (1) TR201906867T4 (enExample)
WO (1) WO2015173378A2 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201319776D0 (en) * 2013-11-08 2013-12-25 Allecra Therapeutics Sas Compound

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080015156A1 (en) 2006-07-12 2008-01-17 Orchid Chemicals & Pharmaceuticals Ltd. Novel 2-substituted methyl penam derivatives
JP2014504279A (ja) 2010-11-25 2014-02-20 アレクラ セラピューティクス ゲーエムベーハー 化合物及びその使用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1319776A (en) 1969-07-15 1973-06-06 Yorkshire Chemicals Ltd Basic dyes
KR20120067257A (ko) * 2010-12-15 2012-06-25 서강대학교산학협력단 3-메틸-1,4-치환된 1,2,3-트라이아졸륨 기반의 이온성 액체 및 그의 제조방법과 응용

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080015156A1 (en) 2006-07-12 2008-01-17 Orchid Chemicals & Pharmaceuticals Ltd. Novel 2-substituted methyl penam derivatives
JP2014504279A (ja) 2010-11-25 2014-02-20 アレクラ セラピューティクス ゲーエムベーハー 化合物及びその使用

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Publication number Publication date
TR201906867T4 (tr) 2019-05-21
BR112016026074B1 (pt) 2023-01-03
EP3231806B1 (en) 2019-02-13
IL248834A0 (en) 2017-01-31
US9963465B2 (en) 2018-05-08
EP3231806A1 (en) 2017-10-18
DK3143028T3 (da) 2019-01-02
EA201991629A3 (ru) 2020-02-28
CR20160580A (es) 2017-05-09
EP3143028A2 (en) 2017-03-22
EA201692306A1 (ru) 2017-05-31
PL3231806T3 (pl) 2019-08-30
MX2016014644A (es) 2017-02-23
AU2015261416B2 (en) 2019-07-11
CL2016002880A1 (es) 2017-06-16
SI3231806T1 (sl) 2019-06-28
PT3143028T (pt) 2018-12-17
CA2945900C (en) 2023-01-24
EA201991629A2 (ru) 2019-12-30
KR20170002466A (ko) 2017-01-06
MX378875B (es) 2025-03-11
NZ725121A (en) 2023-09-29
SI3143028T1 (sl) 2019-01-31
RS58748B1 (sr) 2019-06-28
ES2699644T3 (es) 2019-02-12
LT3143028T (lt) 2018-12-27
CN106459086B (zh) 2018-11-13
CN106459086A (zh) 2017-02-22
WO2015173378A2 (en) 2015-11-19
JP6613303B2 (ja) 2019-11-27
EP3143028B1 (en) 2018-09-26
SG11201609494YA (en) 2016-12-29
ES2725675T3 (es) 2019-09-26
LT3231806T (lt) 2019-05-27
AU2015261416A1 (en) 2016-11-10
CY1121756T1 (el) 2020-07-31
HRP20182065T1 (hr) 2019-02-08
CA2945900A1 (en) 2015-11-19
DK3231806T3 (da) 2019-05-20
WO2015173378A3 (en) 2016-01-14
HRP20190830T1 (hr) 2019-06-28
US20170101421A1 (en) 2017-04-13
IL248834B (en) 2019-05-30
BR112016026074A8 (pt) 2021-03-30
PT3231806T (pt) 2019-05-30
EA033494B1 (ru) 2019-10-31
EP3441395A1 (en) 2019-02-13
RS58430B1 (sr) 2019-04-30
CY1120957T1 (el) 2019-12-11
CL2018001961A1 (es) 2018-08-31
JP2017515907A (ja) 2017-06-15
PE20161433A1 (es) 2017-01-18
GB201408649D0 (en) 2014-07-02
ECSP16085143A (es) 2017-05-31
PL3143028T3 (pl) 2019-04-30
HUE044511T2 (hu) 2019-10-28

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